Design, synthesis, and biological evaluation of 1,2,4-triazolo[1,5-a][1,3,5]triazine derivatives as E. coli DNA gyrase inhibitors.

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Title: Design, synthesis, and biological evaluation of 1,2,4-triazolo[1,5-a][1,3,5]triazine derivatives as E. coli DNA gyrase inhibitors.
Authors: Mokoena, Sithabile1 (AUTHOR), Ganai, Majeed1 (AUTHOR), Pathan, Tabasum1 (AUTHOR), Ike, Blessing1 (AUTHOR), Obakachi, Vincent1 (AUTHOR), Adu, Darko Kwabena1 (AUTHOR), Alake, John1 (AUTHOR), Kajee, Afsana1,2 (AUTHOR), Shaik, Baji Baba1 (AUTHOR), Partap, Sangh1 (AUTHOR), Mohite, Sachin1 (AUTHOR), Nadigar, Siddaram1 (AUTHOR), Karpoormath, Rajshekhar1 (AUTHOR) karpoormath@ukzn.ac.za
Source: Journal of Molecular Structure. Aug2025, Vol. 1336, pN.PAG-N.PAG. 1p.
Database: Academic Search Ultimate
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  Data: Design, synthesis, and biological evaluation of 1,2,4-triazolo[1,5-a][1,3,5]triazine derivatives as E. coli DNA gyrase inhibitors.
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PLink https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=asn&AN=184648536
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      – Type: doi
        Value: 10.1016/j.molstruc.2025.141994
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      – Code: eng
        Text: English
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        PageCount: 1
        StartPage: N.PAG
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      – TitleFull: Design, synthesis, and biological evaluation of 1,2,4-triazolo[1,5-a][1,3,5]triazine derivatives as E. coli DNA gyrase inhibitors.
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              Text: Aug2025
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              Y: 2025
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