New Potent Bisubstrate Inhibitors of Histone Acetyltransferase p300: Design, Synthesis and Biological Evaluation.

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Bibliographic Details
Title: New Potent Bisubstrate Inhibitors of Histone Acetyltransferase p300: Design, Synthesis and Biological Evaluation.
Authors: Kwie, Franciane Ho A.1,2, Briet, Martine2,3, Soupaya, David1,2, Hoffmann, Pascal1,2, Maturano, Marie1,2, Rodriguez, Frédéric1,2, Blonski, Casimir1,2, Lherbet, Christian1,2, Baudoin-Dehoux, Cécile1,2 baudoin@chimie.ups-tlse.fr
Source: Chemical Biology & Drug Design. Jan2011, Vol. 77 Issue 1, p86-92. 7p. 1 Color Photograph, 3 Diagrams, 1 Chart.
Database: Academic Search Ultimate
Description
ISSN:17470277
DOI:10.1111/j.1747-0285.2010.01056.x