Search Results - "McCombie SW"

Exploring chalcone-sulfonyl piperazine hybrids as anti-diabetes candidates: design, synthesis, biological evaluation, and molecular docking study.

Authors: Hosseini Nasab N Raza H Eom YS et al.

Source: Molecular diversity [Mol Divers] 2025 Feb; Vol. 29 (1), pp. 43-59. Date of Electronic Publication: 2024 May 22.

Publication Type: Journal Article

Journal Info: Publisher: ESCOM Science Publishers Country of Publication: Netherlands NLM ID: 9516534 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1573-501X (Electronic) Linking ISSN: 13811991 NLM ISO Abbreviation: Mol Divers Subsets: MEDLINE

Thermochemistry of Solution, Solvation and Hydrogen Bonding of Chloroform in Linear and Cyclic Ethers.

Authors: Rakipov, Ilnaz T. Semenov, Konstantin N. Petrov, Artem A. et al.

Source: Journal of Solution Chemistry. Feb2021, Vol. 50 Issue 2, p290-298. 9p.

Estimation of maximum recommended therapeutic dose of anti-retroviral drugs using diversified sampling and varied descriptors.

Authors: SAHU, Roopshikha YADAV, Amisha NATH, Abhigyan

Source: Minerva Biotechnology & Biomolecular Research. Dec2021, Vol. 33 Issue 4, p210-218. 9p.

Drug metabolic stability in early drug discovery to develop potential lead compounds.

Authors: Gajula, Siva Nageswara Rao Nadimpalli, Nimisha Sonti, Rajesh

Source: Drug Metabolism Reviews. Aug 2021, Vol. 53 Issue 3, p459-477. 19p.

HIV-1 predisposed to acquiring resistance to maraviroc (MVC) and other CCR5 antagonists in vitro has an inherent, low-level ability to utilize MVC-bound CCR5 for entry.

Source: Retrovirology. 2011, Vol. 8 Issue 1, p89-95. 7p. 4 Graphs.

The chemokine system and CCR5 antagonists: potential in HIV treatment and other novel therapies.

Authors: Dhami, H. Fritz, C. E. Gankin, B. et al.

Source: Journal of Clinical Pharmacy & Therapeutics. Apr2009, Vol. 34 Issue 2, p147-160. 14p. 3 Diagrams, 2 Charts.

Structural modification of the tripeptide KPV by reductive “glycoalkylation” of the lysine residue.

Authors: Songok, Abigael C. Panta, Pradip Doerrler, William T. et al.

Source: PLoS ONE. 6/28/2018, Vol. 13 Issue 6, p1-14. 14p.

The interconnected role of chemokines and estrogen in bone metabolism.

Authors: Yingping Xu Nan Chu Xuemin Qiu et al.

Source: BioScience Trends. Dec2016, Vol. 10 Issue 6, p433-444. 12p.

Stereoselective construction of skipped polyol enabled by oxonia-Cope rearrangement and iodolactonization: enantioselective synthesis of (+)-yashabushitriol.

Authors: He, Guoli Wang, Yan Lai, Calvine et al.

Source: SCIENCE CHINA Chemistry. Sep2016, Vol. 59 Issue 9, p1197-1204. 8p.

Modern Methods for Total Synthesis of Important Oxindole Alkaloids.

Authors: Fonseca, German O. Cook, James M.

Source: Organic Chemistry Insights. 2016, Issue 6, p1-55. 55p.

Synthesis of 1-benzhydryl piperazine derivatives and evaluation of their ACE inhibition and antimicrobial activities.

Authors: Santhoshi, Amlipur Kumar, Singam Sujitha, Pombala et al.

Source: Medicinal Chemistry Research. Jun2014, Vol. 23 Issue 6, p3207-3219. 13p.

A common mechanism of clinical HIV-1 resistance to the CCR5 antagonist maraviroc despite divergent resistance levels and lack of common gp120 resistance mutations.

Authors: Roche, Michael Salimi, Hamid Duncan, Renee et al.

Source: Retrovirology. 2013, Vol. 10 Issue 1, p1-20. 20p. 2 Diagrams, 3 Charts, 8 Graphs.

Modifications to five-substituted 3,3-diethyl-4,5-dihydro-2(3 H)-furanones en route to novel muscarinic receptor ligands.

Authors: Bhandare, Richie Canney, Daniel

Source: Medicinal Chemistry Research. Jun2011, Vol. 20 Issue 5, p558-565. 8p.

SmI-promoted imino-Reformatsky reaction for facile synthesis of enantioenriched β-amino acid esters.

Authors: Wang, Li Shen, Chun Xu, Ming-Hua

Source: SCIENCE CHINA Chemistry. Jan2011, Vol. 54 Issue 1, p61-65. 5p.

PEG-related polymer resins as synthetic supports.

Authors: Wang, Zheng Yang, RuLei Zhu, JunDong et al.

Source: SCIENCE CHINA Chemistry. Sep2010, Vol. 53 Issue 9, p1844-1852. 9p.

Conformational HIV-1 Envelope on particulate structures: a tool for chemokine coreceptor binding studies.

Authors: Tagliamonte, Maria Tornesello, Maria Lina Buonaguro, Franco M. et al.

Source: Journal of Translational Medicine. 2010 Supplement 1, p1-10. 10p. 2 Diagrams.

Two HIV-1 Variants Resistant to Small Molecule CCR5 Inhibitors Differ in How They Use CCR5 for Entry.

Authors: Berro, Reem Sanders, Rogier W. Min Lu et al.

Source: PLoS Pathogens. Aug2009, Vol. 5 Issue 8, p1-17. 17p. 1 Color Photograph, 2 Diagrams, 3 Charts, 8 Graphs.

6-Azathymidine-4'-thionucleosides: synthesis and antiviral evaluation.

Authors: Jasamai, Malina Balzarini, Jan Simons, Claire

Source: Journal of Enzyme Inhibition & Medicinal Chemistry. Feb2008, Vol. 23 Issue 1, p56-61. 6p. 3 Diagrams, 2 Charts.

Fused Indole-Diazepines with a Bridgehead Nitrogen Atom: Synthesis and Pharmaceutical Significance.

Authors: Zhou M Yang X Wang S

Source: Drug design, development and therapy [Drug Des Devel Ther] 2026 Apr 08; Vol. 20, pp. 554857. Date of Electronic Publication: 2026 Apr 08 (Print Publication: 2026).

Publication Type: Journal Article; Review

Journal Info: Publisher: Dove Press Limited Country of Publication: New Zealand NLM ID: 101475745 Publication Model: eCollection Cited Medium: Internet ISSN: 1177-8881 (Electronic) Linking ISSN: 11778881 NLM ISO Abbreviation: Drug Des Devel Ther Subsets: MEDLINE

Antipsoriatic effects of avarol-3′-thiosalicylate are mediated by inhibition of TNF-α generation and NF-κB activation in mouse skin.

Authors: Amigó, M. Payá, M. De Rosa, S. et al.

Source: British Journal of Pharmacology. Oct2007, Vol. 152 Issue 3, p353-365. 13p. 4 Black and White Photographs, 1 Diagram, 2 Charts, 5 Graphs.