Search Results - "Coderch, Claire"

The Many Ways to Deal with STING.

Authors: Coderch, Claire Arranz-Herrero, Javier Nistal-Villan, Estanislao et al.

Source: International Journal of Molecular Sciences. May2023, Vol. 24 Issue 10, p9032. 31p.

In silico identification and in vivo characterization of small molecule therapeutic hypothermia mimetics.

Authors: Coderch, Claire Díaz de Cerio, María Zapico, Jose María et al.

Source: Bioorganic & Medicinal Chemistry. Dec2017, Vol. 25 Issue 24, p6597-6604. 8p.

Mechanistic insight into the reaction catalysed by bacterial type II dehydroquinases.

Authors: CODERCH, Claire LENCE, Emilio PEON, Antonio et al.

Source: Biochemical Journal. 3/15/2014, Vol. 458 Issue 3, p547-557. 22p.

Synthesis and Biological Evaluation of a New Series of Highly Functionalized 7′-homo-Anhydrovinblastine Derivatives.

Authors: Gherbovet, Olga Coderch, Claire García Alvarez, María Concepción et al.

Source: Journal of Medicinal Chemistry. Vol. 56 Issue 15, p6088-6100. 13p.

Proteasomal Degradation of Zn-Dependent Hdacs: The E3-Ligases Implicated and the Designed Protacs That Enable Degradation.

Authors: Márquez-Cantudo, Laura Ramos, Ana Coderch, Claire et al.

Source: Molecules. Sep2021, Vol. 26 Issue 18, p5606. 1p.

Design and Synthesis of Water-Soluble and Potent MMP-13 Inhibitors with Activity in Human Osteosarcoma Cells.

Authors: Zapico, Jose Maria Acosta, Lourdes Pastor, Miryam et al.

Source: International Journal of Molecular Sciences. Sep2021, Vol. 22 Issue 18, p9976. 1p.

Pharmacological inhibition of Receptor Protein Tyrosine Phosphatase β/ζ (PTPRZ1) modulates behavioral responses to ethanol.

Authors: Fernández-Calle, Rosalía Vicente-Rodríguez, Marta Pastor, Miryam et al.

Source: Neuropharmacology. Jul2018, Vol. 137, p86-95. 10p.

Development of inhibitors of receptor protein tyrosine phosphatase β/ζ (PTPRZ1) as candidates for CNS disorders.

Authors: Pastor, Miryam Fernández-Calle, Rosalía Di Geronimo, Bruno et al.

Source: European Journal of Medicinal Chemistry. Jan2018, Vol. 144, p318-329. 12p.

Multitarget Anticancer Agents Based on Histone Deacetylase and Protein Kinase CK2 Inhibitors.

Authors: Martínez, Regina Di Geronimo, Bruno Pastor, Miryam et al.

Source: Molecules. Apr2020, Vol. 25 Issue 7, p1497. 1p. 9 Diagrams, 2 Charts, 4 Graphs.

Molecular Imaging Probes Based on Matrix Metalloproteinase Inhibitors (MMPIs).

Authors: Rangasamy, Loganathan Di Geronimo, Bruno Ortín, Irene et al.

Source: Molecules. Aug2019, Vol. 24 Issue 16, p2982-2982. 1p. 27 Diagrams, 2 Charts, 2 Graphs.

Identification of Aldo-Keto Reductase AKR1B10 as a Selective Target for Modification and Inhibition by Prostaglandin A1: Implications for Antitumoral Activity.

Authors: Díez-Dacal, Beatriz Gayarre, Javier Gharbi, Severine et al.

Source: Cancer Research. Jun2011, Vol. 71 Issue 12, p4161-4171. 11p.

Optimization of Taxane Binding to Microtubules: Binding Affinity Dissection and Incremental Construction of a High-Affinity Analog of Paclitaxel

Authors: Matesanz, Ruth Barasoain, Isabel Yang, Chun-Gang et al.

Source: Chemistry & Biology. Jun2008, Vol. 15 Issue 6, p573-585. 13p.

STING activation by teniposide: a potential direct mechanism beyond cGAS stimulation.

Authors: Arranz-Herrero J Marquez-Cantudo L Rius-Rocabert S et al.

