Discovery of the First‐in‐Class Inhibitors of Hypoxia Up‐Regulated Protein 1 (HYOU1) Suppressing Pathogenic Fibroblast Activation.

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Title: Discovery of the First‐in‐Class Inhibitors of Hypoxia Up‐Regulated Protein 1 (HYOU1) Suppressing Pathogenic Fibroblast Activation.
Authors: Papadopoulou, Dimitra1, Mavrikaki, Vasiliki2,3, Charalampous, Filippos1, Tzaferis, Christos1, Samiotaki, Martina1, Papavasileiou, Konstantinos D.4,5,6, Afantitis, Antreas4,5,6, Karagianni, Niki7, Denis, Maria C.7, Sanchez, Julie8,9, Lane, J. Robert8,9, Faidon Brotzakis, Zacharias1,10, Skretas, Georgios1,11, Georgiadis, Dimitris3, Matralis, Alexios N.1, matralis@fleming.gr, Kollias, George1,12,13, kollias@fleming.gr
Source: Angewandte Chemie International Edition; 4/2/2024, Vol. 63 Issue 14, p1-13, 13p
Database: Applied Science & Technology Source
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ISSN:14337851
DOI:10.1002/anie.202319157