The discovery and optimisation of pyrido[2,3-d]pyrimidine-2,4-diamines as potent and selective inhibitors of mTOR kinase
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| Title: | The discovery and optimisation of pyrido[2,3-d]pyrimidine-2,4-diamines as potent and selective inhibitors of mTOR kinase |
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| Authors: | Malagu, Karine1, Duggan, Heather1, Menear, Keith1, Hummersone, Marc1, Gomez, Sylvie1, Bailey, Christine1, Edwards, Peter1, Drzewiecki, Jan1, Leroux, Frédéric1, Quesada, Mar Jimenez1, Hermann, Gesine1, Maine, Stephanie1, Molyneaux, Carrie-Anne1, Le Gall, Armelle1, Pullen, James1, Hickson, Ian1, Smith, Lisa1, Maguire, Sharon1, Martin, Niall1, Smith, Graeme1,2 |
| Source: | Bioorganic & Medicinal Chemistry Letters. Oct2009, Vol. 19 Issue 20, p5950-5953. 4p. |
| Database: | Academic Search Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: asn DbLabel: Academic Search Ultimate An: 44416493 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=asn&AN=44416493 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1016/j.bmcl.2009.08.038 Languages: – Code: eng Text: English PhysicalDescription: Pagination: PageCount: 4 StartPage: 5950 Titles: – TitleFull: The discovery and optimisation of pyrido[2,3-d]pyrimidine-2,4-diamines as potent and selective inhibitors of mTOR kinase Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Malagu, Karine – PersonEntity: Name: NameFull: Duggan, Heather – PersonEntity: Name: NameFull: Menear, Keith – PersonEntity: Name: NameFull: Hummersone, Marc – PersonEntity: Name: NameFull: Gomez, Sylvie – PersonEntity: Name: NameFull: Bailey, Christine – PersonEntity: Name: NameFull: Edwards, Peter – PersonEntity: Name: NameFull: Drzewiecki, Jan – PersonEntity: Name: NameFull: Leroux, Frédéric – PersonEntity: Name: NameFull: Quesada, Mar Jimenez – PersonEntity: Name: NameFull: Hermann, Gesine – PersonEntity: Name: NameFull: Maine, Stephanie – PersonEntity: Name: NameFull: Molyneaux, Carrie-Anne – PersonEntity: Name: NameFull: Le Gall, Armelle – PersonEntity: Name: NameFull: Pullen, James – PersonEntity: Name: NameFull: Hickson, Ian – PersonEntity: Name: NameFull: Smith, Lisa – PersonEntity: Name: NameFull: Maguire, Sharon – PersonEntity: Name: NameFull: Martin, Niall – PersonEntity: Name: NameFull: Smith, Graeme IsPartOfRelationships: – BibEntity: Dates: – D: 15 M: 10 Text: Oct2009 Type: published Y: 2009 Identifiers: – Type: issn-print Value: 0960894X Numbering: – Type: volume Value: 19 – Type: issue Value: 20 Titles: – TitleFull: Bioorganic & Medicinal Chemistry Letters Type: main |
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