Design of selective PI3Kα inhibitors starting from a promiscuous pan kinase scaffold.
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| Title: | Design of selective PI3Kα inhibitors starting from a promiscuous pan kinase scaffold. |
|---|---|
| Authors: | Barlaam, Bernard1 bernard.barlaam2@astrazeneca.com, Cosulich, Sabina1, Fitzek, Martina1, Green, Stephen1, Harris, Craig S.2, Hudson, Kevin1, Lambert-van der Brempt, Christine2, Ouvry, Gilles2, Page, Ken1, Ruston, Linette1, Ward, Lara1, Delouvrié, Bénédicte2 |
| Source: | Bioorganic & Medicinal Chemistry Letters. Jul2015, Vol. 25 Issue 13, p2679-2685. 7p. |
| Database: | Academic Search Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: asn DbLabel: Academic Search Ultimate An: 102981720 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=asn&AN=102981720 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1016/j.bmcl.2015.04.084 Languages: – Code: eng Text: English PhysicalDescription: Pagination: PageCount: 7 StartPage: 2679 Titles: – TitleFull: Design of selective PI3Kα inhibitors starting from a promiscuous pan kinase scaffold. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Barlaam, Bernard – PersonEntity: Name: NameFull: Cosulich, Sabina – PersonEntity: Name: NameFull: Fitzek, Martina – PersonEntity: Name: NameFull: Green, Stephen – PersonEntity: Name: NameFull: Harris, Craig S. – PersonEntity: Name: NameFull: Hudson, Kevin – PersonEntity: Name: NameFull: Lambert-van der Brempt, Christine – PersonEntity: Name: NameFull: Ouvry, Gilles – PersonEntity: Name: NameFull: Page, Ken – PersonEntity: Name: NameFull: Ruston, Linette – PersonEntity: Name: NameFull: Ward, Lara – PersonEntity: Name: NameFull: Delouvrié, Bénédicte IsPartOfRelationships: – BibEntity: Dates: – D: 01 M: 07 Text: Jul2015 Type: published Y: 2015 Identifiers: – Type: issn-print Value: 0960894X Numbering: – Type: volume Value: 25 – Type: issue Value: 13 Titles: – TitleFull: Bioorganic & Medicinal Chemistry Letters Type: main |
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