Discovery of conformation constrained tetracyclic compounds as potent chitinase OfChi-h inhibitors with a novel binding mode.

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Title: Discovery of conformation constrained tetracyclic compounds as potent chitinase OfChi-h inhibitors with a novel binding mode.
Authors: Yuan, Pengtao1,2 (AUTHOR), Jiang, Xi3 (AUTHOR), Ni, Xintong4 (AUTHOR), Shao, Xusheng4 (AUTHOR), Qian, Xuhong4,5 (AUTHOR) xhqian@ecust.edu.cn, Yang, Qing1,2 (AUTHOR) qingyang@caas.cn
Source: Journal of Enzyme Inhibition & Medicinal Chemistry. Dec2025, Vol. 40 Issue 1, p1-11. 11p.
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  Data: Discovery of conformation constrained tetracyclic compounds as potent chitinase OfChi-h inhibitors with a novel binding mode.
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  Data: <searchLink fieldCode="AR" term="%22Yuan%2C+Pengtao%22">Yuan, Pengtao</searchLink><relatesTo>1,2</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Jiang%2C+Xi%22">Jiang, Xi</searchLink><relatesTo>3</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Ni%2C+Xintong%22">Ni, Xintong</searchLink><relatesTo>4</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Shao%2C+Xusheng%22">Shao, Xusheng</searchLink><relatesTo>4</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Qian%2C+Xuhong%22">Qian, Xuhong</searchLink><relatesTo>4,5</relatesTo> (AUTHOR)<i> xhqian@ecust.edu.cn</i><br /><searchLink fieldCode="AR" term="%22Yang%2C+Qing%22">Yang, Qing</searchLink><relatesTo>1,2</relatesTo> (AUTHOR)<i> qingyang@caas.cn</i>
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  Data: <searchLink fieldCode="JN" term="%22Journal+of+Enzyme+Inhibition+%26+Medicinal+Chemistry%22">Journal of Enzyme Inhibition & Medicinal Chemistry</searchLink>. Dec2025, Vol. 40 Issue 1, p1-11. 11p.
PLink https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=asn&AN=190283268
RecordInfo BibRecord:
  BibEntity:
    Identifiers:
      – Type: doi
        Value: 10.1080/14756366.2025.2528056
    Languages:
      – Code: eng
        Text: English
    PhysicalDescription:
      Pagination:
        PageCount: 11
        StartPage: 1
    Titles:
      – TitleFull: Discovery of conformation constrained tetracyclic compounds as potent chitinase OfChi-h inhibitors with a novel binding mode.
        Type: main
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          Name:
            NameFull: Yuan, Pengtao
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          Name:
            NameFull: Jiang, Xi
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          Name:
            NameFull: Ni, Xintong
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            NameFull: Shao, Xusheng
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            NameFull: Qian, Xuhong
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            NameFull: Yang, Qing
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          Dates:
            – D: 01
              M: 12
              Text: Dec2025
              Type: published
              Y: 2025
          Identifiers:
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              Value: 14756366
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              Value: 40
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            – TitleFull: Journal of Enzyme Inhibition & Medicinal Chemistry
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