Search Results - "El-Subbagh HI"

Synthesis, antibacterial activity, in silico ADMET prediction, docking, and molecular dynamics studies of substituted phenyl and furan ring containing thiazole Schiff base derivatives.

Authors: Islam, Md. Din Saha, Joyanta Kumar Marufa, Sumita Saznin et al.

Source: PLoS ONE. 3/10/2025, Vol. 20 Issue 3, p1-28. 28p.

Pyrazolopyridine-Containing Compounds as Multitargeted Anti-Alzheimer Agents: Synthesis, Biological Evaluation, and In Silico Studies.

Authors: Waly OM El-Sayed SM Ghaly MA et al.

Source: Archiv der Pharmazie [Arch Pharm (Weinheim)] 2025 Jun; Vol. 358 (6), pp. e70025.

Publication Type: Journal Article

Journal Info: Publisher: Wiley-VCH Verlag GmbH & Co. KGaA Country of Publication: Germany NLM ID: 0330167 Publication Model: Print Cited Medium: Internet ISSN: 1521-4184 (Electronic) Linking ISSN: 03656233 NLM ISO Abbreviation: Arch Pharm (Weinheim) Subsets: MEDLINE

Synthesis, Invitro Cytotoxic Activity and Optical Analysis of Substituted Schiff Base Derivatives.

Authors: Saleem, Muhammad Hussain, Abrar Hanif, Muhammad et al.

Source: Journal of Fluorescence. Jun2025, Vol. 35 Issue 6, p3981-3989. 9p.

Discovery of a pyrazolopyridine alkaloid that mitigates neuronal ER stress and age-related decline.

Authors: Jantrapirom, Salinee Sangphukieo, Apiwat U-on, Natsinee et al.

Source: Communications Biology. 5/8/2026, p1-17. 17p.

Recent advances in pyrazolo[3,4-b]pyridine chemistry: synthesis techniques and biological activity.

Authors: Abdel-Aziem A Fouad SA

Source: Molecular diversity [Mol Divers] 2025 Jun 25. Date of Electronic Publication: 2025 Jun 25.

Publication Type: Journal Article; Review

Journal Info: Publisher: ESCOM Science Publishers Country of Publication: Netherlands NLM ID: 9516534 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1573-501X (Electronic) Linking ISSN: 13811991 NLM ISO Abbreviation: Mol Divers Subsets: MEDLINE

Synthesis, molecular modeling simulations and anticancer activity of some new Imidazo[2,1-b]thiazole analogues as EGFR/HER2 and DHFR inhibitors.

Authors: Moharram EA El-Sayed SM Ghabbour HA et al.

Source: Bioorganic chemistry [Bioorg Chem] 2024 Sep; Vol. 150, pp. 107538. Date of Electronic Publication: 2024 Jun 06.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Elsevier Country of Publication: United States NLM ID: 1303703 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1090-2120 (Electronic) Linking ISSN: 00452068 NLM ISO Abbreviation: Bioorg Chem Subsets: MEDLINE

Synergistic Sedative Activity of Indirubin on Diazepam in Thiopental Sodium-induced Sleeping Mice: A Potential GABAergic Transmission.

Authors: Khatun T Malik A Alshememry AK et al.

Source: Molecular neurobiology [Mol Neurobiol] 2025 Nov; Vol. 62 (11), pp. 13827-13839. Date of Electronic Publication: 2025 Jul 01.

Publication Type: Journal Article

Journal Info: Publisher: Humana Press Country of Publication: United States NLM ID: 8900963 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1559-1182 (Electronic) Linking ISSN: 08937648 NLM ISO Abbreviation: Mol Neurobiol Subsets: MEDLINE

Multicomponent reaction for synthesis, molecular docking, and anti-inflammatory evaluation of novel indole-thiazole hybrid derivatives.

Authors: Alkorbi F Alshareef SA Abdelaziz MA et al.

Source: Molecular diversity [Mol Divers] 2025 Oct; Vol. 29 (5), pp. 3945-3956. Date of Electronic Publication: 2024 Aug 15.

Publication Type: Journal Article

Journal Info: Publisher: ESCOM Science Publishers Country of Publication: Netherlands NLM ID: 9516534 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1573-501X (Electronic) Linking ISSN: 13811991 NLM ISO Abbreviation: Mol Divers Subsets: MEDLINE

Design, synthesis, and insilico evaluation of 2-aminothiazole derivatives as potential mTOR and EGFR inhibitors.

Authors: Swamy, Pramod Mallikarjuna Somashekar, Preetham Harave Shivamurthy, Santhosh Arehalli et al.

Source: Discover Molecules (3004-9350). Dec2025, Vol. 2 Issue 1, p1-27. 27p.

Recent progress in the exploitation of anti-cancer small molecules targeting angiogenesis.

Authors: Zheng, Ying Qiu, Hao Zhang, Ke et al.

Source: Journal of Enzyme Inhibition & Medicinal Chemistry. Dec2025, Vol. 40 Issue 1, p1-46. 46p.

Rational design, synthesis, and molecular modelling insights of dual DNA binders/DHFR inhibitors bearing arylidene-hydrazinyl-1,3-thiazole scaffold with apoptotic and anti-migratory potential in breast MCF-7 cancer cells.

