Identification of 2-(4,5,6,7-tetrahydro-1H-pyrrolo[3,2-c]pyridin-3-yl)-ethylamine derivatives as novel GnRH receptor antagonists.

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Title: Identification of 2-(4,5,6,7-tetrahydro-1H-pyrrolo[3,2-c]pyridin-3-yl)-ethylamine derivatives as novel GnRH receptor antagonists.
Authors: Chen M; Department of Medicinal Chemistry, Neurocrine Biosciences, Inc., 12790 El Camino Real, San Diego, CA 92130, USA., Guo Z, Lanier MC, Zhao L, Betz SF, Huang CQ, Loweth CJ, Ashweek NJ, Liu XJ, Struthers RS, Bradbury MJ, Behan JW, Wen J, O'Brien Z, Saunders J, Zhu YF
Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2007 Jul 15; Vol. 17 (14), pp. 3845-50. Date of Electronic Publication: 2007 May 10.
Publication Type: Journal Article
Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Print ISSN: 0960-894X (Print) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE
Database: MEDLINE Ultimate
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PubType: Academic Journal
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  Data: Identification of 2-(4,5,6,7-tetrahydro-1H-pyrrolo[3,2-c]pyridin-3-yl)-ethylamine derivatives as novel GnRH receptor antagonists.
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  Data: <searchLink fieldCode="AU" term="%22Chen+M%22">Chen M</searchLink>; Department of Medicinal Chemistry, Neurocrine Biosciences, Inc., 12790 El Camino Real, San Diego, CA 92130, USA.<br /><searchLink fieldCode="AU" term="%22Guo+Z%22">Guo Z</searchLink><br /><searchLink fieldCode="AU" term="%22Lanier+MC%22">Lanier MC</searchLink><br /><searchLink fieldCode="AU" term="%22Zhao+L%22">Zhao L</searchLink><br /><searchLink fieldCode="AU" term="%22Betz+SF%22">Betz SF</searchLink><br /><searchLink fieldCode="AU" term="%22Huang+CQ%22">Huang CQ</searchLink><br /><searchLink fieldCode="AU" term="%22Loweth+CJ%22">Loweth CJ</searchLink><br /><searchLink fieldCode="AU" term="%22Ashweek+NJ%22">Ashweek NJ</searchLink><br /><searchLink fieldCode="AU" term="%22Liu+XJ%22">Liu XJ</searchLink><br /><searchLink fieldCode="AU" term="%22Struthers+RS%22">Struthers RS</searchLink><br /><searchLink fieldCode="AU" term="%22Bradbury+MJ%22">Bradbury MJ</searchLink><br /><searchLink fieldCode="AU" term="%22Behan+JW%22">Behan JW</searchLink><br /><searchLink fieldCode="AU" term="%22Wen+J%22">Wen J</searchLink><br /><searchLink fieldCode="AU" term="%22O'Brien+Z%22">O'Brien Z</searchLink><br /><searchLink fieldCode="AU" term="%22Saunders+J%22">Saunders J</searchLink><br /><searchLink fieldCode="AU" term="%22Zhu+YF%22">Zhu YF</searchLink>
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              Text: 2007 Jul 15
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