The discovery and optimization of pyrimidinone-containing MCH R1 antagonists.

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Title: The discovery and optimization of pyrimidinone-containing MCH R1 antagonists.
Authors: Hertzog DL; Metabolic and Viral Diseases Centre of Excellence for Drug Discovery, GlaxoSmithKline, Five Moore Drive, Research Triangle Park, NC 27707, USA. Donald.L.Hertzog@gsk.com, Al-Barazanji KA, Bigham EC, Bishop MJ, Britt CS, Carlton DL, Cooper JP, Daniels AJ, Garrido DM, Goetz AS, Grizzle MK, Guo YC, Handlon AL, Ignar DM, Morgan RO, Peat AJ, Tavares FX, Zhou H
Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2006 Sep 15; Vol. 16 (18), pp. 4723-7. Date of Electronic Publication: 2006 Jul 25.
Publication Type: Journal Article
Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Print ISSN: 0960-894X (Print) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE
Database: MEDLINE Ultimate
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DbLabel: MEDLINE Ultimate
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PubType: Academic Journal
PubTypeId: academicJournal
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  Data: The discovery and optimization of pyrimidinone-containing MCH R1 antagonists.
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  Data: <searchLink fieldCode="AU" term="%22Hertzog+DL%22">Hertzog DL</searchLink>; Metabolic and Viral Diseases Centre of Excellence for Drug Discovery, GlaxoSmithKline, Five Moore Drive, Research Triangle Park, NC 27707, USA. Donald.L.Hertzog@gsk.com<br /><searchLink fieldCode="AU" term="%22Al-Barazanji+KA%22">Al-Barazanji KA</searchLink><br /><searchLink fieldCode="AU" term="%22Bigham+EC%22">Bigham EC</searchLink><br /><searchLink fieldCode="AU" term="%22Bishop+MJ%22">Bishop MJ</searchLink><br /><searchLink fieldCode="AU" term="%22Britt+CS%22">Britt CS</searchLink><br /><searchLink fieldCode="AU" term="%22Carlton+DL%22">Carlton DL</searchLink><br /><searchLink fieldCode="AU" term="%22Cooper+JP%22">Cooper JP</searchLink><br /><searchLink fieldCode="AU" term="%22Daniels+AJ%22">Daniels AJ</searchLink><br /><searchLink fieldCode="AU" term="%22Garrido+DM%22">Garrido DM</searchLink><br /><searchLink fieldCode="AU" term="%22Goetz+AS%22">Goetz AS</searchLink><br /><searchLink fieldCode="AU" term="%22Grizzle+MK%22">Grizzle MK</searchLink><br /><searchLink fieldCode="AU" term="%22Guo+YC%22">Guo YC</searchLink><br /><searchLink fieldCode="AU" term="%22Handlon+AL%22">Handlon AL</searchLink><br /><searchLink fieldCode="AU" term="%22Ignar+DM%22">Ignar DM</searchLink><br /><searchLink fieldCode="AU" term="%22Morgan+RO%22">Morgan RO</searchLink><br /><searchLink fieldCode="AU" term="%22Peat+AJ%22">Peat AJ</searchLink><br /><searchLink fieldCode="AU" term="%22Tavares+FX%22">Tavares FX</searchLink><br /><searchLink fieldCode="AU" term="%22Zhou+H%22">Zhou H</searchLink>
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Elsevier+Science+Ltd%22">Elsevier Science Ltd </searchLink><i>Country of Publication: </i>England <i>NLM ID: </i>9107377 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Print <i>ISSN: </i>0960-894X (Print) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%220960894X%22">0960894X </searchLink><i>NLM ISO Abbreviation: </i>Bioorg Med Chem Lett <i>Subsets: </i>MEDLINE
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        Value: 10.1016/j.bmcl.2006.07.008
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        Text: English
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              Text: 2006 Sep 15
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