Discovery of 1‐(Cyclopropylmethyl)‐2‐(Dibenzo[b,d]Thiophen‐2‐yl)‐1H‐Benzo[d]Imidazole‐5‐Carboxylic Acid as Orally Bioavailable EP4 Receptor Antagonist.

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Title: Discovery of 1‐(Cyclopropylmethyl)‐2‐(Dibenzo[b,d]Thiophen‐2‐yl)‐1H‐Benzo[d]Imidazole‐5‐Carboxylic Acid as Orally Bioavailable EP4 Receptor Antagonist.
Authors: Kumar, Sanjay1,2 (AUTHOR), Chakraborty, Rajib1 (AUTHOR), Roy, Chandreyee1 (AUTHOR), Basu, Sohini1 (AUTHOR), Hajra, Arun K.1 (AUTHOR), Sen, Priyam1 (AUTHOR), Paul, Debajyoti1 (AUTHOR), Phukan, Karabi1 (AUTHOR), Roy, Subhasis1 (AUTHOR), Bera, Rammohan1 (AUTHOR), Mondal, Trisha1 (AUTHOR), Chakraborty, Sabyasachi1 (AUTHOR), Banerjee, Manish1 (AUTHOR), Mondal, Susanta K.1 (AUTHOR), Das, Sonali1 (AUTHOR), Malik, Pradip1 (AUTHOR), De Mandal, Surajit2 (AUTHOR), Subudhi, Enketeswara2 (AUTHOR) enketeswarasubudhi@soa.ac.in, Kundu, Mrinalkanti1 (AUTHOR) mrinal.kundu@tcgls.com
Source: Chemical Biology & Drug Design. Jun2025, Vol. 105 Issue 6, p1-8. 8p.
Database: Academic Search Ultimate
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Description
ISSN:17470277
DOI:10.1111/cbdd.70132