Structure-based design and synthesis of 2,4-diaminopyrimidines as EGFR L858R/T790M selective inhibitors for NSCLC.
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| Title: | Structure-based design and synthesis of 2,4-diaminopyrimidines as EGFR L858R/T790M selective inhibitors for NSCLC. |
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| Authors: | Chen, Lingfeng1,2, Fu, Weitao2, Feng, Chen2, Qu, Rong3, Tong, Linjiang3, Zheng, Lulu2, Fang, Bo2, Qiu, Yinda2, Hu, Jie2, Cai, Yuepiao2, Feng, Jianpeng2, Xie, Hua3, Ding, Jian3 jding@simm.ac.cn, Liu, Zhiguo2 lzgcnu@163.com, Liang, Guang1,2 wzmcliangguang@163.com |
| Source: | European Journal of Medicinal Chemistry. Nov2017, Vol. 140, p510-527. 18p. |
| Database: | Academic Search Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: asn DbLabel: Academic Search Ultimate An: 125723575 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=asn&AN=125723575 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1016/j.ejmech.2017.08.061 Languages: – Code: eng Text: English PhysicalDescription: Pagination: PageCount: 18 StartPage: 510 Titles: – TitleFull: Structure-based design and synthesis of 2,4-diaminopyrimidines as EGFR L858R/T790M selective inhibitors for NSCLC. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Chen, Lingfeng – PersonEntity: Name: NameFull: Fu, Weitao – PersonEntity: Name: NameFull: Feng, Chen – PersonEntity: Name: NameFull: Qu, Rong – PersonEntity: Name: NameFull: Tong, Linjiang – PersonEntity: Name: NameFull: Zheng, Lulu – PersonEntity: Name: NameFull: Fang, Bo – PersonEntity: Name: NameFull: Qiu, Yinda – PersonEntity: Name: NameFull: Hu, Jie – PersonEntity: Name: NameFull: Cai, Yuepiao – PersonEntity: Name: NameFull: Feng, Jianpeng – PersonEntity: Name: NameFull: Xie, Hua – PersonEntity: Name: NameFull: Ding, Jian – PersonEntity: Name: NameFull: Liu, Zhiguo – PersonEntity: Name: NameFull: Liang, Guang IsPartOfRelationships: – BibEntity: Dates: – D: 10 M: 11 Text: Nov2017 Type: published Y: 2017 Identifiers: – Type: issn-print Value: 02235234 Numbering: – Type: volume Value: 140 Titles: – TitleFull: European Journal of Medicinal Chemistry Type: main |
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