Discovery of N-(piperidin-3-yl)-N-(pyridin-2-yl)piperidine/piperazine-1-carboxamides as small molecule inhibitors of PCSK9. - Londregan, Allyn T.; Aspnes, Gary; Limberakis, Chris; Loria, Paula M.; McClure, Kim F.; Petersen, Donna N.; Raymer, Brian; Ruggeri, Roger B.; Wei, Liuqing; Xiao, Jun; Piotrowski, David W. (Bioorganic & Medicinal Chemistry Letters, 2018)