Search Results - "El-Subbagh HI"

Pyrazolopyridine-Containing Compounds as Multitargeted Anti-Alzheimer Agents: Synthesis, Biological Evaluation, and In Silico Studies.

Authors: Waly OM El-Sayed SM Ghaly MA et al.

Source: Archiv der Pharmazie [Arch Pharm (Weinheim)] 2025 Jun; Vol. 358 (6), pp. e70025.

Publication Type: Journal Article

Journal Info: Publisher: Wiley-VCH Verlag GmbH & Co. KGaA Country of Publication: Germany NLM ID: 0330167 Publication Model: Print Cited Medium: Internet ISSN: 1521-4184 (Electronic) Linking ISSN: 03656233 NLM ISO Abbreviation: Arch Pharm (Weinheim) Subsets: MEDLINE

New quinazolinone-based derivatives as DHFR/EGFR-TK inhibitors: Synthesis, molecular modeling simulations, and anticancer activity.

Authors: El-Gazzar YI Ghaiad HR El Kerdawy AM et al.

Source: Archiv der Pharmazie [Arch Pharm (Weinheim)] 2023 Jan; Vol. 356 (1), pp. e2200417. Date of Electronic Publication: 2022 Oct 18.

Publication Type: Journal Article

Journal Info: Publisher: Wiley-VCH Verlag GmbH & Co. KGaA Country of Publication: Germany NLM ID: 0330167 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1521-4184 (Electronic) Linking ISSN: 03656233 NLM ISO Abbreviation: Arch Pharm (Weinheim) Subsets: MEDLINE

Taguchi Approach for Optimization of a Green Quantitative 1H-NMR Practice for Characterization of Levetiracetam and Brivaracetam in Pharmaceuticals.

Authors: Mansour NM El-Sherbiny DT Ibrahim FA et al.

Source: Journal of AOAC International [J AOAC Int] 2022 Oct 26; Vol. 105 (6), pp. 1516-1527.

Publication Type: Journal Article

Journal Info: Publisher: Oxford University Press Country of Publication: England NLM ID: 9215446 Publication Model: Print Cited Medium: Internet ISSN: 1944-7922 (Electronic) Linking ISSN: 10603271 NLM ISO Abbreviation: J AOAC Int Subsets: MEDLINE

Thiazole-based SARS-CoV-2 protease (COV M^pro ) inhibitors: Design, synthesis, enzyme inhibition, and molecular modeling simulations.

Authors: Elsayed RW Sabry MA El-Subbagh HI et al.

Source: Archiv der Pharmazie [Arch Pharm (Weinheim)] 2022 Sep; Vol. 355 (9), pp. e2200121. Date of Electronic Publication: 2022 May 23.

Publication Type: Journal Article

Journal Info: Publisher: Wiley-VCH Verlag GmbH & Co. KGaA Country of Publication: Germany NLM ID: 0330167 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1521-4184 (Electronic) Linking ISSN: 03656233 NLM ISO Abbreviation: Arch Pharm (Weinheim) Subsets: MEDLINE

Synthesis, molecular modeling simulations and anticancer activity of some new Imidazo[2,1-b]thiazole analogues as EGFR/HER2 and DHFR inhibitors.

Authors: Moharram EA El-Sayed SM Ghabbour HA et al.

Source: Bioorganic chemistry [Bioorg Chem] 2024 Sep; Vol. 150, pp. 107538. Date of Electronic Publication: 2024 Jun 06.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Elsevier Country of Publication: United States NLM ID: 1303703 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1090-2120 (Electronic) Linking ISSN: 00452068 NLM ISO Abbreviation: Bioorg Chem Subsets: MEDLINE

Nanomolar potency of imidazo[2,1-b]thiazole analogs as indoleamine 2,3-dioxygenase inhibitors.

Authors: Ewida MA Ewida HA Ahmed MS et al.

Source: Archiv der Pharmazie [Arch Pharm (Weinheim)] 2021 Nov; Vol. 354 (11), pp. e2100202. Date of Electronic Publication: 2021 Jul 27.

Publication Type: Journal Article

Journal Info: Publisher: Wiley-VCH Verlag GmbH & Co. KGaA Country of Publication: Germany NLM ID: 0330167 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1521-4184 (Electronic) Linking ISSN: 03656233 NLM ISO Abbreviation: Arch Pharm (Weinheim) Subsets: MEDLINE

Multi-targeted anti-Alzheimer's agents: Synthesis, biological evaluation, and molecular modeling study of some pyrazolopyridine hybrids.

