Altered desensitization and internalization patterns of rodent versus human glucose‐dependent insulinotropic polypeptide (GIP) receptors. An important drug discovery challenge.

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Title: Altered desensitization and internalization patterns of rodent versus human glucose‐dependent insulinotropic polypeptide (GIP) receptors. An important drug discovery challenge.
Authors: Gasbjerg, Lærke Smidt1 (AUTHOR), Rasmussen, Rasmus Syberg1 (AUTHOR), Dragan, Adrian1 (AUTHOR), Lindquist, Peter1 (AUTHOR), Melchiorsen, Josefine Ulrikke1 (AUTHOR), Stepniewski, Tomasz Maciej2,3,4 (AUTHOR), Schiellerup, Sine1 (AUTHOR), Tordrup, Esther Karen1 (AUTHOR), Gadgaard, Sarina1,5 (AUTHOR), Kizilkaya, Hüsün Sheyma1 (AUTHOR), Willems, Sabine6 (AUTHOR), Zhong, Yi6,7 (AUTHOR), Wang, Yi7,8,9 (AUTHOR), Wright, Shane C.6 (AUTHOR), Lauschke, Volker M.6,10,11 (AUTHOR), Hartmann, Bolette1 (AUTHOR), Holst, Jens Juul1,12 (AUTHOR), Selent, Jana2 (AUTHOR), Rosenkilde, Mette Marie1 (AUTHOR) rosenkilde@sund.ku.dk
Source: British Journal of Pharmacology. Jul2025, Vol. 182 Issue 14, p3353-3370. 18p.
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  Data: Altered desensitization and internalization patterns of rodent versus human glucose‐dependent insulinotropic polypeptide (GIP) receptors. An important drug discovery challenge.
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  Data: <searchLink fieldCode="JN" term="%22British+Journal+of+Pharmacology%22">British Journal of Pharmacology</searchLink>. Jul2025, Vol. 182 Issue 14, p3353-3370. 18p.
PLink https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=asn&AN=185963900
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