Search Results - "Fallacara AL"

The Pyrazolo[3,4-d]Pyrimidine Derivative Si306 Encapsulated into Anti-GD2-Immunoliposomes as Therapeutic Treatment of Neuroblastoma.

Authors: Rango E Pastorino F Brignole C et al.

Source: Biomedicines [Biomedicines] 2022 Mar 12; Vol. 10 (3). Date of Electronic Publication: 2022 Mar 12.

Publication Type: Journal Article

Journal Info: Publisher: MDPI AG Country of Publication: Switzerland NLM ID: 101691304 Publication Model: Electronic Cited Medium: Print ISSN: 2227-9059 (Print) Linking ISSN: 22279059 NLM ISO Abbreviation: Biomedicines Subsets: PubMed not MEDLINE

Optimization of Aminoimidazole Derivatives as Src Family Kinase Inhibitors.

Authors: Francini CM Musumeci F Fallacara AL et al.

Source: Molecules (Basel, Switzerland) [Molecules] 2018 Sep 17; Vol. 23 (9). Date of Electronic Publication: 2018 Sep 17.

Publication Type: Journal Article

Journal Info: Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049 (Electronic) Linking ISSN: 14203049 NLM ISO Abbreviation: Molecules Subsets: MEDLINE

Si113-prodrugs selectively activated by plasmin against hepatocellular and ovarian carcinoma.

Authors: Rango E D'Antona L Iovenitti G et al.

Source: European journal of medicinal chemistry [Eur J Med Chem] 2021 Nov 05; Vol. 223, pp. 113653. Date of Electronic Publication: 2021 Jun 17.

Publication Type: Journal Article

Journal Info: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1768-3254 (Electronic) Linking ISSN: 02235234 NLM ISO Abbreviation: Eur J Med Chem Subsets: MEDLINE

3-Arylidene-N-hydroxyoxindoles: A New Class of Compounds Endowed with Antitumor Activity.

Authors: Musso L Cincinelli R Zuco V et al.

Source: ChemMedChem [ChemMedChem] 2016 Aug 19; Vol. 11 (16), pp. 1700-4. Date of Electronic Publication: 2016 Jun 17.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Wiley-VCH Country of Publication: Germany NLM ID: 101259013 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1860-7187 (Electronic) Linking ISSN: 18607179 NLM ISO Abbreviation: ChemMedChem Subsets: MEDLINE

Identification of Aminoimidazole and Aminothiazole Derivatives as Src Family Kinase Inhibitors.

Authors: Francini CM Fallacara AL Artusi R et al.

Source: ChemMedChem [ChemMedChem] 2015 Dec; Vol. 10 (12), pp. 2027-41. Date of Electronic Publication: 2015 Oct 30.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Wiley-VCH Country of Publication: Germany NLM ID: 101259013 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1860-7187 (Electronic) Linking ISSN: 18607179 NLM ISO Abbreviation: ChemMedChem Subsets: MEDLINE

The fight against the influenza A virus H1N1: synthesis, molecular modeling, and biological evaluation of benzofurazan derivatives as viral RNA polymerase inhibitors.

Authors: Pagano M Castagnolo D Bernardini M et al.

Source: ChemMedChem [ChemMedChem] 2014 Jan; Vol. 9 (1), pp. 129-50. Date of Electronic Publication: 2013 Nov 27.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Wiley-VCH Country of Publication: Germany NLM ID: 101259013 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1860-7187 (Electronic) Linking ISSN: 18607179 NLM ISO Abbreviation: ChemMedChem Subsets: MEDLINE

Predictive Gene Signature for Pyrazolopyrimidine Derivative c-Src Inhibitor 10a Sensitivity in Melanoma Cells.

Authors: Kucukkaraduman B Turk C Fallacara AL et al.

Source: ACS medicinal chemistry letters [ACS Med Chem Lett] 2020 Feb 18; Vol. 11 (5), pp. 928-932. Date of Electronic Publication: 2020 Feb 18 (Print Publication: 2020).