Authors: El-Wakil, Marwa H. Ghazala, Rasha A. El-Dershaby, Hadeel A. et al.

Source: Journal of Enzyme Inhibition & Medicinal Chemistry. Dec2025, Vol. 40 Issue 1, p1-21. 21p.

Recent advances in the synthesis, reactivity, and applications of symmetrical and asymmetrical cross-conjugated dienones.

Authors: Mouhib, Ayoub Es-Sounni, Bouchra Mouzdahir, Abdelkrim et al.

Source: Journal of the Iranian Chemical Society. Feb2025, Vol. 22 Issue 2, p243-262. 20p.

Design, synthesis, molecular docking, and antibacterial activity of novel amide-linked tetrahydrobenzothienopyrimidinone derivatives as potential DNA gyrase and topoisomerase IV inhibitors.

Authors: Mohamed, Mamdouh F. A. Soliman, Ahmed M. Alshazly, Omar et al.

Source: Medicinal Chemistry Research. Jan2025, Vol. 34 Issue 1, p172-182. 11p.

Novel pyrazole carboxylate derivatives as lonazolac bioisosteres with selective COX-2 inhibition: design, synthesis and anti-inflammatory activity.

Authors: Fadaly WAA Elshewy A Abusabaa AHA et al.

Source: Molecular diversity [Mol Divers] 2026 Feb; Vol. 30 (1), pp. 933-958. Date of Electronic Publication: 2025 May 22.

Publication Type: Journal Article

Journal Info: Publisher: ESCOM Science Publishers Country of Publication: Netherlands NLM ID: 9516534 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1573-501X (Electronic) Linking ISSN: 13811991 NLM ISO Abbreviation: Mol Divers Subsets: MEDLINE

Molecularly diverse lonazolac-inspired pyrazole-cyanopyridin-2-one conjugates: design, synthesis, in vitro, in vivo and in silico studies as multi-target anti-inflammatory agents.

Authors: Aziz MA Malebari AM Ibrahim TS et al.

Source: Molecular diversity [Mol Divers] 2026 May 09. Date of Electronic Publication: 2026 May 09.

Publication Type: Journal Article

Journal Info: Publisher: ESCOM Science Publishers Country of Publication: Netherlands NLM ID: 9516534 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1573-501X (Electronic) Linking ISSN: 13811991 NLM ISO Abbreviation: Mol Divers Subsets: MEDLINE

Multi-targeted anti-Alzheimer's agents: Synthesis, biological evaluation, and molecular modeling study of some pyrazolopyridine hybrids.

Authors: Waly OM El-Sayed SM Ghaly MA et al.

Source: European journal of medicinal chemistry [Eur J Med Chem] 2023 Dec 15; Vol. 262, pp. 115880. Date of Electronic Publication: 2023 Oct 20.

Publication Type: Journal Article

Journal Info: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1768-3254 (Electronic) Linking ISSN: 02235234 NLM ISO Abbreviation: Eur J Med Chem Subsets: MEDLINE

Synthesis, Characterization and Study the Biological Activity for New Schiff Base Compound 2-(((1E,2E)-1,2-Diphenyl-2-((4-(E-1-(Thiazol-2-ylimino) Ethyl) Phenyl) Imino) Ethylidene) Amino) Phenol (DEAP).

Authors: Mahdi, Makarim A. Jasim, Layth S. Jamel, Hayder O.

Source: Journal of Nanostructures. Autumn2025, Vol. 15 Issue 4, p1595-1605. 11p.

Antiproliferative effect of indeno[1,2-d]thiazolo[3,2-a]pyrimidine analogues on IL-6 mediated STAT3 and role of the apoptotic pathway in albino Wistar rats of ethyl carbamate-induced lung carcinoma: In-silico, In-vitro, and In-vivo study.

Authors: Sonkar, Archana Bharti Verma, Abhishek Yadav, Sneha et al.

Source: Cancer Cell International. 6/26/2024, Vol. 24 Issue 1, p1-12. 12p.

Insights into synthesis, reactivity, and biological activity of N-isoindoline-1, 3-diones heterocycles: a systematic literature review.

Authors: Ou-Ichen, Zhor Boussetta, Abdelghani Ouchetto, Khadija et al.

Source: Journal of the Iranian Chemical Society. Jun2024, Vol. 21 Issue 6, p1453-1493. 41p.

Editorial: Recent advances in the research and development of kinase-inhibitory anticancer molecules.

Authors: Al-Karmalawy AA El-Subbagh HI Logoyda L et al.

Source: Frontiers in chemistry [Front Chem] 2023 Nov 09; Vol. 11, pp. 1328424. Date of Electronic Publication: 2023 Nov 09 (Print Publication: 2023).

Publication Type: Editorial

Journal Info: Publisher: Frontiers Media S.A Country of Publication: Switzerland NLM ID: 101627988 Publication Model: eCollection Cited Medium: Print ISSN: 2296-2646 (Print) Linking ISSN: 22962646 NLM ISO Abbreviation: Front Chem Subsets: PubMed not MEDLINE