INCB054828 (pemigatinib), a potent and selective inhibitor of fibroblast growth factor receptors 1, 2, and 3, displays activity against genetically defined tumor models.

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Title: INCB054828 (pemigatinib), a potent and selective inhibitor of fibroblast growth factor receptors 1, 2, and 3, displays activity against genetically defined tumor models.
Authors: Liu, Phillip C. C.1 (AUTHOR), Koblish, Holly1 (AUTHOR) hkoblish@incyte.com, Wu, Liangxing2 (AUTHOR), Bowman, Kevin1 (AUTHOR), Diamond, Sharon1 (AUTHOR), DiMatteo, Darlise1 (AUTHOR), Zhang, Yue1 (AUTHOR), Hansbury, Michael1 (AUTHOR), Rupar, Mark1 (AUTHOR), Wen, Xiaoming1 (AUTHOR), Collier, Paul1 (AUTHOR), Feldman, Patricia1 (AUTHOR), Klabe, Ronald1 (AUTHOR), Burke, Krista A.1 (AUTHOR), Soloviev, Maxim1 (AUTHOR), Gardiner, Christine1 (AUTHOR), He, Xin1 (AUTHOR), Volgina, Alla1 (AUTHOR), Covington, Maryanne1 (AUTHOR), Ruggeri, Bruce1 (AUTHOR)
Source: PLoS ONE. 4/21/2020, Vol. 15 Issue 4, p1-16. 16p.
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