Design of new disubstituted imidazo[1,2-b]pyridazine derivatives as selective Haspin inhibitors. Synthesis, binding mode and anticancer biological evaluation.

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Title: Design of new disubstituted imidazo[1,2-b]pyridazine derivatives as selective Haspin inhibitors. Synthesis, binding mode and anticancer biological evaluation.
Authors: Elie, Jonathan1 (AUTHOR), Feizbakhsh, Omid2 (AUTHOR), Desban, Nathalie2 (AUTHOR), Josselin, Béatrice2,3 (AUTHOR), Baratte, Blandine2,3 (AUTHOR), Bescond, Amandine2 (AUTHOR), Duez, Julien2 (AUTHOR), Fant, Xavier2 (AUTHOR), Bach, Stéphane2,3 (AUTHOR), Marie, Dominique4 (AUTHOR), Place, Matthieu1 (AUTHOR), Ben Salah, Sami1 (AUTHOR), Chartier, Agnes1 (AUTHOR), Berteina-Raboin, Sabine1 (AUTHOR), Chaikuad, Apirat5,6 (AUTHOR), Knapp, Stefan5,6 (AUTHOR), Carles, Fabrice1 (AUTHOR), Bonnet, Pascal1 (AUTHOR), Buron, Frédéric1 (AUTHOR), Routier, Sylvain1 (AUTHOR)
Source: Journal of Enzyme Inhibition & Medicinal Chemistry. Dec2020, Vol. 35 Issue 1, p1840-1853. 14p.
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  Data: Design of new disubstituted imidazo[1,2-b]pyridazine derivatives as selective Haspin inhibitors. Synthesis, binding mode and anticancer biological evaluation.
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  Data: <searchLink fieldCode="JN" term="%22Journal+of+Enzyme+Inhibition+%26+Medicinal+Chemistry%22">Journal of Enzyme Inhibition & Medicinal Chemistry</searchLink>. Dec2020, Vol. 35 Issue 1, p1840-1853. 14p.
PLink https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=asn&AN=147176860
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              Text: Dec2020
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