Source: Frontiers in immunology [Front Immunol] 2026 Jan 02; Vol. 16, pp. 1677836. Date of Electronic Publication: 2026 Jan 02 (Print Publication: 2025).

Publication Type: Journal Article

Journal Info: Publisher: Frontiers Research Foundation] Country of Publication: Switzerland NLM ID: 101560960 Publication Model: eCollection Cited Medium: Internet ISSN: 1664-3224 (Electronic) Linking ISSN: 16643224 NLM ISO Abbreviation: Front Immunol Subsets: MEDLINE

Computational Insights into the Structural Basis for Reduced Hepatotoxicity of Novel Nonopioid Analgesics.

Authors: Coderch C Bazán HA Bazan NG et al.

Source: ChemMedChem [ChemMedChem] 2025 Nov 18; Vol. 20 (22), pp. e202500639. Date of Electronic Publication: 2025 Oct 21.

Publication Type: Journal Article

Journal Info: Publisher: Wiley-VCH Country of Publication: Germany NLM ID: 101259013 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1860-7187 (Electronic) Linking ISSN: 18607179 NLM ISO Abbreviation: ChemMedChem Subsets: MEDLINE

Comparative binding energy COMBINE analysis for understanding the binding determinants of type II dehydroquinase inhibitors.

Authors: Peón A Coderch C Gago F et al.

Source: ChemMedChem [ChemMedChem] 2013 May; Vol. 8 (5), pp. 740-7. Date of Electronic Publication: 2013 Mar 01.

Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Wiley-VCH Country of Publication: Germany NLM ID: 101259013 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1860-7187 (Electronic) Linking ISSN: 18607179 NLM ISO Abbreviation: ChemMedChem Subsets: MEDLINE

New Dual CK2/HDAC1 Inhibitors with Nanomolar Inhibitory Activity against Both Enzymes.

Authors: Rangasamy L Ortín I Zapico JM et al.

Source: ACS medicinal chemistry letters [ACS Med Chem Lett] 2020 Apr 07; Vol. 11 (5), pp. 713-719. Date of Electronic Publication: 2020 Apr 07 (Print Publication: 2020).

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE

From a MMP2/CK2 multitarget approach to the identification of potent and selective MMP13 inhibitors.

Authors: Pastor M Zapico JM Coderch C et al.

Source: Organic & biomolecular chemistry [Org Biomol Chem] 2019 Jan 23; Vol. 17 (4), pp. 916-929.

Publication Type: Journal Article

Journal Info: Publisher: Royal Society of Chemistry Country of Publication: England NLM ID: 101154995 Publication Model: Print Cited Medium: Internet ISSN: 1477-0539 (Electronic) Linking ISSN: 14770520 NLM ISO Abbreviation: Org Biomol Chem Subsets: MEDLINE

Discovery of potent calpain inhibitors based on the azolo-imidazolidenone scaffold.

Authors: Gutiérrez S Morón M Griera M et al.

Source: European journal of medicinal chemistry [Eur J Med Chem] 2018 Sep 05; Vol. 157, pp. 946-959. Date of Electronic Publication: 2018 Aug 17.

Publication Type: Journal Article

Journal Info: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1768-3254 (Electronic) Linking ISSN: 02235234 NLM ISO Abbreviation: Eur J Med Chem Subsets: MEDLINE

Design and synthesis of potent hydroxamate inhibitors with increased selectivity within the gelatinase family.

Authors: Zapico JM Puckowska A Filipiak K et al.

Source: Organic & biomolecular chemistry [Org Biomol Chem] 2015 Jan 07; Vol. 13 (1), pp. 142-56.

Publication Type: Journal Article

Journal Info: Publisher: Royal Society of Chemistry Country of Publication: England NLM ID: 101154995 Publication Model: Print Cited Medium: Internet ISSN: 1477-0539 (Electronic) Linking ISSN: 14770520 NLM ISO Abbreviation: Org Biomol Chem Subsets: MEDLINE

One-pot synthesis of vinca alkaloids-phomopsin hybrids.

Authors: Gherbovet O Coderch C García Alvarez MC et al.

Source: Journal of medicinal chemistry [J Med Chem] 2014 Jun 26; Vol. 57 (12), pp. 5470-6. Date of Electronic Publication: 2014 Jun 10.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE