Discovery of covalent inhibitors for MIF tautomerase via cocrystal structures with phantom hits from virtual screening

Saved in:
Bibliographic Details
Title: Discovery of covalent inhibitors for MIF tautomerase via cocrystal structures with phantom hits from virtual screening
Authors: McLean, Larry R.1 Larry.Mclean@sanofi-aventis.com, Zhang, Ying1, Li, Hua1, Li, Ziyu2, Lukasczyk, Ulrike2, Choi, Yong-Mi1, Han, Zuoning1, Prisco, Joy1, Fordham, Jeremy1, Tsay, Joseph T.1, Reiling, Stephan1, Vaz, Roy J.1, Li, Yi1 yi.li@sanofi-aventis.com
Source: Bioorganic & Medicinal Chemistry Letters. Dec2009, Vol. 19 Issue 23, p6717-6720. 4p.
Database: Academic Search Ultimate
Description
ISSN:0960894X
DOI:10.1016/j.bmcl.2009.09.106