Synthesis and biological activity of heteroaryl 3-(1,1-dioxo-2H-(1,2,4)-benzothiadizin-3-yl)-4-hydroxy-2(1H)-quinolinone derivatives as hepatitis C virus NS5B polymerase inhibitors

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Title: Synthesis and biological activity of heteroaryl 3-(1,1-dioxo-2H-(1,2,4)-benzothiadizin-3-yl)-4-hydroxy-2(1H)-quinolinone derivatives as hepatitis C virus NS5B polymerase inhibitors
Authors: Tedesco, Rosanna1 Rosanna_2_Tedesco@gsk.com, Chai, Deping1, Darcy, Michael G.1, Dhanak, Dashyant1, Fitch, Duke M.1, Gates, Adam2, Johnston, Victor K.2, Keenan, Richard M.1, Lin-Goerke, Juili2, Sarisky, Robert T.2, Shaw, Antony N.1, Valko, Klara L.3, Wiggall, Kenneth J.1, Zimmerman, Michael N.1, Duffy, Kevin J.1
Source: Bioorganic & Medicinal Chemistry Letters. Aug2009, Vol. 19 Issue 15, p4354-4358. 5p.
Database: Academic Search Ultimate
Description
ISSN:0960894X
DOI:10.1016/j.bmcl.2009.05.080