Structure based design of a series of potent and selective non peptidic PTP-1B inhibitors.

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Title: Structure based design of a series of potent and selective non peptidic PTP-1B inhibitors.
Authors: Lau CK; Department of Medicinal Chemistry, Merck Frosst Centre for Therapeutic Research, PO Box 1005, Pointe Claire-Dorval, Quebec H9R 4P8, Canada. lau@merck.com, Bayly CI, Gauthier JY, Li CS, Therien M, Asante-Appiah E, Cromlish W, Boie Y, Forghani F, Desmarais S, Wang Q, Skorey K, Waddleton D, Payette P, Ramachandran C, Kennedy BP, Scapin G
Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2004 Feb 23; Vol. 14 (4), pp. 1043-8.
Publication Type: Journal Article
Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print Cited Medium: Print ISSN: 0960-894X (Print) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: Structure based design of a series of potent and selective non peptidic PTP-1B inhibitors.
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  Data: <searchLink fieldCode="AU" term="%22Lau+CK%22">Lau CK</searchLink>; Department of Medicinal Chemistry, Merck Frosst Centre for Therapeutic Research, PO Box 1005, Pointe Claire-Dorval, Quebec H9R 4P8, Canada. lau@merck.com<br /><searchLink fieldCode="AU" term="%22Bayly+CI%22">Bayly CI</searchLink><br /><searchLink fieldCode="AU" term="%22Gauthier+JY%22">Gauthier JY</searchLink><br /><searchLink fieldCode="AU" term="%22Li+CS%22">Li CS</searchLink><br /><searchLink fieldCode="AU" term="%22Therien+M%22">Therien M</searchLink><br /><searchLink fieldCode="AU" term="%22Asante-Appiah+E%22">Asante-Appiah E</searchLink><br /><searchLink fieldCode="AU" term="%22Cromlish+W%22">Cromlish W</searchLink><br /><searchLink fieldCode="AU" term="%22Boie+Y%22">Boie Y</searchLink><br /><searchLink fieldCode="AU" term="%22Forghani+F%22">Forghani F</searchLink><br /><searchLink fieldCode="AU" term="%22Desmarais+S%22">Desmarais S</searchLink><br /><searchLink fieldCode="AU" term="%22Wang+Q%22">Wang Q</searchLink><br /><searchLink fieldCode="AU" term="%22Skorey+K%22">Skorey K</searchLink><br /><searchLink fieldCode="AU" term="%22Waddleton+D%22">Waddleton D</searchLink><br /><searchLink fieldCode="AU" term="%22Payette+P%22">Payette P</searchLink><br /><searchLink fieldCode="AU" term="%22Ramachandran+C%22">Ramachandran C</searchLink><br /><searchLink fieldCode="AU" term="%22Kennedy+BP%22">Kennedy BP</searchLink><br /><searchLink fieldCode="AU" term="%22Scapin+G%22">Scapin G</searchLink>
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        Value: 10.1016/j.bmcl.2003.11.076
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        Text: English
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              Text: 2004 Feb 23
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