Search Results - "Hogendorf, Adam"

Unraveling psilocybin's therapeutic potential: behavioral and neuroplasticity insights in Wistar-Kyoto and Wistar male rat models of treatment-resistant depression.

Authors: Kolasa, Magdalena Nikiforuk, Agnieszka Korlatowicz, Agata et al.

Source: Psychopharmacology. Jul2025, Vol. 242 Issue 7, p1607-1625. 19p.

Subjects: Psilocybin, Neuroplasticity, Mental depression, Laboratory rats, Behavioral assessment, Brain-derived neurotrophic factor

Effects of ketamine optical isomers, psilocybin, psilocin and norpsilocin on time estimation and cognition in rats.

Authors: Popik, Piotr Hogendorf, Adam Bugno, Ryszard et al.

Source: Psychopharmacology. Jun2022, Vol. 239 Issue 6, p1689-1703. 15p. 3 Charts, 5 Graphs.

Subjects: Ketamine, Psilocybin, Cognition, Rats, Time perception in animals

Correction to: Unraveling psilocybin's therapeutic potential: behavioral and neuroplasticity insights in Wistar-Kyoto and Wistar male rat models of treatment-resistant depression.

Authors: Kolasa, Magdalena Nikiforuk, Agnieszka Korlatowicz, Agata et al.

Source: Psychopharmacology. Jun2025, Vol. 242 Issue 6, p1455-1455. 1p.

Neuroprotective and Neurite Outgrowth Stimulating Effects of New Low-Basicity 5-HT7 Receptor Agonists: In Vitro Study in Human Neuroblastoma SH-SY5Y Cells.

Authors: Jakubowska, Klaudia Hogendorf, Adam S. Gołda, Sławomir et al.

Source: Neurochemical Research. Aug2024, Vol. 49 Issue 8, p2179-2196. 18p.

2-Aminoimidazole-based antagonists of the 5-HT6 receptor – A new concept in aminergic GPCR ligand design.

Authors: Hogendorf, Adam S. Hogendorf, Agata Kurczab, Rafał et al.

Source: European Journal of Medicinal Chemistry. Oct2019, Vol. 179, p1-15. 15p.

Fluorinated indole-imidazole conjugates: Selective orally bioavailable 5-HT7 receptor low-basicity agonists, potential neuropathic painkillers.

Authors: Hogendorf, Adam S. Hogendorf, Agata Popiołek-Barczyk, Katarzyna et al.

Source: European Journal of Medicinal Chemistry. May2019, Vol. 170, p261-275. 15p.

N -Skatyltryptamines—Dual 5-HT 6 R/D 2 R Ligands with Antipsychotic and Procognitive Potential.

Authors: Hogendorf, Agata Hogendorf, Adam S. Kurczab, Rafał et al.

Source: Molecules. Aug2021, Vol. 26 Issue 15, p4605-4605. 1p.

Design and Synthesis of New Quinazolin-4-one Derivatives with Negative mGlu 7 Receptor Modulation Activity and Antipsychotic-Like Properties.

Authors: Kaczorowska, Katarzyna Stankiewicz, Anna Bugno, Ryszard et al.

Source: International Journal of Molecular Sciences. Feb2023, Vol. 24 Issue 3, p1981. 23p.

Radiolabeling and in vivo evaluation of [¹¹C]AGH-44: a potential lead structure to develop a positron emission tomography radioligand for the 5-HT7 receptor.

Authors: L'Estrade, Elina T. Petersen, Ida N. Xiong, Mengfei et al.

Source: Journal of Radioanalytical & Nuclear Chemistry. Nov2019, Vol. 322 Issue 2, p847-851. 5p. 3 Diagrams, 2 Charts, 3 Graphs.

Serotonin type 5A receptor antagonists inhibit D-lysergic acid diethylamide discriminatory cue in rats.

Authors: Popik, Piotr Krawczyk, Martyna Kuziak, Agata et al.

Source: Journal of Psychopharmacology. Nov2019, Vol. 33 Issue 11, p1447-1455. 9p.

Design, synthesis, and biological evaluation of novel combretastatin A-4 thio derivatives as microtubule targeting agents.

Authors: Stefański, Tomasz Mikstacka, Renata Kurczab, Rafał et al.

