Discovery of covalent inhibitors for MIF tautomerase via cocrystal structures with phantom hits from virtual screening
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| Title: | Discovery of covalent inhibitors for MIF tautomerase via cocrystal structures with phantom hits from virtual screening |
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| Authors: | McLean, Larry R.1 Larry.Mclean@sanofi-aventis.com, Zhang, Ying1, Li, Hua1, Li, Ziyu2, Lukasczyk, Ulrike2, Choi, Yong-Mi1, Han, Zuoning1, Prisco, Joy1, Fordham, Jeremy1, Tsay, Joseph T.1, Reiling, Stephan1, Vaz, Roy J.1, Li, Yi1 yi.li@sanofi-aventis.com |
| Source: | Bioorganic & Medicinal Chemistry Letters. Dec2009, Vol. 19 Issue 23, p6717-6720. 4p. |
| Database: | Academic Search Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: asn DbLabel: Academic Search Ultimate An: 45068341 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=asn&AN=45068341 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1016/j.bmcl.2009.09.106 Languages: – Code: eng Text: English PhysicalDescription: Pagination: PageCount: 4 StartPage: 6717 Titles: – TitleFull: Discovery of covalent inhibitors for MIF tautomerase via cocrystal structures with phantom hits from virtual screening Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: McLean, Larry R. – PersonEntity: Name: NameFull: Zhang, Ying – PersonEntity: Name: NameFull: Li, Hua – PersonEntity: Name: NameFull: Li, Ziyu – PersonEntity: Name: NameFull: Lukasczyk, Ulrike – PersonEntity: Name: NameFull: Choi, Yong-Mi – PersonEntity: Name: NameFull: Han, Zuoning – PersonEntity: Name: NameFull: Prisco, Joy – PersonEntity: Name: NameFull: Fordham, Jeremy – PersonEntity: Name: NameFull: Tsay, Joseph T. – PersonEntity: Name: NameFull: Reiling, Stephan – PersonEntity: Name: NameFull: Vaz, Roy J. – PersonEntity: Name: NameFull: Li, Yi IsPartOfRelationships: – BibEntity: Dates: – D: 01 M: 12 Text: Dec2009 Type: published Y: 2009 Identifiers: – Type: issn-print Value: 0960894X Numbering: – Type: volume Value: 19 – Type: issue Value: 23 Titles: – TitleFull: Bioorganic & Medicinal Chemistry Letters Type: main |
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