Search Results - "Mocking TAM"

From dual norepinephrine-dopamine reuptake inhibition to selective dopamine reuptake inhibitors: a case of aromatically substituted N,2-cyclopentylamines.

Authors: Dilweg MA Jespers W Kasture AS et al.

Source: RSC medicinal chemistry [RSC Med Chem] 2026 Jun 24; Vol. 17 (7), pp. 3447-3462. Date of Electronic Publication: 2026 Jun 24 (Print Publication: 2026).

Publication Type: Journal Article

Journal Info: Publisher: Royal Society of Chemistry Country of Publication: England NLM ID: 101759460 Publication Model: eCollection Cited Medium: Internet ISSN: 2632-8682 (Electronic) Linking ISSN: 26328682 NLM ISO Abbreviation: RSC Med Chem Subsets: PubMed not MEDLINE

The solute carrier superfamily interactome.

Authors: Frommelt F Ladurner R Goldmann U et al.

Source: Molecular systems biology [Mol Syst Biol] 2025 Jun; Vol. 21 (6), pp. 632-675. Date of Electronic Publication: 2025 May 12.

Publication Type: Journal Article

Journal Info: Publisher: EMBO Press Country of Publication: Germany NLM ID: 101235389 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1744-4292 (Electronic) Linking ISSN: 17444292 NLM ISO Abbreviation: Mol Syst Biol Subsets: MEDLINE

Advancing drug discovery through assay development: a survey of tool compounds within the human solute carrier superfamily.

Authors: Digles D Ingles-Prieto A Dvorak V et al.

Source: Frontiers in pharmacology [Front Pharmacol] 2024 Jul 09; Vol. 15, pp. 1401599. Date of Electronic Publication: 2024 Jul 09 (Print Publication: 2024).

Publication Type: Journal Article

Journal Info: Publisher: Frontiers Media] Country of Publication: Switzerland NLM ID: 101548923 Publication Model: eCollection Cited Medium: Print ISSN: 1663-9812 (Print) Linking ISSN: 16639812 NLM ISO Abbreviation: Front Pharmacol Subsets: PubMed not MEDLINE

Label-free detection of prostaglandin transporter (SLCO2A1) function and inhibition: insights by wound healing and TRACT assays.

Authors: Mocking TAM van Oostveen WM van Veldhoven JPD et al.

Source: Frontiers in pharmacology [Front Pharmacol] 2024 May 09; Vol. 15, pp. 1372109. Date of Electronic Publication: 2024 May 09 (Print Publication: 2024).

Publication Type: Journal Article

Journal Info: Publisher: Frontiers Media] Country of Publication: Switzerland NLM ID: 101548923 Publication Model: eCollection Cited Medium: Print ISSN: 1663-9812 (Print) Linking ISSN: 16639812 NLM ISO Abbreviation: Front Pharmacol Subsets: PubMed not MEDLINE

SAR exploration of the non-imidazole histamine H3 receptor ligand ZEL-H16 reveals potent inverse agonism.

Authors: Wágner G Mocking TAM Ma X et al.

Source: Archiv der Pharmazie [Arch Pharm (Weinheim)] 2023 Jan; Vol. 356 (1), pp. e2200451. Date of Electronic Publication: 2022 Oct 30.

Publication Type: Journal Article

Journal Info: Publisher: Wiley-VCH Verlag GmbH & Co. KGaA Country of Publication: Germany NLM ID: 0330167 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1521-4184 (Electronic) Linking ISSN: 03656233 NLM ISO Abbreviation: Arch Pharm (Weinheim) Subsets: MEDLINE

Stereochemical optimization of N,2-substituted cycloalkylamines as norepinephrine reuptake inhibitors.

Authors: Dilweg MA Mocking TAM Maragkoudakis P et al.

Source: RSC medicinal chemistry [RSC Med Chem] 2024 Sep 12. Date of Electronic Publication: 2024 Sep 12.

Publication Type: Journal Article

Journal Info: Publisher: Royal Society of Chemistry Country of Publication: England NLM ID: 101759460 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2632-8682 (Electronic) Linking ISSN: 26328682 NLM ISO Abbreviation: RSC Med Chem

Still in Search for an EAAT Activator: GT949 Does Not Activate EAAT2, nor EAAT3 in Impedance and Radioligand Uptake Assays.

Authors: van Veggel L Mocking TAM Sijben HJ et al.

Source: ACS chemical neuroscience [ACS Chem Neurosci] 2024 Apr 03; Vol. 15 (7), pp. 1424-1431. Date of Electronic Publication: 2024 Mar 13.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101525337 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1948-7193 (Electronic) Linking ISSN: 19487193 NLM ISO Abbreviation: ACS Chem Neurosci Subsets: MEDLINE

Covalent Inhibition of the Histamine H3 Receptor.

Authors: Wágner G Mocking TAM Kooistra AJ et al.

