Heteroaryl derivatives of suvorexant as OX1R selective PET ligand candidates: Cu-mediated 18F-fluorination of boroxines, in vitro and initial in vivo evaluation.

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Title: Heteroaryl derivatives of suvorexant as OX1R selective PET ligand candidates: Cu-mediated 18F-fluorination of boroxines, in vitro and initial in vivo evaluation.
Authors: Bolik, Kim-Viktoria1 (AUTHOR), Hellmann, Jan2 (AUTHOR), Maschauer, Simone1 (AUTHOR), Neu, Eduard2,3 (AUTHOR), Einsiedel, Jürgen2 (AUTHOR), Riss, Patrick4 (AUTHOR), Vogg, Nora5 (AUTHOR), König, Jörg3,5 (AUTHOR), Fromm, Martin F.3,5 (AUTHOR), Hübner, Harald2 (AUTHOR), Gmeiner, Peter2,3 (AUTHOR), Prante, Olaf1,3 (AUTHOR) olaf.prante@uk-erlangen.de
Source: EJNMMI Research. 9/4/2024, Vol. 14 Issue 1, p1-16. 16p.
Database: Academic Search Ultimate
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ISSN:2191219X
DOI:10.1186/s13550-024-01141-2