Utilization of in vitro Caco-2 permeability and liver microsomal half-life screens in discovering BMS-488043, a novel HIV-1 attachment inhibitor with improved pharmacokinetic properties. - Zheng Yang; Zadjura, Lisa M.; Marino, Anthony M.; D'Arienzo, Celia J.; Malinowski, Jacek; Gesenberg, Christoph; Pin-Fang Lin; Colonno, Richard J.; Tao Wang; Kadow, John F.; Meanwell, Nicholas A.; Hansel, Steven B. (Journal of Pharmaceutical Sciences, 2010)