Source: European Journal of Medicinal Chemistry. Jan2018, Vol. 144, p797-816. 20p.

Tuning the activity of known drugs via the introduction of halogen atoms, a case study of SERT ligands – Fluoxetine and fluvoxamine.

Authors: Staroń, Jakub Pietruś, Wojciech Bugno, Ryszard et al.

Source: European Journal of Medicinal Chemistry. Aug2021, Vol. 220, pN.PAG-N.PAG. 1p.

How can fluorine directly and indirectly affect the hydrogen bonding in molecular systems? – A case study for monofluoroanilines.

Authors: Pietruś, Wojciech Kurczab, Rafał Kafel, Rafał et al.

Source: Spectrochimica Acta Part A: Molecular & Biomolecular Spectroscopy. May2021, Vol. 252, pN.PAG-N.PAG. 1p.

Rationally designed N-phenylsulfonylindoles as a tool for the analysis of the non-basic 5-HT6R ligands binding mode.

Authors: Staroń, Jakub Bugno, Ryszard Pietruś, Wojciech et al.

Source: European Journal of Medicinal Chemistry. Jan2021, Vol. 209, pN.PAG-N.PAG. 1p.

Distinct cognitive and discriminative stimulus effects of ketamine enantiomers in rats.

Authors: Popik, Piotr Khoo, Shaun Yon-Seng Kuziak, Agata et al.

Source: Pharmacology, Biochemistry & Behavior. Oct2020, Vol. 197, pN.PAG-N.PAG. 1p.

Virtual screening-driven discovery of dual 5-HT6/5-HT2A receptor ligands with pro-cognitive properties.

Authors: Staroń, Jakub Kurczab, Rafał Warszycki, Dawid et al.

Source: European Journal of Medicinal Chemistry. Jan2020, Vol. 185, pN.PAG-N.PAG. 1p.

Chronic 5-HT7R activation drives depressive phenotypes and synaptic dysfunction.

Authors: Pochwat B Masternak J Bobula B et al.

Source: Acta pharmacologica Sinica [Acta Pharmacol Sin] 2026 Jun; Vol. 47 (6), pp. 1454-1470. Date of Electronic Publication: 2026 Feb 03.

Publication Type: Journal Article

Journal Info: Publisher: Nature Publishing Group Country of Publication: United States NLM ID: 100956087 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1745-7254 (Electronic) Linking ISSN: 16714083 NLM ISO Abbreviation: Acta Pharmacol Sin Subsets: MEDLINE

EVALUATION OF NEURITE OUTGROWTH INDUCED BY LOW-BASICITY 5-HT7 AGONISTS IN HUMAN NEUROBLASTOMA SH-SY5Y CELLS.

Authors: Jakubowska, Klaudia Gołda, Sławomir Hogendorf, Adam et al.

Source: Acta neurobiologiae experimentalis 2023 Supplement; Vol. 83.

Journal Info: Publisher: Acta Neurobiologiae Experimentalis ISSN: 0065-1400

Widespread false negatives in DNA-encoded library data: how linker effects impair machine learning-based lead prediction.

Authors: Montoya AL Hogendorf AS Tingey S et al.

Source: Chemical science [Chem Sci] 2025 May 09; Vol. 16 (24), pp. 10918-10927. Date of Electronic Publication: 2025 May 09 (Print Publication: 2025).

Publication Type: Journal Article

Journal Info: Publisher: Royal Society of Chemistry Country of Publication: England NLM ID: 101545951 Publication Model: eCollection Cited Medium: Print ISSN: 2041-6520 (Print) Linking ISSN: 20416520 NLM ISO Abbreviation: Chem Sci Subsets: PubMed not MEDLINE

Activation of the 5-HT7 receptor and MMP-9 signaling module in the hippocampal CA1 region is necessary for the development of depressive-like behavior.

Authors: Bijata M Bączyńska E Müller FE et al.

Source: Cell reports [Cell Rep] 2022 Mar 15; Vol. 38 (11), pp. 110532.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Cell Press Country of Publication: United States NLM ID: 101573691 Publication Model: Print Cited Medium: Internet ISSN: 2211-1247 (Electronic) NLM ISO Abbreviation: Cell Rep Subsets: MEDLINE