Discovery of a novel aminopyrazine series as selective PI3Kα inhibitors.
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| Title: | Discovery of a novel aminopyrazine series as selective PI3Kα inhibitors. |
|---|---|
| Authors: | Barlaam, Bernard1 bernard.barlaam2@astrazeneca.com, Cosulich, Sabina1, Fitzek, Martina2, Germain, Hervé3, Green, Stephen2, Hanson, Lyndsey L.2, Harris, Craig S.3, Hancox, Urs2, Hudson, Kevin2, Lambert-van der Brempt, Christine3, Lamorlette, Maryannick3, Magnien, Françoise3, Ouvry, Gilles3, Page, Ken2, Ruston, Linette2, Ward, Lara2, Delouvrié, Bénédicte3 |
| Source: | Bioorganic & Medicinal Chemistry Letters. Jul2017, Vol. 27 Issue 13, p3030-3035. 6p. |
| Database: | Academic Search Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: asn DbLabel: Academic Search Ultimate An: 123258343 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=asn&AN=123258343 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1016/j.bmcl.2017.05.028 Languages: – Code: eng Text: English PhysicalDescription: Pagination: PageCount: 6 StartPage: 3030 Titles: – TitleFull: Discovery of a novel aminopyrazine series as selective PI3Kα inhibitors. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Barlaam, Bernard – PersonEntity: Name: NameFull: Cosulich, Sabina – PersonEntity: Name: NameFull: Fitzek, Martina – PersonEntity: Name: NameFull: Germain, Hervé – PersonEntity: Name: NameFull: Green, Stephen – PersonEntity: Name: NameFull: Hanson, Lyndsey L. – PersonEntity: Name: NameFull: Harris, Craig S. – PersonEntity: Name: NameFull: Hancox, Urs – PersonEntity: Name: NameFull: Hudson, Kevin – PersonEntity: Name: NameFull: Lambert-van der Brempt, Christine – PersonEntity: Name: NameFull: Lamorlette, Maryannick – PersonEntity: Name: NameFull: Magnien, Françoise – PersonEntity: Name: NameFull: Ouvry, Gilles – PersonEntity: Name: NameFull: Page, Ken – PersonEntity: Name: NameFull: Ruston, Linette – PersonEntity: Name: NameFull: Ward, Lara – PersonEntity: Name: NameFull: Delouvrié, Bénédicte IsPartOfRelationships: – BibEntity: Dates: – D: 01 M: 07 Text: Jul2017 Type: published Y: 2017 Identifiers: – Type: issn-print Value: 0960894X Numbering: – Type: volume Value: 27 – Type: issue Value: 13 Titles: – TitleFull: Bioorganic & Medicinal Chemistry Letters Type: main |
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