Design, synthesis, and antitumor activity study of β-carboline derivatives as selective HDAC1/2 inhibitors.

Saved in:
Bibliographic Details
Title: Design, synthesis, and antitumor activity study of β-carboline derivatives as selective HDAC1/2 inhibitors.
Authors: Wang, Zhiya1,2 (AUTHOR), Wu, Limeng1 (AUTHOR), Yang, Kaisi1 (AUTHOR), Qi, Yiming1 (AUTHOR), Li, Zhenshu1 (AUTHOR), Liu, Wenjie3 (AUTHOR), Xu, Xiangbo1 (AUTHOR), Zheng, Fangyuan1 (AUTHOR), Zeng, Wenbo1 (AUTHOR), Gong, Hao1 (AUTHOR), Tian, Caizhi2 (AUTHOR), Geng, Hefeng4 (AUTHOR), Xu, Zihua1 (AUTHOR), Zhou, Kangyao5 (AUTHOR), Tian, Haihong1,6 (AUTHOR), Ren, Tianshu1 (AUTHOR), Zhao, Qingchun1 (AUTHOR)
Source: Bioorganic Chemistry. Aug2025, Vol. 163, pN.PAG-N.PAG. 1p.
Database: Academic Search Ultimate
FullText Text:
  Availability: 0
Header DbId: asn
DbLabel: Academic Search Ultimate
An: 187140247
AccessLevel: 2
PubType: Academic Journal
PubTypeId: academicJournal
PreciseRelevancyScore: 0
IllustrationInfo
Items – Name: Title
  Label: Title
  Group: Ti
  Data: Design, synthesis, and antitumor activity study of β-carboline derivatives as selective HDAC1/2 inhibitors.
– Name: Author
  Label: Authors
  Group: Au
  Data: <searchLink fieldCode="AR" term="%22Wang%2C+Zhiya%22">Wang, Zhiya</searchLink><relatesTo>1,2</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Wu%2C+Limeng%22">Wu, Limeng</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Yang%2C+Kaisi%22">Yang, Kaisi</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Qi%2C+Yiming%22">Qi, Yiming</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Li%2C+Zhenshu%22">Li, Zhenshu</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Liu%2C+Wenjie%22">Liu, Wenjie</searchLink><relatesTo>3</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Xu%2C+Xiangbo%22">Xu, Xiangbo</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Zheng%2C+Fangyuan%22">Zheng, Fangyuan</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Zeng%2C+Wenbo%22">Zeng, Wenbo</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Gong%2C+Hao%22">Gong, Hao</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Tian%2C+Caizhi%22">Tian, Caizhi</searchLink><relatesTo>2</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Geng%2C+Hefeng%22">Geng, Hefeng</searchLink><relatesTo>4</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Xu%2C+Zihua%22">Xu, Zihua</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Zhou%2C+Kangyao%22">Zhou, Kangyao</searchLink><relatesTo>5</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Tian%2C+Haihong%22">Tian, Haihong</searchLink><relatesTo>1,6</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Ren%2C+Tianshu%22">Ren, Tianshu</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Zhao%2C+Qingchun%22">Zhao, Qingchun</searchLink><relatesTo>1</relatesTo> (AUTHOR)
– Name: TitleSource
  Label: Source
  Group: Src
  Data: <searchLink fieldCode="JN" term="%22Bioorganic+Chemistry%22">Bioorganic Chemistry</searchLink>. Aug2025, Vol. 163, pN.PAG-N.PAG. 1p.
PLink https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=asn&AN=187140247
RecordInfo BibRecord:
  BibEntity:
    Identifiers:
      – Type: doi
        Value: 10.1016/j.bioorg.2025.108763
    Languages:
      – Code: eng
        Text: English
    PhysicalDescription:
      Pagination:
        PageCount: 1
        StartPage: N.PAG
    Titles:
      – TitleFull: Design, synthesis, and antitumor activity study of β-carboline derivatives as selective HDAC1/2 inhibitors.
        Type: main
  BibRelationships:
    HasContributorRelationships:
      – PersonEntity:
          Name:
            NameFull: Wang, Zhiya
      – PersonEntity:
          Name:
            NameFull: Wu, Limeng
      – PersonEntity:
          Name:
            NameFull: Yang, Kaisi
      – PersonEntity:
          Name:
            NameFull: Qi, Yiming
      – PersonEntity:
          Name:
            NameFull: Li, Zhenshu
      – PersonEntity:
          Name:
            NameFull: Liu, Wenjie
      – PersonEntity:
          Name:
            NameFull: Xu, Xiangbo
      – PersonEntity:
          Name:
            NameFull: Zheng, Fangyuan
      – PersonEntity:
          Name:
            NameFull: Zeng, Wenbo
      – PersonEntity:
          Name:
            NameFull: Gong, Hao
      – PersonEntity:
          Name:
            NameFull: Tian, Caizhi
      – PersonEntity:
          Name:
            NameFull: Geng, Hefeng
      – PersonEntity:
          Name:
            NameFull: Xu, Zihua
      – PersonEntity:
          Name:
            NameFull: Zhou, Kangyao
      – PersonEntity:
          Name:
            NameFull: Tian, Haihong
      – PersonEntity:
          Name:
            NameFull: Ren, Tianshu
      – PersonEntity:
          Name:
            NameFull: Zhao, Qingchun
    IsPartOfRelationships:
      – BibEntity:
          Dates:
            – D: 01
              M: 08
              Text: Aug2025
              Type: published
              Y: 2025
          Identifiers:
            – Type: issn-print
              Value: 00452068
          Numbering:
            – Type: volume
              Value: 163
          Titles:
            – TitleFull: Bioorganic Chemistry
              Type: main
ResultId 1