Development of an Activity-Based Probe and In Silico Design Reveal Highly Selective Inhibitors for Diacylglycerol Lipase-α in Brain.
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| Title: | Development of an Activity-Based Probe and In Silico Design Reveal Highly Selective Inhibitors for Diacylglycerol Lipase-α in Brain. |
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| Authors: | Baggelaar, Marc P.1, Janssen, Freek J.1, van Esbroeck, Annelot C. M.1, den Dulk, Hans2, Allarà, Marco3, Hoogendoorn, Sascha1, McGuire, Ross4, Florea, Bogdan I.1, Meeuwenoord, Nico1, van den Elst, Hans1, van der Marel, Gijsbert A.1, Brouwer, Jaap2, Di Marzo, Vincenzo3, Overkleeft, Herman S.1, van der Stelt, Mario1 m.van.der.stelt@chem.leidenuniv.nl |
| Source: | Angewandte Chemie. Nov2013, Vol. 125 Issue 46, p12303-12307. 5p. |
| Database: | Academic Search Ultimate |
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| Header | DbId: asn DbLabel: Academic Search Ultimate An: 91899252 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=asn&AN=91899252 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1002/ange.201306295 Languages: – Code: eng Text: English PhysicalDescription: Pagination: PageCount: 5 StartPage: 12303 Titles: – TitleFull: Development of an Activity-Based Probe and In Silico Design Reveal Highly Selective Inhibitors for Diacylglycerol Lipase-α in Brain. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Baggelaar, Marc P. – PersonEntity: Name: NameFull: Janssen, Freek J. – PersonEntity: Name: NameFull: van Esbroeck, Annelot C. M. – PersonEntity: Name: NameFull: den Dulk, Hans – PersonEntity: Name: NameFull: Allarà, Marco – PersonEntity: Name: NameFull: Hoogendoorn, Sascha – PersonEntity: Name: NameFull: McGuire, Ross – PersonEntity: Name: NameFull: Florea, Bogdan I. – PersonEntity: Name: NameFull: Meeuwenoord, Nico – PersonEntity: Name: NameFull: van den Elst, Hans – PersonEntity: Name: NameFull: van der Marel, Gijsbert A. – PersonEntity: Name: NameFull: Brouwer, Jaap – PersonEntity: Name: NameFull: Di Marzo, Vincenzo – PersonEntity: Name: NameFull: Overkleeft, Herman S. – PersonEntity: Name: NameFull: van der Stelt, Mario IsPartOfRelationships: – BibEntity: Dates: – D: 11 M: 11 Text: Nov2013 Type: published Y: 2013 Identifiers: – Type: issn-print Value: 00448249 Numbering: – Type: volume Value: 125 – Type: issue Value: 46 Titles: – TitleFull: Angewandte Chemie Type: main |
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