Discovery and evaluation of novel Benzohydroxamic acid-indole derivatives as dual inhibitors of ADAM17 and HDAC2 with antitumor activity.
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| Title: | Discovery and evaluation of novel Benzohydroxamic acid-indole derivatives as dual inhibitors of ADAM17 and HDAC2 with antitumor activity. |
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| Authors: | Song, Xiaoxuan1,2 (AUTHOR), Tong, Xin1 (AUTHOR), Yang, Kaisi1 (AUTHOR), Qi, Yiming1 (AUTHOR), Liu, Wenwu3 (AUTHOR), Sun, Yuzhu4 (AUTHOR), Wang, Chengkang1 (AUTHOR), Xun, Fanghua1 (AUTHOR), Wang, Ziyi1 (AUTHOR), Jiang, Muxuan1 (AUTHOR), Zhang, Yingshi5 (AUTHOR), Ren, Tianshu1 (AUTHOR), Chen, Di6,7 (AUTHOR), Hou, Shanbo8 (AUTHOR), Song, Aigang8 (AUTHOR), Gao, Huiyuan1,2,9,10 (AUTHOR) sypugaohy@163.com, Zhao, Qingchun1,2,5 (AUTHOR) zhaoqingchun1967@163.com |
| Source: | Bioorganic Chemistry. Apr2025, Vol. 157, pN.PAG-N.PAG. 1p. |
| Database: | Academic Search Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: asn DbLabel: Academic Search Ultimate An: 183947971 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Discovery and evaluation of novel Benzohydroxamic acid-indole derivatives as dual inhibitors of ADAM17 and HDAC2 with antitumor activity. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AR" term="%22Song%2C+Xiaoxuan%22">Song, Xiaoxuan</searchLink><relatesTo>1,2</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Tong%2C+Xin%22">Tong, Xin</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Yang%2C+Kaisi%22">Yang, Kaisi</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Qi%2C+Yiming%22">Qi, Yiming</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Liu%2C+Wenwu%22">Liu, Wenwu</searchLink><relatesTo>3</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Sun%2C+Yuzhu%22">Sun, Yuzhu</searchLink><relatesTo>4</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Wang%2C+Chengkang%22">Wang, Chengkang</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Xun%2C+Fanghua%22">Xun, Fanghua</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Wang%2C+Ziyi%22">Wang, Ziyi</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Jiang%2C+Muxuan%22">Jiang, Muxuan</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Zhang%2C+Yingshi%22">Zhang, Yingshi</searchLink><relatesTo>5</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Ren%2C+Tianshu%22">Ren, Tianshu</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Chen%2C+Di%22">Chen, Di</searchLink><relatesTo>6,7</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Hou%2C+Shanbo%22">Hou, Shanbo</searchLink><relatesTo>8</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Song%2C+Aigang%22">Song, Aigang</searchLink><relatesTo>8</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Gao%2C+Huiyuan%22">Gao, Huiyuan</searchLink><relatesTo>1,2,9,10</relatesTo> (AUTHOR)<i> sypugaohy@163.com</i><br /><searchLink fieldCode="AR" term="%22Zhao%2C+Qingchun%22">Zhao, Qingchun</searchLink><relatesTo>1,2,5</relatesTo> (AUTHOR)<i> zhaoqingchun1967@163.com</i> – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%22Bioorganic+Chemistry%22">Bioorganic Chemistry</searchLink>. Apr2025, Vol. 157, pN.PAG-N.PAG. 1p. |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=asn&AN=183947971 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1016/j.bioorg.2025.108308 Languages: – Code: eng Text: English PhysicalDescription: Pagination: PageCount: 1 StartPage: N.PAG Titles: – TitleFull: Discovery and evaluation of novel Benzohydroxamic acid-indole derivatives as dual inhibitors of ADAM17 and HDAC2 with antitumor activity. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Song, Xiaoxuan – PersonEntity: Name: NameFull: Tong, Xin – PersonEntity: Name: NameFull: Yang, Kaisi – PersonEntity: Name: NameFull: Qi, Yiming – PersonEntity: Name: NameFull: Liu, Wenwu – PersonEntity: Name: NameFull: Sun, Yuzhu – PersonEntity: Name: NameFull: Wang, Chengkang – PersonEntity: Name: NameFull: Xun, Fanghua – PersonEntity: Name: NameFull: Wang, Ziyi – PersonEntity: Name: NameFull: Jiang, Muxuan – PersonEntity: Name: NameFull: Zhang, Yingshi – PersonEntity: Name: NameFull: Ren, Tianshu – PersonEntity: Name: NameFull: Chen, Di – PersonEntity: Name: NameFull: Hou, Shanbo – PersonEntity: Name: NameFull: Song, Aigang – PersonEntity: Name: NameFull: Gao, Huiyuan – PersonEntity: Name: NameFull: Zhao, Qingchun IsPartOfRelationships: – BibEntity: Dates: – D: 01 M: 04 Text: Apr2025 Type: published Y: 2025 Identifiers: – Type: issn-print Value: 00452068 Numbering: – Type: volume Value: 157 Titles: – TitleFull: Bioorganic Chemistry Type: main |
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