Assessing Drug–Drug Interaction and Food Effect for BCS Class 2 Compound BI 730357 (Retinoic Acid-Related Orphan Receptor Gamma Antagonist, Bevurogant) Using a Physiology-Based Pharmacokinetics Modeling (PBPK) Approach with Semi-Mechanistic Absorption
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| Title: | Assessing Drug–Drug Interaction and Food Effect for BCS Class 2 Compound BI 730357 (Retinoic Acid-Related Orphan Receptor Gamma Antagonist, Bevurogant) Using a Physiology-Based Pharmacokinetics Modeling (PBPK) Approach with Semi-Mechanistic Absorption |
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| Authors: | Kanacher, Tobias1 (AUTHOR) tobias.kanacher@pharmetheus.com, Sjögren, Erik1,2 (AUTHOR), Korell, Julia2,3 (AUTHOR), Plan, Elodie L.1 (AUTHOR), Gómez-Mantilla, Jose David2,3 (AUTHOR), Ince, Ibrahim3 (AUTHOR) |
| Source: | Pharmaceutics. Mar2025, Vol. 17 Issue 3, p314. 16p. |
| Database: | Academic Search Ultimate |
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| Header | DbId: asn DbLabel: Academic Search Ultimate An: 184102077 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Assessing Drug–Drug Interaction and Food Effect for BCS Class 2 Compound BI 730357 (Retinoic Acid-Related Orphan Receptor Gamma Antagonist, Bevurogant) Using a Physiology-Based Pharmacokinetics Modeling (PBPK) Approach with Semi-Mechanistic Absorption – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AR" term="%22Kanacher%2C+Tobias%22">Kanacher, Tobias</searchLink><relatesTo>1</relatesTo> (AUTHOR)<i> tobias.kanacher@pharmetheus.com</i><br /><searchLink fieldCode="AR" term="%22Sjögren%2C+Erik%22">Sjögren, Erik</searchLink><relatesTo>1,2</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Korell%2C+Julia%22">Korell, Julia</searchLink><relatesTo>2,3</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Plan%2C+Elodie+L%2E%22">Plan, Elodie L.</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Gómez-Mantilla%2C+Jose+David%22">Gómez-Mantilla, Jose David</searchLink><relatesTo>2,3</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Ince%2C+Ibrahim%22">Ince, Ibrahim</searchLink><relatesTo>3</relatesTo> (AUTHOR) – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%22Pharmaceutics%22">Pharmaceutics</searchLink>. Mar2025, Vol. 17 Issue 3, p314. 16p. |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=asn&AN=184102077 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.3390/pharmaceutics17030314 Languages: – Code: eng Text: English PhysicalDescription: Pagination: PageCount: 16 StartPage: 314 Titles: – TitleFull: Assessing Drug–Drug Interaction and Food Effect for BCS Class 2 Compound BI 730357 (Retinoic Acid-Related Orphan Receptor Gamma Antagonist, Bevurogant) Using a Physiology-Based Pharmacokinetics Modeling (PBPK) Approach with Semi-Mechanistic Absorption Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Kanacher, Tobias – PersonEntity: Name: NameFull: Sjögren, Erik – PersonEntity: Name: NameFull: Korell, Julia – PersonEntity: Name: NameFull: Plan, Elodie L. – PersonEntity: Name: NameFull: Gómez-Mantilla, Jose David – PersonEntity: Name: NameFull: Ince, Ibrahim IsPartOfRelationships: – BibEntity: Dates: – D: 01 M: 03 Text: Mar2025 Type: published Y: 2025 Identifiers: – Type: issn-print Value: 19994923 Numbering: – Type: volume Value: 17 – Type: issue Value: 3 Titles: – TitleFull: Pharmaceutics Type: main |
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