Search Results - "Block MH"

Transcriptome-Derived Amplicon Sequencing Markers Elucidate the U.S. Podosphaera macularis Population Structure Across Feral and Commercial Plantings of Humulus lupulus.

Authors: Weldon WA Knaus BJ Grünwald NJ et al.

Source: Phytopathology [Phytopathology] 2021 Jan; Vol. 111 (1), pp. 194-203. Date of Electronic Publication: 2020 Dec 01.

Publication Type: Journal Article

Journal Info: Publisher: American Phytopathological Society] Country of Publication: United States NLM ID: 9427222 Publication Model: Print-Electronic Cited Medium: Print ISSN: 0031-949X (Print) Linking ISSN: 0031949X NLM ISO Abbreviation: Phytopathology Subsets: MEDLINE

Selective antagonism of the NPY Y5 receptor does not have a major effect on feeding in rats.

Authors: Turnbull AV Ellershaw L Masters DJ et al.

Source: Diabetes [Diabetes] 2002 Aug; Vol. 51 (8), pp. 2441-9.

Publication Type: Journal Article

Journal Info: Publisher: American Diabetes Association Country of Publication: United States NLM ID: 0372763 Publication Model: Print Cited Medium: Print ISSN: 0012-1797 (Print) Linking ISSN: 00121797 NLM ISO Abbreviation: Diabetes Subsets: MEDLINE

Discovery of 2,6-disubstituted pyrazine derivatives as inhibitors of CK2 and PIM kinases.

Authors: Gingipalli L Block MH Bao L et al.

Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2018 May 01; Vol. 28 (8), pp. 1336-1341. Date of Electronic Publication: 2018 Mar 07.

Publication Type: Journal Article

Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE

Discovery of potent KIFC1 inhibitors using a method of integrated high-throughput synthesis and screening.

Authors: Yang B Lamb ML Zhang T et al.

Source: Journal of medicinal chemistry [J Med Chem] 2014 Dec 11; Vol. 57 (23), pp. 9958-70. Date of Electronic Publication: 2014 Dec 02.

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

Structure-based design and synthesis of tricyclic IAP (Inhibitors of Apoptosis Proteins) inhibitors.

Authors: Hird AW Aquila BM Block MH et al.

Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2014 Apr 01; Vol. 24 (7), pp. 1820-4. Date of Electronic Publication: 2014 Feb 24.

Publication Type: Journal Article

Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE

Structure and Property Based Design of Pyrazolo[1,5-a]pyrimidine Inhibitors of CK2 Kinase with Activity in Vivo.

Authors: Dowling JE Alimzhanov M Bao L et al.

Source: ACS medicinal chemistry letters [ACS Med Chem Lett] 2013 Jul 03; Vol. 4 (8), pp. 800-5. Date of Electronic Publication: 2013 Jul 03 (Print Publication: 2013).

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE

Discovery of Disubstituted Imidazo[4,5-b]pyridines and Purines as Potent TrkA Inhibitors.

Authors: Wang T Lamb ML Block MH et al.

Source: ACS medicinal chemistry letters [ACS Med Chem Lett] 2012 Jul 26; Vol. 3 (9), pp. 705-9. Date of Electronic Publication: 2012 Jul 26 (Print Publication: 2012).

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE

Discovery of novel benzylidene-1,3-thiazolidine-2,4-diones as potent and selective inhibitors of the PIM-1, PIM-2, and PIM-3 protein kinases.

Authors: Dakin LA Block MH Chen H et al.

Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2012 Jul 15; Vol. 22 (14), pp. 4599-604. Date of Electronic Publication: 2012 Jun 06.

Publication Type: Journal Article

Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE

Potent and Selective Inhibitors of CK2 Kinase Identified through Structure-Guided Hybridization.

Authors: Dowling JE Chuaqui C Pontz TW et al.

Source: ACS medicinal chemistry letters [ACS Med Chem Lett] 2012 Jan 24; Vol. 3 (4), pp. 278-83. Date of Electronic Publication: 2012 Jan 24 (Print Publication: 2012).

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE

Discovery of (+)-N-(3-aminopropyl)-N-[1-(5-benzyl-3-methyl-4-oxo-[1,2]thiazolo[5,4-d]pyrimidin-6-yl)-2-methylpropyl]-4-methylbenzamide (AZD4877), a kinesin spindle protein inhibitor and potential anticancer agent.

Authors: Theoclitou ME Aquila B Block MH et al.

Source: Journal of medicinal chemistry [J Med Chem] 2011 Oct 13; Vol. 54 (19), pp. 6734-50. Date of Electronic Publication: 2011 Sep 07.

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

In vitro and in vivo evaluation of 6-aminopyrazolyl-pyridine-3-carbonitriles as JAK2 kinase inhibitors.

Authors: Wang T Ioannidis S Almeida L et al.

Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2011 May 15; Vol. 21 (10), pp. 2958-61. Date of Electronic Publication: 2011 Mar 21.

Publication Type: Journal Article

Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE

Discovery of 5-chloro-N2-[(1S)-1-(5-fluoropyrimidin-2-yl)ethyl]-N4-(5-methyl-1H-pyrazol-3-yl)pyrimidine-2,4-diamine (AZD1480) as a novel inhibitor of the Jak/Stat pathway.

Authors: Ioannidis S Lamb ML Wang T et al.

Source: Journal of medicinal chemistry [J Med Chem] 2011 Jan 13; Vol. 54 (1), pp. 262-76. Date of Electronic Publication: 2010 Dec 07.

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

Identification of amidoheteroaryls as potent inhibitors of mutant (V600E) B-Raf kinase with in vivo activity.

Authors: Lyne PD Aquila B Cook DJ et al.

Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2009 Feb 01; Vol. 19 (3), pp. 1026-9. Date of Electronic Publication: 2008 Oct 15.

Publication Type: Journal Article

Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE

Identification of 4-aminopyrazolylpyrimidines as potent inhibitors of Trk kinases.

Authors: Wang T Lamb ML Scott DA et al.

Source: Journal of medicinal chemistry [J Med Chem] 2008 Aug 14; Vol. 51 (15), pp. 4672-84. Date of Electronic Publication: 2008 Jul 23.

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

Cross coupling reactions of organozinc iodides with solid-supported electrophiles: synthesis of 4-substituted benzoic and 3-substituted (E)- and (Z)-propenoic acids and amides.

Authors: Oates LJ Jackson RF Block MH

Source: Organic & biomolecular chemistry [Org Biomol Chem] 2003 Jan 07; Vol. 1 (1), pp. 140-4.

Publication Type: Journal Article

Journal Info: Publisher: Royal Society of Chemistry Country of Publication: England NLM ID: 101154995 Publication Model: Print Cited Medium: Print ISSN: 1477-0520 (Print) Linking ISSN: 14770520 NLM ISO Abbreviation: Org Biomol Chem Subsets: PubMed not MEDLINE

Discovery and optimization of a series of carbazole ureas as NPY5 antagonists for the treatment of obesity.

Authors: Block MH Boyer S Brailsford W et al.

Source: Journal of medicinal chemistry [J Med Chem] 2002 Aug 01; Vol. 45 (16), pp. 3509-23.

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print Cited Medium: Print ISSN: 0022-2623 (Print) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

A Coagulation Defect Produced by Nitrogen Mustard.

Authors: Smith TR Jacobson LO Spurr CL et al.

Source: Science (New York, N.Y.) [Science] 1948 May 07; Vol. 107 (2784), pp. 474.

Publication Type: Journal Article

Journal Info: Publisher: American Association for the Advancement of Science Country of Publication: United States NLM ID: 0404511 Publication Model: Print Cited Medium: Print ISSN: 0036-8075 (Print) Linking ISSN: 00368075 NLM ISO Abbreviation: Science Subsets: OLDMEDLINE

Studies on Radiosensitivity of Cells.

Authors: Jacobson LO Marks EK Gaston EO et al.

Source: Science (New York, N.Y.) [Science] 1948 Mar 05; Vol. 107 (2775), pp. 248-50.

Publication Type: Journal Article

Journal Info: Publisher: American Association for the Advancement of Science Country of Publication: United States NLM ID: 0404511 Publication Model: Print Cited Medium: Print ISSN: 0036-8075 (Print) Linking ISSN: 00368075 NLM ISO Abbreviation: Science Subsets: OLDMEDLINE

The aminoquinazoline group as a replacement for the salicylamide group: the design and synthesis of a novel highly selective beta 1 adrenoceptor partial agonist.

Authors: Block MH Kenny PW Thomson DS et al.

Source: Drug design and discovery [Drug Des Discov] 1992; Vol. 9 (2), pp. 167-76.

Publication Type: Journal Article

Journal Info: Publisher: Harwood Academic Publishers Country of Publication: Switzerland NLM ID: 9200627 Publication Model: Print Cited Medium: Print ISSN: 1055-9612 (Print) Linking ISSN: 10267921 NLM ISO Abbreviation: Drug Des Discov Subsets: MEDLINE

Intravenous iron dextran in clinical medicine.

Authors: Hamstra RD Block MH Schocket AL

Source: JAMA [JAMA] 1980 May 02; Vol. 243 (17), pp. 1726-31.

Publication Type: Comparative Study; Journal Article; Research Support, U.S. Gov't, P.H.S.

Journal Info: Publisher: American Medical Association Country of Publication: United States NLM ID: 7501160 Publication Model: Print Cited Medium: Print ISSN: 0098-7484 (Print) Linking ISSN: 00987484 NLM ISO Abbreviation: JAMA Subsets: MEDLINE