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE

Identification of a new family of pyrazolo[3,4-d]pyrimidine derivatives as multitarget Fyn-Blk-Lyn inhibitors active on B- and T-lymphoma cell lines.

Authors: Fallacara AL Passannanti R Mori M et al.

Source: European journal of medicinal chemistry [Eur J Med Chem] 2019 Nov 01; Vol. 181, pp. 111545. Date of Electronic Publication: 2019 Jul 18.

Publication Type: Journal Article

Journal Info: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1768-3254 (Electronic) Linking ISSN: 02235234 NLM ISO Abbreviation: Eur J Med Chem Subsets: MEDLINE

Proton Therapy and Src Family Kinase Inhibitor Combined Treatments on U87 Human Glioblastoma Multiforme Cell Line.

Authors: Cammarata FP Torrisi F Forte GI et al.

Source: International journal of molecular sciences [Int J Mol Sci] 2019 Sep 24; Vol. 20 (19). Date of Electronic Publication: 2019 Sep 24.

Publication Type: Journal Article

Journal Info: Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium: Internet ISSN: 1422-0067 (Electronic) Linking ISSN: 14220067 NLM ISO Abbreviation: Int J Mol Sci Subsets: MEDLINE

A New Strategy for Glioblastoma Treatment: In Vitro and In Vivo Preclinical Characterization of Si306, a Pyrazolo[3,4-d]Pyrimidine Dual Src/P-Glycoprotein Inhibitor.

Authors: Fallacara AL Zamperini C Podolski-Renić A et al.

Source: Cancers [Cancers (Basel)] 2019 Jun 19; Vol. 11 (6). Date of Electronic Publication: 2019 Jun 19.

Publication Type: Journal Article

Journal Info: Publisher: MDPI Country of Publication: Switzerland NLM ID: 101526829 Publication Model: Electronic Cited Medium: Print ISSN: 2072-6694 (Print) Linking ISSN: 20726694 NLM ISO Abbreviation: Cancers (Basel) Subsets: PubMed not MEDLINE

An Update on JAK Inhibitors.

Authors: Musumeci F Greco C Giacchello I et al.

Source: Current medicinal chemistry [Curr Med Chem] 2019; Vol. 26 (10), pp. 1806-1832.

Publication Type: Journal Article; Review

Journal Info: Publisher: Bentham Science Publishers Country of Publication: United Arab Emirates NLM ID: 9440157 Publication Model: Print Cited Medium: Internet ISSN: 1875-533X (Electronic) Linking ISSN: 09298673 NLM ISO Abbreviation: Curr Med Chem Subsets: MEDLINE

One-pot synthesis of spiro(indoline-3,4'-pyrazolo[3,4-b]pyridine)-5'-carbonitriles as p53-MDM2 interaction inhibitors.

Authors: Ibrahim HS Eldehna WM Fallacara AL et al.

Source: Future medicinal chemistry [Future Med Chem] 2018 Dec; Vol. 10 (24), pp. 2771-2789. Date of Electronic Publication: 2018 Dec 10.

Publication Type: Journal Article

Journal Info: Publisher: Taylor & Francis Country of Publication: England NLM ID: 101511162 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1756-8927 (Electronic) Linking ISSN: 17568919 NLM ISO Abbreviation: Future Med Chem Subsets: MEDLINE

Efficient optimization of pyrazolo[3,4-d]pyrimidines derivatives as c-Src kinase inhibitors in neuroblastoma treatment.

Authors: Molinari A Fallacara AL Di Maria S et al.

Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2018 Nov 15; Vol. 28 (21), pp. 3454-3457. Date of Electronic Publication: 2018 Sep 20.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE

Synthesis and biological evaluation of a library of hybrid derivatives as inhibitors of influenza virus PA-PB1 interaction.

