Design, synthesis, and biological evaluation of 1,2,4-triazolo[1,5-a][1,3,5]triazine derivatives as E. coli DNA gyrase inhibitors.

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Title: Design, synthesis, and biological evaluation of 1,2,4-triazolo[1,5-a][1,3,5]triazine derivatives as E. coli DNA gyrase inhibitors.
Authors: Mokoena, Sithabile1 (AUTHOR), Ganai, Majeed1 (AUTHOR), Pathan, Tabasum1 (AUTHOR), Ike, Blessing1 (AUTHOR), Obakachi, Vincent1 (AUTHOR), Adu, Darko Kwabena1 (AUTHOR), Alake, John1 (AUTHOR), Kajee, Afsana1,2 (AUTHOR), Shaik, Baji Baba1 (AUTHOR), Partap, Sangh1 (AUTHOR), Mohite, Sachin1 (AUTHOR), Nadigar, Siddaram1 (AUTHOR), Karpoormath, Rajshekhar1 (AUTHOR) karpoormath@ukzn.ac.za
Source: Journal of Molecular Structure. Aug2025, Vol. 1336, pN.PAG-N.PAG. 1p.
Database: Academic Search Ultimate
Description
ISSN:00222860
DOI:10.1016/j.molstruc.2025.141994