Discovery of covalent inhibitors for MIF tautomerase via cocrystal structures with phantom hits from virtual screening

Saved in:
Bibliographic Details
Title: Discovery of covalent inhibitors for MIF tautomerase via cocrystal structures with phantom hits from virtual screening
Authors: McLean, Larry R.1 Larry.Mclean@sanofi-aventis.com, Zhang, Ying1, Li, Hua1, Li, Ziyu2, Lukasczyk, Ulrike2, Choi, Yong-Mi1, Han, Zuoning1, Prisco, Joy1, Fordham, Jeremy1, Tsay, Joseph T.1, Reiling, Stephan1, Vaz, Roy J.1, Li, Yi1 yi.li@sanofi-aventis.com
Source: Bioorganic & Medicinal Chemistry Letters. Dec2009, Vol. 19 Issue 23, p6717-6720. 4p.
Database: Academic Search Ultimate
FullText Text:
  Availability: 0
Header DbId: asn
DbLabel: Academic Search Ultimate
An: 45068341
AccessLevel: 2
PubType: Academic Journal
PubTypeId: academicJournal
PreciseRelevancyScore: 0
IllustrationInfo
Items – Name: Title
  Label: Title
  Group: Ti
  Data: Discovery of covalent inhibitors for MIF tautomerase via cocrystal structures with phantom hits from virtual screening
– Name: Author
  Label: Authors
  Group: Au
  Data: <searchLink fieldCode="AR" term="%22McLean%2C+Larry+R%2E%22">McLean, Larry R.</searchLink><relatesTo>1</relatesTo><i> Larry.Mclean@sanofi-aventis.com</i><br /><searchLink fieldCode="AR" term="%22Zhang%2C+Ying%22">Zhang, Ying</searchLink><relatesTo>1</relatesTo><br /><searchLink fieldCode="AR" term="%22Li%2C+Hua%22">Li, Hua</searchLink><relatesTo>1</relatesTo><br /><searchLink fieldCode="AR" term="%22Li%2C+Ziyu%22">Li, Ziyu</searchLink><relatesTo>2</relatesTo><br /><searchLink fieldCode="AR" term="%22Lukasczyk%2C+Ulrike%22">Lukasczyk, Ulrike</searchLink><relatesTo>2</relatesTo><br /><searchLink fieldCode="AR" term="%22Choi%2C+Yong-Mi%22">Choi, Yong-Mi</searchLink><relatesTo>1</relatesTo><br /><searchLink fieldCode="AR" term="%22Han%2C+Zuoning%22">Han, Zuoning</searchLink><relatesTo>1</relatesTo><br /><searchLink fieldCode="AR" term="%22Prisco%2C+Joy%22">Prisco, Joy</searchLink><relatesTo>1</relatesTo><br /><searchLink fieldCode="AR" term="%22Fordham%2C+Jeremy%22">Fordham, Jeremy</searchLink><relatesTo>1</relatesTo><br /><searchLink fieldCode="AR" term="%22Tsay%2C+Joseph+T%2E%22">Tsay, Joseph T.</searchLink><relatesTo>1</relatesTo><br /><searchLink fieldCode="AR" term="%22Reiling%2C+Stephan%22">Reiling, Stephan</searchLink><relatesTo>1</relatesTo><br /><searchLink fieldCode="AR" term="%22Vaz%2C+Roy+J%2E%22">Vaz, Roy J.</searchLink><relatesTo>1</relatesTo><br /><searchLink fieldCode="AR" term="%22Li%2C+Yi%22">Li, Yi</searchLink><relatesTo>1</relatesTo><i> yi.li@sanofi-aventis.com</i>
– Name: TitleSource
  Label: Source
  Group: Src
  Data: <searchLink fieldCode="JN" term="%22Bioorganic+%26+Medicinal+Chemistry+Letters%22">Bioorganic & Medicinal Chemistry Letters</searchLink>. Dec2009, Vol. 19 Issue 23, p6717-6720. 4p.
PLink https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=asn&AN=45068341
RecordInfo BibRecord:
  BibEntity:
    Identifiers:
      – Type: doi
        Value: 10.1016/j.bmcl.2009.09.106
    Languages:
      – Code: eng
        Text: English
    PhysicalDescription:
      Pagination:
        PageCount: 4
        StartPage: 6717
    Titles:
      – TitleFull: Discovery of covalent inhibitors for MIF tautomerase via cocrystal structures with phantom hits from virtual screening
        Type: main
  BibRelationships:
    HasContributorRelationships:
      – PersonEntity:
          Name:
            NameFull: McLean, Larry R.
      – PersonEntity:
          Name:
            NameFull: Zhang, Ying
      – PersonEntity:
          Name:
            NameFull: Li, Hua
      – PersonEntity:
          Name:
            NameFull: Li, Ziyu
      – PersonEntity:
          Name:
            NameFull: Lukasczyk, Ulrike
      – PersonEntity:
          Name:
            NameFull: Choi, Yong-Mi
      – PersonEntity:
          Name:
            NameFull: Han, Zuoning
      – PersonEntity:
          Name:
            NameFull: Prisco, Joy
      – PersonEntity:
          Name:
            NameFull: Fordham, Jeremy
      – PersonEntity:
          Name:
            NameFull: Tsay, Joseph T.
      – PersonEntity:
          Name:
            NameFull: Reiling, Stephan
      – PersonEntity:
          Name:
            NameFull: Vaz, Roy J.
      – PersonEntity:
          Name:
            NameFull: Li, Yi
    IsPartOfRelationships:
      – BibEntity:
          Dates:
            – D: 01
              M: 12
              Text: Dec2009
              Type: published
              Y: 2009
          Identifiers:
            – Type: issn-print
              Value: 0960894X
          Numbering:
            – Type: volume
              Value: 19
            – Type: issue
              Value: 23
          Titles:
            – TitleFull: Bioorganic & Medicinal Chemistry Letters
              Type: main
ResultId 1