Development of an Activity-Based Probe and In Silico Design Reveal Highly Selective Inhibitors for Diacylglycerol Lipase-α in Brain.

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Title: Development of an Activity-Based Probe and In Silico Design Reveal Highly Selective Inhibitors for Diacylglycerol Lipase-α in Brain.
Authors: Baggelaar, Marc P.1, Janssen, Freek J.1, van Esbroeck, Annelot C. M.1, den Dulk, Hans2, Allarà, Marco3, Hoogendoorn, Sascha1, McGuire, Ross4, Florea, Bogdan I.1, Meeuwenoord, Nico1, van den Elst, Hans1, van der Marel, Gijsbert A.1, Brouwer, Jaap2, Di Marzo, Vincenzo3, Overkleeft, Herman S.1, van der Stelt, Mario1 m.van.der.stelt@chem.leidenuniv.nl
Source: Angewandte Chemie. Nov2013, Vol. 125 Issue 46, p12303-12307. 5p.
Database: Academic Search Ultimate
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ISSN:00448249
DOI:10.1002/ange.201306295