Authors: Waly OM El-Sayed SM Ghaly MA et al.

Source: European journal of medicinal chemistry [Eur J Med Chem] 2023 Dec 15; Vol. 262, pp. 115880. Date of Electronic Publication: 2023 Oct 20.

Publication Type: Journal Article

Journal Info: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1768-3254 (Electronic) Linking ISSN: 02235234 NLM ISO Abbreviation: Eur J Med Chem Subsets: MEDLINE

Editorial: Recent advances in the research and development of kinase-inhibitory anticancer molecules.

Authors: Al-Karmalawy AA El-Subbagh HI Logoyda L et al.

Source: Frontiers in chemistry [Front Chem] 2023 Nov 09; Vol. 11, pp. 1328424. Date of Electronic Publication: 2023 Nov 09 (Print Publication: 2023).

Publication Type: Editorial

Journal Info: Publisher: Frontiers Media S.A Country of Publication: Switzerland NLM ID: 101627988 Publication Model: eCollection Cited Medium: Print ISSN: 2296-2646 (Print) Linking ISSN: 22962646 NLM ISO Abbreviation: Front Chem Subsets: PubMed not MEDLINE

Discovery of new pyridine heterocyclic hybrids; design, synthesis, dynamic simulations, and in vitro and in vivo breast cancer biological assays.

Authors: Abdelshaheed MM El Subbagh HI Tantawy MA et al.

Source: RSC advances [RSC Adv] 2023 May 24; Vol. 13 (23), pp. 15689-15703. Date of Electronic Publication: 2023 May 24 (Print Publication: 2023).

Publication Type: Journal Article

Journal Info: Publisher: Royal Society of Chemistry Country of Publication: England NLM ID: 101581657 Publication Model: eCollection Cited Medium: Internet ISSN: 2046-2069 (Electronic) Linking ISSN: 20462069 NLM ISO Abbreviation: RSC Adv Subsets: PubMed not MEDLINE

Hydrazinecarbonyl-thiazol-2-acetamides with pronounced apoptotic behavior: synthesis, in vitro/in vivo anti-proliferative activity and molecular modeling simulations.

Authors: Elsayed RW Bayoumi SM El-Subbagh HI et al.

Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2023 May 01; Vol. 87, pp. 129285. Date of Electronic Publication: 2023 Apr 11.

Publication Type: Journal Article

Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE

New thiazole-based derivatives as EGFR/HER2 and DHFR inhibitors: Synthesis, molecular modeling simulations and anticancer activity.

Authors: Sabry MA Ghaly MA Maarouf AR et al.

Source: European journal of medicinal chemistry [Eur J Med Chem] 2022 Nov 05; Vol. 241, pp. 114661. Date of Electronic Publication: 2022 Aug 10.

Publication Type: Journal Article

Journal Info: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1768-3254 (Electronic) Linking ISSN: 02235234 NLM ISO Abbreviation: Eur J Med Chem Subsets: MEDLINE

Analysis of two mixtures containing racetams in their pharmaceuticals using simple spectrophotometric methodologies.

Authors: Mansour NM El-Sherbiny DT Ibrahim FA et al.

Source: Annales pharmaceutiques francaises [Ann Pharm Fr] 2022 Nov; Vol. 80 (6), pp. 885-896. Date of Electronic Publication: 2022 Jun 16.

Publication Type: Journal Article

Journal Info: Publisher: Elsevier Masson Editeur Country of Publication: France NLM ID: 2985176R Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2772-803X (Electronic) Linking ISSN: 00034509 NLM ISO Abbreviation: Ann Pharm Fr Subsets: MEDLINE

New phthalimide-based derivatives as EGFR-TK inhibitors: Synthesis, biological evaluation, and molecular modeling study.

Authors: Mansour NI El-Sayed SM El-Gohary NS et al.

Source: Bioorganic chemistry [Bioorg Chem] 2022 Oct; Vol. 127, pp. 105966. Date of Electronic Publication: 2022 Jun 14.

Publication Type: Journal Article

Journal Info: Publisher: Elsevier Country of Publication: United States NLM ID: 1303703 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1090-2120 (Electronic) Linking ISSN: 00452068 NLM ISO Abbreviation: Bioorg Chem Subsets: MEDLINE

Synthesis, biological evaluation, and molecular modeling simulations of new heterocyclic hybrids as multi-targeted anti-Alzheimer's agents.

Authors: Waly OM Saad KM El-Subbagh HI et al.

