Search Results - "Hummersone, Marc G."

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  1. 1

    Optimization of potent and selective dual mTORC1 and mTORC2 inhibitors: The discovery of AZD8055 and AZD2014

    Authors: Pike, Kurt G. Malagu, Karine Hummersone, Marc G. et al.

    Source: Bioorganic & Medicinal Chemistry Letters. Mar2013, Vol. 23 Issue 5, p1212-1216. 5p.

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  2. 2

    On and off-target effects of telomere uncapping G-quadruplex selective ligands based on pentacyclic acridinium salts.

    Authors: Sara Iachettini Stevens, Malcolm F. G. Frigerio, Mark et al.

    Source: Journal of Experimental & Clinical Cancer Research (17569966). 2013, Vol. 32 Issue 1, p1-12. 12p.

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  3. 3

    1-Substituted(Dibenzo[b,d]thiophen-4-yl)-2-morpholino-4H-chromen-4-onesEndowed with Dual DNA-PK/PI3-K Inhibitory Activity.

    Authors: Cano, Céline Saravanan, Kappusamy Bailey, Chris et al.

    Source: Journal of Medicinal Chemistry. Vol. 56 Issue 16, p6386-6401. 16p.

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  4. 4

    DNA-Dependent Protein Kinase (DNA-PK) Inhibitors. Synthesis and Biological Activity of Quinolin-4-one and Pyridopyrimidin-4-one Surrogates for the Chromen-4-one Chemotype.

    Authors: Cano, Céline Barbeau, Olivier R. Bailey, Christine et al.

    Source: Journal of Medicinal Chemistry. 12/23/2010, Vol. 53 Issue 24, p8498-8507. 10p.

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  5. 5

    Synthesis and growth-inhibitory activities of imidazo[5,1-d]-1,2,3,5-tetrazine-8-carboxamides related to the anti-tumour drug temozolomide, with appended silicon, benzyl and heteromethyl groups at the 3-position.

    Authors: Cousin D Hummersone MG Bradshaw TD et al.

    Source: MedChemComm [Medchemcomm] 2018 Jan 19; Vol. 9 (3), pp. 545-553. Date of Electronic Publication: 2018 Jan 19 (Print Publication: 2018).

    Publication Type: Journal Article

    Journal Info: Publisher: Royal Society of Chemistry Country of Publication: England NLM ID: 101531525 Publication Model: eCollection Cited Medium: Print ISSN: 2040-2503 (Print) Linking ISSN: 20402503 NLM ISO Abbreviation: Medchemcomm Subsets: PubMed not MEDLINE

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  6. 6

    Pyranone, thiopyranone, and pyridone inhibitors of phosphatidylinositol 3-kinase related kinases. Structure-activity relationships for DNA-dependent protein kinase inhibition, and identification of the first potent and selective inhibitor of the ataxia telangiectasia mutated kinase.

    Authors: Hollick JJ Rigoreau LJ Cano-Soumillac C et al.

    Source: Journal of medicinal chemistry [J Med Chem] 2007 Apr 19; Vol. 50 (8), pp. 1958-72. Date of Electronic Publication: 2007 Mar 20.

    Publication Type: Journal Article

    Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Print ISSN: 0022-2623 (Print) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

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  7. 7

    Enantioselective formal total synthesis of the antitumor macrolide bryostatin 7.

    Authors: Manaviazar S Frigerio M Bhatia GS et al.

    Source: Organic letters [Org Lett] 2006 Sep 28; Vol. 8 (20), pp. 4477-80.

    Publication Type: Journal Article; Research Support, Non-U.S. Gov't

    Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 100890393 Publication Model: Print Cited Medium: Print ISSN: 1523-7060 (Print) Linking ISSN: 15237052 NLM ISO Abbreviation: Org Lett Subsets: MEDLINE

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  8. 8

    Synthesis of a simplified bryostatin C-ring analogue that binds to the CRD2 of human PKC-alpha and construction of a novel BC-analogue by an unusual Julia olefination process.

    Authors: Hale KJ Frigerio M Manaviazar S et al.

    Source: Organic letters [Org Lett] 2003 Feb 20; Vol. 5 (4), pp. 499-502.

    Publication Type: Journal Article; Research Support, Non-U.S. Gov't

    Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 100890393 Publication Model: Print Cited Medium: Print ISSN: 1523-7060 (Print) Linking ISSN: 15237052 NLM ISO Abbreviation: Org Lett Subsets: MEDLINE

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  9. 9

    The chemistry and biology of the bryostatin antitumour macrolides.

    Authors: Hale KJ Hummersone MG Manaviazar S et al.

    Source: Natural product reports [Nat Prod Rep] 2002 Aug; Vol. 19 (4), pp. 413-53.

    Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Review

    Journal Info: Publisher: Royal Society of Chemistry Country of Publication: England NLM ID: 8502408 Publication Model: Print Cited Medium: Print ISSN: 0265-0568 (Print) Linking ISSN: 02650568 NLM ISO Abbreviation: Nat Prod Rep Subsets: MEDLINE

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