Search Results - "Edink E"

To Target or Not to Target Schistosoma mansoni Cyclic Nucleotide Phosphodiesterase 4A?

Authors: Zheng Y Schroeder S Kanev GK et al.

Source: International journal of molecular sciences [Int J Mol Sci] 2023 Apr 06; Vol. 24 (7). Date of Electronic Publication: 2023 Apr 06.

Publication Type: Journal Article

Journal Info: Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium: Internet ISSN: 1422-0067 (Electronic) Linking ISSN: 14220067 NLM ISO Abbreviation: Int J Mol Sci Subsets: MEDLINE

From recipe to research: introducing undergraduate students to the nature of science using a hybrid practical course centred on drug discovery for neglected diseases.

Authors: Wijtmans M Edink E van Linden OP et al.

Source: Drug discovery today [Drug Discov Today] 2021 Jun; Vol. 26 (6), pp. 1359-1368. Date of Electronic Publication: 2021 Feb 18.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Review

Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9604391 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1878-5832 (Electronic) Linking ISSN: 13596446 NLM ISO Abbreviation: Drug Discov Today Subsets: MEDLINE

Discovery of Diaryl Ether Substituted Tetrahydrophthalazinones as TbrPDEB1 Inhibitors Following Structure-Based Virtual Screening.

Authors: de Heuvel E Kooistra AJ Edink E et al.

Source: Frontiers in chemistry [Front Chem] 2021 Jan 21; Vol. 8, pp. 608030. Date of Electronic Publication: 2021 Jan 21 (Print Publication: 2020).

Publication Type: Journal Article

Journal Info: Publisher: Frontiers Media S.A Country of Publication: Switzerland NLM ID: 101627988 Publication Model: eCollection Cited Medium: Print ISSN: 2296-2646 (Print) Linking ISSN: 22962646 NLM ISO Abbreviation: Front Chem Subsets: PubMed not MEDLINE

Alkynamide phthalazinones as a new class of TbrPDEB1 inhibitors.

Authors: de Heuvel E Singh AK Edink E et al.

Source: Bioorganic & medicinal chemistry [Bioorg Med Chem] 2019 Sep 15; Vol. 27 (18), pp. 3998-4012. Date of Electronic Publication: 2019 Jun 18.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Elsevier Science Country of Publication: England NLM ID: 9413298 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3391 (Electronic) Linking ISSN: 09680896 NLM ISO Abbreviation: Bioorg Med Chem Subsets: MEDLINE

Targeting a Subpocket in Trypanosoma brucei Phosphodiesterase B1 (TbrPDEB1) Enables the Structure-Based Discovery of Selective Inhibitors with Trypanocidal Activity.

Authors: Blaazer AR Singh AK de Heuvel E et al.

Source: Journal of medicinal chemistry [J Med Chem] 2018 May 10; Vol. 61 (9), pp. 3870-3888. Date of Electronic Publication: 2018 May 01.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

4,6-Diphenylpyridines as Promising Novel Anti-Influenza Agents Targeting the PA-PB1 Protein-Protein Interaction: Structure-Activity Relationships Exploration with the Aid of Molecular Modeling.

Authors: Trist IM Nannetti G Tintori C et al.

Source: Journal of medicinal chemistry [J Med Chem] 2016 Mar 24; Vol. 59 (6), pp. 2688-703. Date of Electronic Publication: 2016 Mar 11.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

Fragment-based screening in tandem with phenotypic screening provides novel antiparasitic hits.

Authors: Blaazer AR Orrling KM Shanmugham A et al.

Source: Journal of biomolecular screening [J Biomol Screen] 2015 Jan; Vol. 20 (1), pp. 131-40. Date of Electronic Publication: 2014 Sep 17.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Sage Publications Country of Publication: United States NLM ID: 9612112 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1552-454X (Electronic) Linking ISSN: 10870571 NLM ISO Abbreviation: J Biomol Screen Subsets: MEDLINE

Identification of novel α7 nicotinic receptor ligands by in silico screening against the crystal structure of a chimeric α7 receptor ligand binding domain.

Authors: Akdemir A Edink E Thompson AJ et al.

Source: Bioorganic & medicinal chemistry [Bioorg Med Chem] 2012 Oct 01; Vol. 20 (19), pp. 5992-6002. Date of Electronic Publication: 2012 Jul 11.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Elsevier Science Country of Publication: England NLM ID: 9413298 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3391 (Electronic) Linking ISSN: 09680896 NLM ISO Abbreviation: Bioorg Med Chem Subsets: MEDLINE

Structure-based design, synthesis and structure-activity relationships of dibenzosuberyl- and benzoate-substituted tropines as ligands for acetylcholine-binding protein.

Authors: Edink E Akdemir A Jansen C et al.

Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2012 Feb 01; Vol. 22 (3), pp. 1448-54. Date of Electronic Publication: 2011 Dec 09.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE

High-resolution bioactivity profiling of mixtures toward the acetylcholine binding protein using a nanofractionation spotter technology.

Authors: Kool J Heus F de Kloe G et al.

Source: Journal of biomolecular screening [J Biomol Screen] 2011 Sep; Vol. 16 (8), pp. 917-24. Date of Electronic Publication: 2011 Jul 28.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Sage Publications Country of Publication: United States NLM ID: 9612112 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1552-454X (Electronic) Linking ISSN: 10870571 NLM ISO Abbreviation: J Biomol Screen Subsets: MEDLINE

Fragment growing induces conformational changes in acetylcholine-binding protein: a structural and thermodynamic analysis.

Authors: Edink E Rucktooa P Retra K et al.

Source: Journal of the American Chemical Society [J Am Chem Soc] 2011 Apr 13; Vol. 133 (14), pp. 5363-71. Date of Electronic Publication: 2011 Feb 15.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 7503056 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-5126 (Electronic) Linking ISSN: 00027863 NLM ISO Abbreviation: J Am Chem Soc Subsets: MEDLINE

Conjugation of penicillin acylase with the reactive copolymer of N-isopropylacrylamide: a step toward a thermosensitive industrial biocatalyst.

Authors: Ivanov AE Edink E Kumar A et al.

Source: Biotechnology progress [Biotechnol Prog] 2003 Jul-Aug; Vol. 19 (4), pp. 1167-75.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Wiley-Blackwell Country of Publication: United States NLM ID: 8506292 Publication Model: Print Cited Medium: Print ISSN: 8756-7938 (Print) Linking ISSN: 15206033 NLM ISO Abbreviation: Biotechnol Prog Subsets: MEDLINE