Source: Molecules (Basel, Switzerland) [Molecules] 2019 Dec 11; Vol. 24 (24). Date of Electronic Publication: 2019 Dec 11.

Publication Type: Journal Article

Journal Info: Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049 (Electronic) Linking ISSN: 14203049 NLM ISO Abbreviation: Molecules Subsets: MEDLINE

Optimization of Peptide Linker-Based Fluorescent Ligands for the Histamine H1 Receptor.

Authors: Kok ZY Stoddart LA Mistry SJ et al.

Source: Journal of medicinal chemistry [J Med Chem] 2022 Jun 23; Vol. 65 (12), pp. 8258-8288. Date of Electronic Publication: 2022 Jun 03.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

MPP⁺-Induced Changes in Cellular Impedance as a Measure for Organic Cation Transporter (SLC22A1-3) Activity and Inhibition.

Authors: Mocking TAM Sijben HJ Vermeulen YW et al.

Source: International journal of molecular sciences [Int J Mol Sci] 2022 Jan 21; Vol. 23 (3). Date of Electronic Publication: 2022 Jan 21.

Publication Type: Journal Article

Journal Info: Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium: Internet ISSN: 1422-0067 (Electronic) Linking ISSN: 14220067 NLM ISO Abbreviation: Int J Mol Sci Subsets: MEDLINE

4-(3-Aminoazetidin-1-yl)pyrimidin-2-amines as High-Affinity Non-imidazole Histamine H3 Receptor Agonists with in Vivo Central Nervous System Activity.

Authors: Wágner G Mocking TAM Arimont M et al.

Source: Journal of medicinal chemistry [J Med Chem] 2019 Dec 12; Vol. 62 (23), pp. 10848-10866. Date of Electronic Publication: 2019 Nov 20.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

A toolbox of molecular photoswitches to modulate the CXCR3 chemokine receptor with light.

Authors: Gómez-Santacana X de Munnik SM Mocking TAM et al.

Source: Beilstein journal of organic chemistry [Beilstein J Org Chem] 2019 Oct 23; Vol. 15, pp. 2509-2523. Date of Electronic Publication: 2019 Oct 23 (Print Publication: 2019).

Publication Type: Journal Article

Journal Info: Publisher: Beilstein-Institut Country of Publication: Germany NLM ID: 101250746 Publication Model: eCollection Cited Medium: Print ISSN: 1860-5397 (Print) Linking ISSN: 18605397 NLM ISO Abbreviation: Beilstein J Org Chem Subsets: PubMed not MEDLINE

Bioluminescence Resonance Energy Transfer Based G Protein-Activation Assay to Probe Duration of Antagonism at the Histamine H3 Receptor.

Authors: Mocking TAM Buzink MCML Leurs R et al.

Source: International journal of molecular sciences [Int J Mol Sci] 2019 Jul 30; Vol. 20 (15). Date of Electronic Publication: 2019 Jul 30.

Publication Type: Journal Article

Journal Info: Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium: Internet ISSN: 1422-0067 (Electronic) Linking ISSN: 14220067 NLM ISO Abbreviation: Int J Mol Sci Subsets: MEDLINE

A Photoswitchable Agonist for the Histamine H3 Receptor, a Prototypic Family A G-Protein-Coupled Receptor.

Authors: Hauwert NJ Mocking TAM Da Costa Pereira D et al.

Source: Angewandte Chemie (International ed. in English) [Angew Chem Int Ed Engl] 2019 Mar 26; Vol. 58 (14), pp. 4531-4535. Date of Electronic Publication: 2019 Feb 27.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Wiley-VCH Country of Publication: Germany NLM ID: 0370543 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1521-3773 (Electronic) Linking ISSN: 14337851 NLM ISO Abbreviation: Angew Chem Int Ed Engl Subsets: MEDLINE

Homogeneous, Real-Time NanoBRET Binding Assays for the Histamine H3 and H4 Receptors on Living Cells.

Authors: Mocking TAM Verweij EWE Vischer HF et al.

Source: Molecular pharmacology [Mol Pharmacol] 2018 Dec; Vol. 94 (6), pp. 1371-1381. Date of Electronic Publication: 2018 Sep 24.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Elsevier Country of Publication: Netherlands NLM ID: 0035623 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1521-0111 (Electronic) Linking ISSN: 0026895X NLM ISO Abbreviation: Mol Pharmacol Subsets: MEDLINE

Synthesis and Characterization of a Bidirectional Photoswitchable Antagonist Toolbox for Real-Time GPCR Photopharmacology.

Authors: Hauwert NJ Mocking TAM Da Costa Pereira D et al.

Source: Journal of the American Chemical Society [J Am Chem Soc] 2018 Mar 28; Vol. 140 (12), pp. 4232-4243. Date of Electronic Publication: 2018 Mar 14.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 7503056 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-5126 (Electronic) Linking ISSN: 00027863 NLM ISO Abbreviation: J Am Chem Soc Subsets: MEDLINE