Discovery of a novel aminopyrazine series as selective PI3Kα inhibitors.

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Title: Discovery of a novel aminopyrazine series as selective PI3Kα inhibitors.
Authors: Barlaam, Bernard1 bernard.barlaam2@astrazeneca.com, Cosulich, Sabina1, Fitzek, Martina2, Germain, Hervé3, Green, Stephen2, Hanson, Lyndsey L.2, Harris, Craig S.3, Hancox, Urs2, Hudson, Kevin2, Lambert-van der Brempt, Christine3, Lamorlette, Maryannick3, Magnien, Françoise3, Ouvry, Gilles3, Page, Ken2, Ruston, Linette2, Ward, Lara2, Delouvrié, Bénédicte3
Source: Bioorganic & Medicinal Chemistry Letters. Jul2017, Vol. 27 Issue 13, p3030-3035. 6p.
Database: Academic Search Ultimate
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  Data: <searchLink fieldCode="JN" term="%22Bioorganic+%26+Medicinal+Chemistry+Letters%22">Bioorganic & Medicinal Chemistry Letters</searchLink>. Jul2017, Vol. 27 Issue 13, p3030-3035. 6p.
PLink https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=asn&AN=123258343
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      – Type: doi
        Value: 10.1016/j.bmcl.2017.05.028
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      – Code: eng
        Text: English
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        PageCount: 6
        StartPage: 3030
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              Text: Jul2017
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              Y: 2017
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