Design of new disubstituted imidazo[1,2-b]pyridazine derivatives as selective Haspin inhibitors. Synthesis, binding mode and anticancer biological evaluation.

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Title: Design of new disubstituted imidazo[1,2-b]pyridazine derivatives as selective Haspin inhibitors. Synthesis, binding mode and anticancer biological evaluation.
Authors: Elie, Jonathan1 (AUTHOR), Feizbakhsh, Omid2 (AUTHOR), Desban, Nathalie2 (AUTHOR), Josselin, Béatrice2,3 (AUTHOR), Baratte, Blandine2,3 (AUTHOR), Bescond, Amandine2 (AUTHOR), Duez, Julien2 (AUTHOR), Fant, Xavier2 (AUTHOR), Bach, Stéphane2,3 (AUTHOR), Marie, Dominique4 (AUTHOR), Place, Matthieu1 (AUTHOR), Ben Salah, Sami1 (AUTHOR), Chartier, Agnes1 (AUTHOR), Berteina-Raboin, Sabine1 (AUTHOR), Chaikuad, Apirat5,6 (AUTHOR), Knapp, Stefan5,6 (AUTHOR), Carles, Fabrice1 (AUTHOR), Bonnet, Pascal1 (AUTHOR), Buron, Frédéric1 (AUTHOR), Routier, Sylvain1 (AUTHOR)
Source: Journal of Enzyme Inhibition & Medicinal Chemistry. Dec2020, Vol. 35 Issue 1, p1840-1853. 14p.
Database: Academic Search Ultimate
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ISSN:14756366
DOI:10.1080/14756366.2020.1825408