Cu-Catalyzed Aerobic Oxidative Cyclization of Guanidylpyridines and Derivatives.
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| Title: | Cu-Catalyzed Aerobic Oxidative Cyclization of Guanidylpyridines and Derivatives. |
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| Authors: | Bartels, Björn1 bjoern.bartels@roche.com, Bolas, Conor Gordon1, Cueni, Philipp1, Fantasia, Serena2 serena_maria.fantasia@roche.com, Gaeng, Nicolas1, Trita, Andrada Stefania2 |
| Source: | Journal of Organic Chemistry. 1/16/2015, Vol. 80 Issue 2, p1249-1257. 9p. |
| Subjects: | Copper research, Metals, Pyridine, Heterocyclic compounds, 2-Mercaptopyridine |
| Abstract: | A new method for the straightforward synthesis of 2-amino-[1,2,4]triazolo[1,5-a]pyridines and derivatives is presented. The target products are synthesized in high yields from guanidylpyridines and analogues via copper-catalyzed N-N coupling. The present methodology shows a wide scope, tolerating not only different substituents on the pyridine ring but also different heterocylic rings such as pyrazines, pyrimidines, and pyridazines. [ABSTRACT FROM AUTHOR] |
| Copyright of Journal of Organic Chemistry is the property of American Chemical Society and its content may not be copied or emailed to multiple sites without the copyright holder's express written permission. Additionally, content may not be used with any artificial intelligence tools or machine learning technologies. However, users may print, download, or email articles for individual use. This abstract may be abridged. No warranty is given about the accuracy of the copy. Users should refer to the original published version of the material for the full abstract. (Copyright applies to all Abstracts.) | |
| Database: | Engineering Source |
| FullText | Text: Availability: 0 |
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| Header | DbId: egs DbLabel: Engineering Source An: 101085423 AccessLevel: 6 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Cu-Catalyzed Aerobic Oxidative Cyclization of Guanidylpyridines and Derivatives. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AR" term="%22Bartels%2C+Björn%22">Bartels, Björn</searchLink><relatesTo>1</relatesTo><i> bjoern.bartels@roche.com</i><br /><searchLink fieldCode="AR" term="%22Bolas%2C+Conor+Gordon%22">Bolas, Conor Gordon</searchLink><relatesTo>1</relatesTo><br /><searchLink fieldCode="AR" term="%22Cueni%2C+Philipp%22">Cueni, Philipp</searchLink><relatesTo>1</relatesTo><br /><searchLink fieldCode="AR" term="%22Fantasia%2C+Serena%22">Fantasia, Serena</searchLink><relatesTo>2</relatesTo><i> serena_maria.fantasia@roche.com</i><br /><searchLink fieldCode="AR" term="%22Gaeng%2C+Nicolas%22">Gaeng, Nicolas</searchLink><relatesTo>1</relatesTo><br /><searchLink fieldCode="AR" term="%22Trita%2C+Andrada+Stefania%22">Trita, Andrada Stefania</searchLink><relatesTo>2</relatesTo> – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%22Journal+of+Organic+Chemistry%22">Journal of Organic Chemistry</searchLink>. 1/16/2015, Vol. 80 Issue 2, p1249-1257. 9p. – Name: Subject Label: Subjects Group: Su Data: <searchLink fieldCode="DE" term="%22Copper+research%22">Copper research</searchLink><br /><searchLink fieldCode="DE" term="%22Metals%22">Metals</searchLink><br /><searchLink fieldCode="DE" term="%22Pyridine%22">Pyridine</searchLink><br /><searchLink fieldCode="DE" term="%22Heterocyclic+compounds%22">Heterocyclic compounds</searchLink><br /><searchLink fieldCode="DE" term="%222-Mercaptopyridine%22">2-Mercaptopyridine</searchLink> – Name: Abstract Label: Abstract Group: Ab Data: A new method for the straightforward synthesis of 2-amino-[1,2,4]triazolo[1,5-a]pyridines and derivatives is presented. The target products are synthesized in high yields from guanidylpyridines and analogues via copper-catalyzed N-N coupling. The present methodology shows a wide scope, tolerating not only different substituents on the pyridine ring but also different heterocylic rings such as pyrazines, pyrimidines, and pyridazines. [ABSTRACT FROM AUTHOR] – Name: AbstractSuppliedCopyright Label: Group: Ab Data: <i>Copyright of Journal of Organic Chemistry is the property of American Chemical Society and its content may not be copied or emailed to multiple sites without the copyright holder's express written permission. Additionally, content may not be used with any artificial intelligence tools or machine learning technologies. However, users may print, download, or email articles for individual use. This abstract may be abridged. No warranty is given about the accuracy of the copy. Users should refer to the original published version of the material for the full abstract.</i> (Copyright applies to all Abstracts.) |
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| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1021/jo502536t Languages: – Code: eng Text: English PhysicalDescription: Pagination: PageCount: 9 StartPage: 1249 Subjects: – SubjectFull: Copper research Type: general – SubjectFull: Metals Type: general – SubjectFull: Pyridine Type: general – SubjectFull: Heterocyclic compounds Type: general – SubjectFull: 2-Mercaptopyridine Type: general Titles: – TitleFull: Cu-Catalyzed Aerobic Oxidative Cyclization of Guanidylpyridines and Derivatives. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Bartels, Björn – PersonEntity: Name: NameFull: Bolas, Conor Gordon – PersonEntity: Name: NameFull: Cueni, Philipp – PersonEntity: Name: NameFull: Fantasia, Serena – PersonEntity: Name: NameFull: Gaeng, Nicolas – PersonEntity: Name: NameFull: Trita, Andrada Stefania IsPartOfRelationships: – BibEntity: Dates: – D: 16 M: 01 Text: 1/16/2015 Type: published Y: 2015 Identifiers: – Type: issn-print Value: 00223263 Numbering: – Type: volume Value: 80 – Type: issue Value: 2 Titles: – TitleFull: Journal of Organic Chemistry Type: main |
| ResultId | 1 |
