Design, synthesis, and biological evaluation of pyrido[2,3-d]pyrimidine and thieno[2,3-d]pyrimidine derivatives as novel EGFRL858R/T790M inhibitors. - Fu, Jianfang; Yu, Jie; Zhang, Xiang; Chang, Yaoyao; Fan, Hongze; Dong, Mengzhen; Li, Mengjia; Liu, Yue; Hu, Jinxing (Journal of Enzyme Inhibition & Medicinal Chemistry, 2023)