Design, synthesis and biological evaluation of symmetric thiadiazole carboxamide derivative as glutaminase inhibitor.

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Title: Design, synthesis and biological evaluation of symmetric thiadiazole carboxamide derivative as glutaminase inhibitor.
Authors: Cyriac, Rajath1,2 (AUTHOR), Lee, Eun Ji1,3 (AUTHOR), Kwon, Yeongju1,4 (AUTHOR), Yun, Mi Ran1,5,6 (AUTHOR), Jung, Myoung Eun1 (AUTHOR), Ahn, Sunjoo1,2 (AUTHOR), Chae, Chang Hak1 (AUTHOR) chchae@krict.re.kr, Choi, Gildon1,2 (AUTHOR) gchoi@krict.re.kr, Cho, Byoung Chul1,7 (AUTHOR) CBC1971@yuhs.ac, Lee, Kwangho1,2 (AUTHOR) kwangho@krict.re.kr
Source: Bioorganic & Medicinal Chemistry Letters. Jul2026, Vol. 136, pN.PAG-N.PAG. 1p.
Database: Academic Search Ultimate
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  Data: Design, synthesis and biological evaluation of symmetric thiadiazole carboxamide derivative as glutaminase inhibitor.
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  Data: <searchLink fieldCode="AR" term="%22Cyriac%2C+Rajath%22">Cyriac, Rajath</searchLink><relatesTo>1,2</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Lee%2C+Eun+Ji%22">Lee, Eun Ji</searchLink><relatesTo>1,3</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Kwon%2C+Yeongju%22">Kwon, Yeongju</searchLink><relatesTo>1,4</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Yun%2C+Mi+Ran%22">Yun, Mi Ran</searchLink><relatesTo>1,5,6</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Jung%2C+Myoung+Eun%22">Jung, Myoung Eun</searchLink><relatesTo>1</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Ahn%2C+Sunjoo%22">Ahn, Sunjoo</searchLink><relatesTo>1,2</relatesTo> (AUTHOR)<br /><searchLink fieldCode="AR" term="%22Chae%2C+Chang+Hak%22">Chae, Chang Hak</searchLink><relatesTo>1</relatesTo> (AUTHOR)<i> chchae@krict.re.kr</i><br /><searchLink fieldCode="AR" term="%22Choi%2C+Gildon%22">Choi, Gildon</searchLink><relatesTo>1,2</relatesTo> (AUTHOR)<i> gchoi@krict.re.kr</i><br /><searchLink fieldCode="AR" term="%22Cho%2C+Byoung+Chul%22">Cho, Byoung Chul</searchLink><relatesTo>1,7</relatesTo> (AUTHOR)<i> CBC1971@yuhs.ac</i><br /><searchLink fieldCode="AR" term="%22Lee%2C+Kwangho%22">Lee, Kwangho</searchLink><relatesTo>1,2</relatesTo> (AUTHOR)<i> kwangho@krict.re.kr</i>
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  Data: <searchLink fieldCode="JN" term="%22Bioorganic+%26+Medicinal+Chemistry+Letters%22">Bioorganic & Medicinal Chemistry Letters</searchLink>. Jul2026, Vol. 136, pN.PAG-N.PAG. 1p.
PLink https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=asn&AN=192666204
RecordInfo BibRecord:
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      – Type: doi
        Value: 10.1016/j.bmcl.2026.130595
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      – Code: eng
        Text: English
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      – TitleFull: Design, synthesis and biological evaluation of symmetric thiadiazole carboxamide derivative as glutaminase inhibitor.
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            NameFull: Cyriac, Rajath
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            NameFull: Lee, Eun Ji
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            NameFull: Kwon, Yeongju
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            – D: 01
              M: 07
              Text: Jul2026
              Type: published
              Y: 2026
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              Value: 0960894X
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              Value: 136
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