Authors: D'Agostino I Giacchello I Nannetti G et al.

Source: European journal of medicinal chemistry [Eur J Med Chem] 2018 Sep 05; Vol. 157, pp. 743-758. Date of Electronic Publication: 2018 Aug 13.

Publication Type: Journal Article

Journal Info: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1768-3254 (Electronic) Linking ISSN: 02235234 NLM ISO Abbreviation: Eur J Med Chem Subsets: MEDLINE

Pyrrolo[2,3-d]pyrimidines active as Btk inhibitors.

Authors: Musumeci F Sanna M Greco C et al.

Source: Expert opinion on therapeutic patents [Expert Opin Ther Pat] 2017 Dec; Vol. 27 (12), pp. 1305-1318. Date of Electronic Publication: 2017 Jul 20.

Publication Type: Journal Article; Review

Journal Info: Publisher: Informa Healthcare Country of Publication: England NLM ID: 9516419 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1744-7674 (Electronic) Linking ISSN: 13543776 NLM ISO Abbreviation: Expert Opin Ther Pat Subsets: MEDLINE

Prodrugs of Pyrazolo[3,4-d]pyrimidines: From Library Synthesis to Evaluation as Potential Anticancer Agents in an Orthotopic Glioblastoma Model.

Authors: Vignaroli G Iovenitti G Zamperini C et al.

Source: Journal of medicinal chemistry [J Med Chem] 2017 Jul 27; Vol. 60 (14), pp. 6305-6320. Date of Electronic Publication: 2017 Jul 18.

Publication Type: Journal Article

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

Pyrazolo[3,4-d]pyrimidines-loaded human serum albumin (HSA) nanoparticles: Preparation, characterization and cytotoxicity evaluation against neuroblastoma cell line.

Authors: Fallacara AL Mancini A Zamperini C et al.

Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2017 Jul 15; Vol. 27 (14), pp. 3196-3200. Date of Electronic Publication: 2017 May 17.

Publication Type: Journal Article

Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE

Identification of new pyrrolo[2,3-d]pyrimidines as Src tyrosine kinase inhibitors in vitro active against Glioblastoma.

Authors: Musumeci F Fallacara AL Brullo C et al.

Source: European journal of medicinal chemistry [Eur J Med Chem] 2017 Feb 15; Vol. 127, pp. 369-378. Date of Electronic Publication: 2016 Dec 19.

Publication Type: Journal Article

Journal Info: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1768-3254 (Electronic) Linking ISSN: 02235234 NLM ISO Abbreviation: Eur J Med Chem Subsets: MEDLINE

Phenotype-based variation as a biomarker of sensitivity to molecularly targeted therapy in melanoma.

Authors: Senses KM Ghasemi M Akbar MW et al.

Source: MedChemComm [Medchemcomm] 2017 Jan 01; Vol. 8 (1), pp. 88-95. Date of Electronic Publication: 2016 Oct 27.

Publication Type: Journal Article

Journal Info: Publisher: Royal Society of Chemistry Country of Publication: England NLM ID: 101531525 Publication Model: Print-Electronic Cited Medium: Print ISSN: 2040-2503 (Print) Linking ISSN: 20402503 NLM ISO Abbreviation: Medchemcomm Subsets: PubMed not MEDLINE

Pyrrolo[2,3-d]Pyrimidines as Kinase Inhibitors.

Authors: Musumeci F Sanna M Grossi G et al.

Source: Current medicinal chemistry [Curr Med Chem] 2017; Vol. 24 (19), pp. 2059-2085.

Publication Type: Journal Article; Review

Journal Info: Publisher: Bentham Science Publishers Country of Publication: United Arab Emirates NLM ID: 9440157 Publication Model: Print Cited Medium: Internet ISSN: 1875-533X (Electronic) Linking ISSN: 09298673 NLM ISO Abbreviation: Curr Med Chem Subsets: MEDLINE