Search Results - "Burkard MR"

Identification of the Clinical Development Candidate MRTX849, a Covalent KRAS^G12C Inhibitor for the Treatment of Cancer.

Authors: Fell JB Fischer JP Baer BR et al.

Source: Journal of medicinal chemistry [J Med Chem] 2020 Jul 09; Vol. 63 (13), pp. 6679-6693. Date of Electronic Publication: 2020 Apr 06.

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

The KRAS^G12C Inhibitor MRTX849 Provides Insight toward Therapeutic Susceptibility of KRAS-Mutant Cancers in Mouse Models and Patients.

Authors: Hallin J Engstrom LD Hargis L et al.

Source: Cancer discovery [Cancer Discov] 2020 Jan; Vol. 10 (1), pp. 54-71. Date of Electronic Publication: 2019 Oct 28.

Publication Type: Case Reports; Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

Journal Info: Publisher: American Association for Cancer Research Country of Publication: United States NLM ID: 101561693 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2159-8290 (Electronic) Linking ISSN: 21598274 NLM ISO Abbreviation: Cancer Discov Subsets: MEDLINE

Emergence and Targeting of Acquired and Hereditary Resistance to Multikinase RET Inhibition in Patients With RET-Altered Cancer.

Authors: Wirth LJ Kohno T Udagawa H et al.

Source: JCO precision oncology [JCO Precis Oncol] 2019 Sep 11; Vol. 3. Date of Electronic Publication: 2019 Sep 11 (Print Publication: 2019).

Publication Type: Case Reports; Journal Article

Journal Info: Publisher: American Society of Clinical Oncology Country of Publication: United States NLM ID: 101705370 Publication Model: eCollection Cited Medium: Internet ISSN: 2473-4284 (Electronic) Linking ISSN: 24734284 NLM ISO Abbreviation: JCO Precis Oncol Subsets: PubMed not MEDLINE

Discovery of Tetrahydropyridopyrimidines as Irreversible Covalent Inhibitors of KRAS-G12C with In Vivo Activity.

Authors: Fell JB Fischer JP Baer BR et al.

Source: ACS medicinal chemistry letters [ACS Med Chem Lett] 2018 Nov 07; Vol. 9 (12), pp. 1230-1234. Date of Electronic Publication: 2018 Nov 07 (Print Publication: 2018).

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE

Transient reexpression of an embryonic autonomous growth phenotype by adult carotid artery smooth muscle cells after vascular injury.

Authors: Weiser-Evans MC Quinn BE Burkard MR et al.

Source: Journal of cellular physiology [J Cell Physiol] 2000 Jan; Vol. 182 (1), pp. 12-23.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.

Journal Info: Publisher: Wiley-Liss Country of Publication: United States NLM ID: 0050222 Publication Model: Print Cited Medium: Print ISSN: 0021-9541 (Print) Linking ISSN: 00219541 NLM ISO Abbreviation: J Cell Physiol Subsets: MEDLINE

In vitro studies of a bradykinin B1/B2 antagonist linked to a human neutrophil elastase inhibitor; a heterodimer for the treatment of inflammatory disorders.

Authors: Leimer AH Kroona HB Blodgett JK et al.

Source: Canadian journal of physiology and pharmacology [Can J Physiol Pharmacol] 1997 Jun; Vol. 75 (6), pp. 633-8.

Publication Type: Journal Article

Journal Info: Publisher: Canadian Science Publishing Country of Publication: Canada NLM ID: 0372712 Publication Model: Print Cited Medium: Print ISSN: 0008-4212 (Print) Linking ISSN: 00084212 NLM ISO Abbreviation: Can J Physiol Pharmacol Subsets: MEDLINE

Inducible bradykinin B1 receptor in isolated human ileum.

Authors: Zuzack JS Burkard MR Cuadrado DK et al.

Source: Immunopharmacology [Immunopharmacology] 1996 Jun; Vol. 33 (1-3), pp. 113-5.

Publication Type: Journal Article

Journal Info: Publisher: Elsevier/North-Holland Country of Publication: Netherlands NLM ID: 7902474 Publication Model: Print Cited Medium: Print ISSN: 0162-3109 (Print) Linking ISSN: 01623109 NLM ISO Abbreviation: Immunopharmacology Subsets: MEDLINE

Evidence of a bradykinin B1 receptor in human ileum: pharmacological comparison to the rabbit aorta B1 receptor.

Authors: Zuzack JS Burkard MR Cuadrado DK et al.

Source: The Journal of pharmacology and experimental therapeutics [J Pharmacol Exp Ther] 1996 Jun; Vol. 277 (3), pp. 1337-43.

Publication Type: Journal Article

Journal Info: Publisher: Elsevier Country of Publication: Netherlands NLM ID: 0376362 Publication Model: Print Cited Medium: Print ISSN: 0022-3565 (Print) Linking ISSN: 00223565 NLM ISO Abbreviation: J Pharmacol Exp Ther Subsets: MEDLINE