Source: European journal of medicinal chemistry [Eur J Med Chem] 2022 Mar 05; Vol. 231, pp. 114152. Date of Electronic Publication: 2022 Jan 22.

Publication Type: Journal Article

Journal Info: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1768-3254 (Electronic) Linking ISSN: 02235234 NLM ISO Abbreviation: Eur J Med Chem Subsets: MEDLINE

3-Methyl-imidazo[2,1-b]thiazole derivatives as a new class of antifolates: Synthesis, in vitro/in vivo bio-evaluation and molecular modeling simulations.

Authors: Ewida MA Ewida HA Ahmed MS et al.

Source: Bioorganic chemistry [Bioorg Chem] 2021 Oct; Vol. 115, pp. 105205. Date of Electronic Publication: 2021 Jul 24.

Publication Type: Journal Article

Journal Info: Publisher: Elsevier Country of Publication: United States NLM ID: 1303703 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1090-2120 (Electronic) Linking ISSN: 00452068 NLM ISO Abbreviation: Bioorg Chem Subsets: MEDLINE

Novel 1,2,4-oxadiazole-chalcone/oxime hybrids as potential antibacterial DNA gyrase inhibitors: Design, synthesis, ADMET prediction and molecular docking study.

Authors: Ibrahim TS Almalki AJ Moustafa AH et al.

Source: Bioorganic chemistry [Bioorg Chem] 2021 Jun; Vol. 111, pp. 104885. Date of Electronic Publication: 2021 Apr 01.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Elsevier Country of Publication: United States NLM ID: 1303703 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1090-2120 (Electronic) Linking ISSN: 00452068 NLM ISO Abbreviation: Bioorg Chem Subsets: MEDLINE

Novel GABAA Agonist Entities: Pharmacological Investigation and Molecular Modeling Study of Thiazolo- and Thiadiazolo-[3,2-a][1,3]diazepine Analogs.

Authors: El-Subbagh HI; Department of Medicinal Chemistry, College of Pharmacy, Mansoura University, Mansoura 35516, Egypt.

Source: Mini reviews in medicinal chemistry [Mini Rev Med Chem] 2021; Vol. 21 (9), pp. 1048-1057.

Publication Type: Journal Article; Review

Journal Info: Publisher: Bentham Science Publishers Country of Publication: Netherlands NLM ID: 101094212 Publication Model: Print Cited Medium: Internet ISSN: 1875-5607 (Electronic) Linking ISSN: 13895575 NLM ISO Abbreviation: Mini Rev Med Chem Subsets: MEDLINE

2-Substituted-mercapto-quinazolin-4(3H)-ones as DHFR Inhibitors.

Authors: El-Subbagh HI Sabry MA

Source: Mini reviews in medicinal chemistry [Mini Rev Med Chem] 2021; Vol. 21 (16), pp. 2249-2260.

Publication Type: Journal Article; Review

Journal Info: Publisher: Bentham Science Publishers Country of Publication: Netherlands NLM ID: 101094212 Publication Model: Print Cited Medium: Internet ISSN: 1875-5607 (Electronic) Linking ISSN: 13895575 NLM ISO Abbreviation: Mini Rev Med Chem Subsets: MEDLINE

Design, synthesis and molecular modeling of novel aryl carboximidamides and 3-aryl-1,2,4-oxadiazoles derived from indomethacin as potent anti-inflammatory iNOS/PGE2 inhibitors.

Authors: Mohamed MFA Marzouk AA Nafady A et al.

Source: Bioorganic chemistry [Bioorg Chem] 2020 Dec; Vol. 105, pp. 104439. Date of Electronic Publication: 2020 Oct 28.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Elsevier Country of Publication: United States NLM ID: 1303703 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1090-2120 (Electronic) Linking ISSN: 00452068 NLM ISO Abbreviation: Bioorg Chem Subsets: MEDLINE

Multiobjective optimization of microemulsion- thin layer chromatography with image processing as analytical platform for determination of drugs in plasma using desirability functions.

Authors: Abou-Taleb NH El-Sherbiny DT El-Enany NM et al.

Source: Journal of chromatography. A [J Chromatogr A] 2020 May 24; Vol. 1619, pp. 460945. Date of Electronic Publication: 2020 Feb 05.

Publication Type: Journal Article

Journal Info: Publisher: Elsevier Country of Publication: Netherlands NLM ID: 9318488 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1873-3778 (Electronic) Linking ISSN: 00219673 NLM ISO Abbreviation: J Chromatogr A Subsets: MEDLINE