Search Results - "Reboud-Ravaux M"

N-Acetylbenzotriazole hydrolysis and aminolysis.

Authors: Reboud-Ravaux, M.

Source: Journal of the American Chemical Society; January 30 1980, Vol. 102, p1039-1046, 8p

Efficient Synthesis and Biological Evaluation of 1,4-Disubstituted 3-Cyanopyridin-2(1H)-ones as Selective Inhibitors of the Post-Acid Activity of Mammalian 20S Proteasomes.

Authors: Karapetyan, L. V. Tokmajyan, G. G. Melikyan, G. S. et al.

Source: Russian Journal of Organic Chemistry. Mar2025, Vol. 61 Issue 3, p449-455. 7p.

3-Bromophenyl 6-acetoxymethyl-2-oxo-2H-1-benzopyran-3-carboxylate inhibits cancer cell invasion in vitro and tumour growth in vivo.

Authors: Kempen, I Papapostolou, D Thierry, N et al.

Source: British Journal of Cancer. 4/7/2003, Vol. 88 Issue 7, p1111-1118. 8p.

[Protein induced proximity and targeted degradations by new degraders: concepts, developments, challenges for clinical applications].

Transliterated Title: Induction de proximité et dégradation de cibles thérapeutiques par les nouveaux dégradeurs : quels concepts, quels développements, quel futur ?

Authors: Reboud-Ravaux M; Sorbonne Université, Institut de Biologie Paris Seine (IBPS), CNRS UMR 8256, Inserm ERL U1164, 7 quai Saint-Bernard, 75252 Paris, France.

Source: Biologie aujourd'hui [Biol Aujourdhui] 2024; Vol. 218 (1-2), pp. 41-54. Date of Electronic Publication: 2024 Jul 15.

Publication Type: Journal Article; Review; English Abstract

Journal Info: Publisher: La Société de biologie Country of Publication: France NLM ID: 101544020 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2105-0686 (Electronic) Linking ISSN: 21050678 NLM ISO Abbreviation: Biol Aujourdhui Subsets: MEDLINE

Genuine selective caspase-2 inhibition with new irreversible small peptidomimetics.

Authors: Bosc E Anastasie J Soualmia F et al.

Source: Cell death & disease [Cell Death Dis] 2022 Nov 15; Vol. 13 (11), pp. 959. Date of Electronic Publication: 2022 Nov 15.

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Nature Pub. Group Country of Publication: England NLM ID: 101524092 Publication Model: Electronic Cited Medium: Internet ISSN: 2041-4889 (Electronic) NLM ISO Abbreviation: Cell Death Dis Subsets: MEDLINE

[The proteasome - structural aspects and inhibitors: a second life for a validated drug target].

Transliterated Title: Le protéasome, la seconde vie d’une cible thérapeutique validée : aspects structuraux et nouveaux inhibiteurs.

Authors: Reboud-Ravaux M; Sorbonne Université, Institut de Biologie Paris Seine (IBPS), CNRS UMR 8256, Inserm ERL U1164, 7 quai Saint Bernard, 75252 Paris Cedex 05, France.

Source: Biologie aujourd'hui [Biol Aujourdhui] 2021; Vol. 215 (1-2), pp. 1-23. Date of Electronic Publication: 2021 Aug 16.

Publication Type: Journal Article

Journal Info: Publisher: La Société de biologie Country of Publication: France NLM ID: 101544020 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2105-0686 (Electronic) Linking ISSN: 21050678 NLM ISO Abbreviation: Biol Aujourdhui Subsets: MEDLINE

[Induced degradation of proteins by PROTACs and other strategies: towards promising drugs].

Transliterated Title: Dégradation induite des protéines par des molécules PROTAC et stratégies apparentées : développements à visée thérapeutique.

Authors: Reboud-Ravaux M; Sorbonne Université, Institut de Biologie Paris Seine (IBPS), CNRS UMR 8256, Inserm ERL U1164, 7 quai Saint-Bernard, 75252 Paris Cedex 05, France.

Source: Biologie aujourd'hui [Biol Aujourdhui] 2021; Vol. 215 (1-2), pp. 25-43. Date of Electronic Publication: 2021 Aug 16.

Publication Type: Journal Article

Journal Info: Publisher: La Société de biologie Country of Publication: France NLM ID: 101544020 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2105-0686 (Electronic) Linking ISSN: 21050678 NLM ISO Abbreviation: Biol Aujourdhui Subsets: MEDLINE

Transliterated Title: Erratum : Dégradation induite des protéines par des molécules PROTAC et stratégies apparentées : développements à visée thérapeutique - Biologie Aujourd’hui 215 (1-2), 25-43 (2021) https://doi.org/10.1051/jbio/2021007.

Authors: Reboud-Ravaux M; Sorbonne Université, Institut de Biologie Paris Seine (IBPS), CNRS UMR 8256, Inserm ERL U1164, 7 quai Saint-Bernard, 75252 Paris Cedex 05, France.

Source: Biologie aujourd'hui [Biol Aujourdhui] 2021; Vol. 215 (3-4), pp. 143. Date of Electronic Publication: 2022 Mar 11.

Publication Type: Journal Article; Published Erratum

Journal Info: Publisher: La Société de biologie Country of Publication: France NLM ID: 101544020 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2105-0686 (Electronic) Linking ISSN: 21050678 NLM ISO Abbreviation: Biol Aujourdhui Subsets: MEDLINE; PubMed not MEDLINE

Insights into the activity control of the kallikrein-related peptidase 6: small-molecule modulators and allosterism.

Authors: Soualmia F Bosc E Amiri SA et al.

