Discovery and optimization of novel pyridines as highly potent and selective glycogen synthase kinase 3 inhibitors.
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| Title: | Discovery and optimization of novel pyridines as highly potent and selective glycogen synthase kinase 3 inhibitors. |
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| Authors: | Ramurthy, Savithri1 (AUTHOR), Pfister, Keith B.2 (AUTHOR), Boyce, Rustum S.3 (AUTHOR), Brown, Sean P.4 (AUTHOR), Costales, Abran Q.5 (AUTHOR), Desai, Manoj C.6 (AUTHOR), Fang, Eric7 (AUTHOR), Levine, Barry H.8 (AUTHOR), Ng, Simon C.9 (AUTHOR), Nuss, John M.10 (AUTHOR), Ring, David B.11 (AUTHOR), Shafer, Cynthia M.12 (AUTHOR), Shu, Wei2 (AUTHOR), Subramanian, Sharadha13 (AUTHOR), Wagman, Allan S.14 (AUTHOR), Wang, Haixia15 (AUTHOR), Bussiere, Dirksen E.1,2 (AUTHOR) dirksen.bussiere@novartis.com |
| Source: | Bioorganic & Medicinal Chemistry Letters. Feb2020, Vol. 30 Issue 4, pN.PAG-N.PAG. 1p. |
| Database: | Academic Search Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: asn DbLabel: Academic Search Ultimate An: 141380068 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Discovery and optimization of novel pyridines as highly potent and selective glycogen synthase kinase 3 inhibitors. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AR" term="%22Ramurthy%2C+Savithri%22">Ramurthy, Savithri</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Pfister%2C+Keith+B%2E%22">Pfister, Keith B.</searchLink><relatesTo>2</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Boyce%2C+Rustum+S%2E%22">Boyce, Rustum S.</searchLink><relatesTo>3</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Brown%2C+Sean+P%2E%22">Brown, Sean P.</searchLink><relatesTo>4</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Costales%2C+Abran+Q%2E%22">Costales, Abran Q.</searchLink><relatesTo>5</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Desai%2C+Manoj+C%2E%22">Desai, Manoj C.</searchLink><relatesTo>6</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Fang%2C+Eric%22">Fang, Eric</searchLink><relatesTo>7</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Levine%2C+Barry+H%2E%22">Levine, Barry H.</searchLink><relatesTo>8</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Ng%2C+Simon+C%2E%22">Ng, Simon C.</searchLink><relatesTo>9</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Nuss%2C+John+M%2E%22">Nuss, John M.</searchLink><relatesTo>10</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Ring%2C+David+B%2E%22">Ring, David B.</searchLink><relatesTo>11</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Shafer%2C+Cynthia+M%2E%22">Shafer, Cynthia M.</searchLink><relatesTo>12</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Shu%2C+Wei%22">Shu, Wei</searchLink><relatesTo>2</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Subramanian%2C+Sharadha%22">Subramanian, Sharadha</searchLink><relatesTo>13</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Wagman%2C+Allan+S%2E%22">Wagman, Allan S.</searchLink><relatesTo>14</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Wang%2C+Haixia%22">Wang, Haixia</searchLink><relatesTo>15</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Bussiere%2C+Dirksen+E%2E%22">Bussiere, Dirksen E.</searchLink><relatesTo>1,2</relatesTo> (AUTHOR)<i> dirksen.bussiere@novartis.com</i> – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%22Bioorganic+%26+Medicinal+Chemistry+Letters%22">Bioorganic & Medicinal Chemistry Letters</searchLink>. Feb2020, Vol. 30 Issue 4, pN.PAG-N.PAG. 1p. |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=asn&AN=141380068 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1016/j.bmcl.2019.126930 Languages: – Code: eng Text: English PhysicalDescription: Pagination: PageCount: 1 StartPage: N.PAG Titles: – TitleFull: Discovery and optimization of novel pyridines as highly potent and selective glycogen synthase kinase 3 inhibitors. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Ramurthy, Savithri – PersonEntity: Name: NameFull: Pfister, Keith B. – PersonEntity: Name: NameFull: Boyce, Rustum S. – PersonEntity: Name: NameFull: Brown, Sean P. – PersonEntity: Name: NameFull: Costales, Abran Q. – PersonEntity: Name: NameFull: Desai, Manoj C. – PersonEntity: Name: NameFull: Fang, Eric – PersonEntity: Name: NameFull: Levine, Barry H. – PersonEntity: Name: NameFull: Ng, Simon C. – PersonEntity: Name: NameFull: Nuss, John M. – PersonEntity: Name: NameFull: Ring, David B. – PersonEntity: Name: NameFull: Shafer, Cynthia M. – PersonEntity: Name: NameFull: Shu, Wei – PersonEntity: Name: NameFull: Subramanian, Sharadha – PersonEntity: Name: NameFull: Wagman, Allan S. – PersonEntity: Name: NameFull: Wang, Haixia – PersonEntity: Name: NameFull: Bussiere, Dirksen E. IsPartOfRelationships: – BibEntity: Dates: – D: 15 M: 02 Text: Feb2020 Type: published Y: 2020 Identifiers: – Type: issn-print Value: 0960894X Numbering: – Type: volume Value: 30 – Type: issue Value: 4 Titles: – TitleFull: Bioorganic & Medicinal Chemistry Letters Type: main |
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