Discovery of the first known small-molecule inhibitors of heme-regulated eukaryotic initiation factor 2alpha (HRI) kinase.
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| Title: | Discovery of the first known small-molecule inhibitors of heme-regulated eukaryotic initiation factor 2alpha (HRI) kinase. |
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| Authors: | Rosen MD; Johnson & Johnson Pharmaceutical Research and Development, LLC, San Diego, CA 92121, United States. mrosen1@its.jnj.com, Woods CR, Goldberg SD, Hack MD, Bounds AD, Yang Y, Wagaman PC, Phuong VK, Ameriks AP, Barrett TD, Kanelakis KC, Chuang JC, Shankley NP, Rabinowitz MH |
| Source: | Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2009 Dec 01; Vol. 19 (23), pp. 6548-51. Date of Electronic Publication: 2009 Oct 13. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 19854648 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Discovery of the first known small-molecule inhibitors of heme-regulated eukaryotic initiation factor 2alpha (HRI) kinase. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Rosen+MD%22">Rosen MD</searchLink>; Johnson & Johnson Pharmaceutical Research and Development, LLC, San Diego, CA 92121, United States. mrosen1@its.jnj.com<br /><searchLink fieldCode="AU" term="%22Woods+CR%22">Woods CR</searchLink><br /><searchLink fieldCode="AU" term="%22Goldberg+SD%22">Goldberg SD</searchLink><br /><searchLink fieldCode="AU" term="%22Hack+MD%22">Hack MD</searchLink><br /><searchLink fieldCode="AU" term="%22Bounds+AD%22">Bounds AD</searchLink><br /><searchLink fieldCode="AU" term="%22Yang+Y%22">Yang Y</searchLink><br /><searchLink fieldCode="AU" term="%22Wagaman+PC%22">Wagaman PC</searchLink><br /><searchLink fieldCode="AU" term="%22Phuong+VK%22">Phuong VK</searchLink><br /><searchLink fieldCode="AU" term="%22Ameriks+AP%22">Ameriks AP</searchLink><br /><searchLink fieldCode="AU" term="%22Barrett+TD%22">Barrett TD</searchLink><br /><searchLink fieldCode="AU" term="%22Kanelakis+KC%22">Kanelakis KC</searchLink><br /><searchLink fieldCode="AU" term="%22Chuang+JC%22">Chuang JC</searchLink><br /><searchLink fieldCode="AU" term="%22Shankley+NP%22">Shankley NP</searchLink><br /><searchLink fieldCode="AU" term="%22Rabinowitz+MH%22">Rabinowitz MH</searchLink> – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%229107377%22">Bioorganic & medicinal chemistry letters</searchLink> [Bioorg Med Chem Lett] 2009 Dec 01; Vol. 19 (23), pp. 6548-51. <i>Date of Electronic Publication: </i>2009 Oct 13. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Elsevier+Science+Ltd%22">Elsevier Science Ltd </searchLink><i>Country of Publication: </i>England <i>NLM ID: </i>9107377 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1464-3405 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%220960894X%22">0960894X </searchLink><i>NLM ISO Abbreviation: </i>Bioorg Med Chem Lett <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=19854648 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1016/j.bmcl.2009.10.033 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 6548 Titles: – TitleFull: Discovery of the first known small-molecule inhibitors of heme-regulated eukaryotic initiation factor 2alpha (HRI) kinase. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Rosen MD – PersonEntity: Name: NameFull: Woods CR – PersonEntity: Name: NameFull: Goldberg SD – PersonEntity: Name: NameFull: Hack MD – PersonEntity: Name: NameFull: Bounds AD – PersonEntity: Name: NameFull: Yang Y – PersonEntity: Name: NameFull: Wagaman PC – PersonEntity: Name: NameFull: Phuong VK – PersonEntity: Name: NameFull: Ameriks AP – PersonEntity: Name: NameFull: Barrett TD – PersonEntity: Name: NameFull: Kanelakis KC – PersonEntity: Name: NameFull: Chuang JC – PersonEntity: Name: NameFull: Shankley NP – PersonEntity: Name: NameFull: Rabinowitz MH IsPartOfRelationships: – BibEntity: Dates: – D: 01 M: 12 Text: 2009 Dec 01 Type: published Y: 2009 Identifiers: – Type: issn-electronic Value: 1464-3405 Numbering: – Type: volume Value: 19 – Type: issue Value: 23 Titles: – TitleFull: Bioorganic & medicinal chemistry letters Type: main |
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