Source: Biological chemistry [Biol Chem] 2018 Sep 25; Vol. 399 (9), pp. 1073-1078.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Walter De Gruyter Country of Publication: Germany NLM ID: 9700112 Publication Model: Print Cited Medium: Internet ISSN: 1437-4315 (Electronic) Linking ISSN: 14316730 NLM ISO Abbreviation: Biol Chem Subsets: MEDLINE

The HIV-1 Nucleocapsid Regulates Its Own Condensation by Phase-Separated Activity-Enhancing Sequestration of the Viral Protease during Maturation.

Authors: Lyonnais S Sadiq SK Lorca-Oró C et al.

Source: Viruses [Viruses] 2021 Nov 19; Vol. 13 (11). Date of Electronic Publication: 2021 Nov 19.

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

Journal Info: Publisher: MDPI Country of Publication: Switzerland NLM ID: 101509722 Publication Model: Electronic Cited Medium: Internet ISSN: 1999-4915 (Electronic) Linking ISSN: 19994915 NLM ISO Abbreviation: Viruses Subsets: MEDLINE

Structural Studies on the Inhibitory Binding Mode of Aromatic Coumarinic Esters to Human Kallikrein-Related Peptidase 7.

Authors: Hanke S Tindall CA Pippel J et al.

Source: Journal of medicinal chemistry [J Med Chem] 2020 Jun 11; Vol. 63 (11), pp. 5723-5733. Date of Electronic Publication: 2020 May 21.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

Piperlongumine and some of its analogs inhibit selectively the human immunoproteasome over the constitutive proteasome.

Authors: Bosc E Nastri J Lefort V et al.

Source: Biochemical and biophysical research communications [Biochem Biophys Res Commun] 2018 Feb 12; Vol. 496 (3), pp. 961-966. Date of Electronic Publication: 2018 Feb 02.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Elsevier Country of Publication: United States NLM ID: 0372516 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1090-2104 (Electronic) Linking ISSN: 0006291X NLM ISO Abbreviation: Biochem Biophys Res Commun Subsets: MEDLINE

Structure-based design of human immuno- and constitutive proteasomes inhibitors.

Authors: Richy N Sarraf D Maréchal X et al.

Source: European journal of medicinal chemistry [Eur J Med Chem] 2018 Feb 10; Vol. 145, pp. 570-587. Date of Electronic Publication: 2018 Jan 08.

Publication Type: Journal Article

Journal Info: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1768-3254 (Electronic) Linking ISSN: 02235234 NLM ISO Abbreviation: Eur J Med Chem Subsets: MEDLINE

Phenoxypropanolamine derivatives as selective inhibitors of the 20S proteasome β1 and β5 subunits.

Authors: Hovhannisyan AA Pham TH Bouvier D et al.

Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2017 Dec 01; Vol. 27 (23), pp. 5172-5178. Date of Electronic Publication: 2017 Oct 23.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE

Blockade of the malignant phenotype by β-subunit selective noncovalent inhibition of immuno- and constitutive proteasomes.

Authors: Villoutreix BO Khatib AM Cheng Y et al.

Source: Oncotarget [Oncotarget] 2017 Feb 07; Vol. 8 (6), pp. 10437-10449.

Publication Type: Journal Article

Journal Info: Publisher: Impact Journals Country of Publication: United States NLM ID: 101532965 Publication Model: Print Cited Medium: Internet ISSN: 1949-2553 (Electronic) Linking ISSN: 19492553 NLM ISO Abbreviation: Oncotarget Subsets: MEDLINE

Identification of a β1/β2-specific sulfonamide proteasome ligand by crystallographic screening.

Authors: Beck P Reboud-Ravaux M Groll M

Source: Angewandte Chemie (International ed. in English) [Angew Chem Int Ed Engl] 2015 Sep 14; Vol. 54 (38), pp. 11275-8. Date of Electronic Publication: 2015 Aug 04.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Wiley-VCH Country of Publication: Germany NLM ID: 0370543 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1521-3773 (Electronic) Linking ISSN: 14337851 NLM ISO Abbreviation: Angew Chem Int Ed Engl Subsets: MEDLINE

Toward the first class of suicide inhibitors of kallikreins involved in skin diseases.

Authors: Tan X Soualmia F Furio L et al.

Source: Journal of medicinal chemistry [J Med Chem] 2015 Jan 22; Vol. 58 (2), pp. 598-612. Date of Electronic Publication: 2014 Dec 22.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

Bisbenzimidazole derivatives as potent inhibitors of the trypsin-like sites of the immunoproteasome core particle.

Authors: Koroleva ON Pham TH Bouvier D et al.

Source: Biochimie [Biochimie] 2015 Jan; Vol. 108, pp. 94-100. Date of Electronic Publication: 2014 Nov 13.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 1264604 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1638-6183 (Electronic) Linking ISSN: 03009084 NLM ISO Abbreviation: Biochimie Subsets: MEDLINE

Noncovalent fluorescent probes of human immuno- and constitutive proteasomes.

Authors: Desvergne A Cheng Y Grosay-Gaudrel S et al.

Source: Journal of medicinal chemistry [J Med Chem] 2014 Nov 13; Vol. 57 (21), pp. 9211-7. Date of Electronic Publication: 2014 Nov 04.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

Jatrophidin I, a cyclic peptide from Brazilian Jatropha curcas L.: isolation, characterization, conformational studies and biological activity.

Authors: Altei WF Picchi DG Abissi BM et al.

Source: Phytochemistry [Phytochemistry] 2014 Nov; Vol. 107, pp. 91-6. Date of Electronic Publication: 2014 Sep 05.

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

Journal Info: Publisher: Elsevier Country of Publication: England NLM ID: 0151434 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1873-3700 (Electronic) Linking ISSN: 00319422 NLM ISO Abbreviation: Phytochemistry Subsets: MEDLINE