Design of new disubstituted imidazo[1,2-b]pyridazine derivatives as selective Haspin inhibitors. Synthesis, binding mode and anticancer biological evaluation.
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| Title: | Design of new disubstituted imidazo[1,2-b]pyridazine derivatives as selective Haspin inhibitors. Synthesis, binding mode and anticancer biological evaluation. |
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| Authors: | Elie, Jonathan1 (AUTHOR), Feizbakhsh, Omid2 (AUTHOR), Desban, Nathalie2 (AUTHOR), Josselin, Béatrice2,3 (AUTHOR), Baratte, Blandine2,3 (AUTHOR), Bescond, Amandine2 (AUTHOR), Duez, Julien2 (AUTHOR), Fant, Xavier2 (AUTHOR), Bach, Stéphane2,3 (AUTHOR), Marie, Dominique4 (AUTHOR), Place, Matthieu1 (AUTHOR), Ben Salah, Sami1 (AUTHOR), Chartier, Agnes1 (AUTHOR), Berteina-Raboin, Sabine1 (AUTHOR), Chaikuad, Apirat5,6 (AUTHOR), Knapp, Stefan5,6 (AUTHOR), Carles, Fabrice1 (AUTHOR), Bonnet, Pascal1 (AUTHOR), Buron, Frédéric1 (AUTHOR), Routier, Sylvain1 (AUTHOR) |
| Source: | Journal of Enzyme Inhibition & Medicinal Chemistry. Dec2020, Vol. 35 Issue 1, p1840-1853. 14p. |
| Database: | Academic Search Ultimate |
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| Header | DbId: asn DbLabel: Academic Search Ultimate An: 147176860 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=asn&AN=147176860 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1080/14756366.2020.1825408 Languages: – Code: eng Text: English PhysicalDescription: Pagination: PageCount: 14 StartPage: 1840 Titles: – TitleFull: Design of new disubstituted imidazo[1,2-b]pyridazine derivatives as selective Haspin inhibitors. Synthesis, binding mode and anticancer biological evaluation. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Elie, Jonathan – PersonEntity: Name: NameFull: Feizbakhsh, Omid – PersonEntity: Name: NameFull: Desban, Nathalie – PersonEntity: Name: NameFull: Josselin, Béatrice – PersonEntity: Name: NameFull: Baratte, Blandine – PersonEntity: Name: NameFull: Bescond, Amandine – PersonEntity: Name: NameFull: Duez, Julien – PersonEntity: Name: NameFull: Fant, Xavier – PersonEntity: Name: NameFull: Bach, Stéphane – PersonEntity: Name: NameFull: Marie, Dominique – PersonEntity: Name: NameFull: Place, Matthieu – PersonEntity: Name: NameFull: Ben Salah, Sami – PersonEntity: Name: NameFull: Chartier, Agnes – PersonEntity: Name: NameFull: Berteina-Raboin, Sabine – PersonEntity: Name: NameFull: Chaikuad, Apirat – PersonEntity: Name: NameFull: Knapp, Stefan – PersonEntity: Name: NameFull: Carles, Fabrice – PersonEntity: Name: NameFull: Bonnet, Pascal – PersonEntity: Name: NameFull: Buron, Frédéric – PersonEntity: Name: NameFull: Routier, Sylvain IsPartOfRelationships: – BibEntity: Dates: – D: 01 M: 12 Text: Dec2020 Type: published Y: 2020 Identifiers: – Type: issn-print Value: 14756366 Numbering: – Type: volume Value: 35 – Type: issue Value: 1 Titles: – TitleFull: Journal of Enzyme Inhibition & Medicinal Chemistry Type: main |
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