Discovery of the first known small-molecule inhibitors of heme-regulated eukaryotic initiation factor 2alpha (HRI) kinase.

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Title: Discovery of the first known small-molecule inhibitors of heme-regulated eukaryotic initiation factor 2alpha (HRI) kinase.
Authors: Rosen MD; Johnson & Johnson Pharmaceutical Research and Development, LLC, San Diego, CA 92121, United States. mrosen1@its.jnj.com, Woods CR, Goldberg SD, Hack MD, Bounds AD, Yang Y, Wagaman PC, Phuong VK, Ameriks AP, Barrett TD, Kanelakis KC, Chuang JC, Shankley NP, Rabinowitz MH
Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2009 Dec 01; Vol. 19 (23), pp. 6548-51. Date of Electronic Publication: 2009 Oct 13.
Publication Type: Journal Article
Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE
Database: MEDLINE Ultimate
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PubType: Academic Journal
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  Data: Discovery of the first known small-molecule inhibitors of heme-regulated eukaryotic initiation factor 2alpha (HRI) kinase.
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  Data: <searchLink fieldCode="AU" term="%22Rosen+MD%22">Rosen MD</searchLink>; Johnson & Johnson Pharmaceutical Research and Development, LLC, San Diego, CA 92121, United States. mrosen1@its.jnj.com<br /><searchLink fieldCode="AU" term="%22Woods+CR%22">Woods CR</searchLink><br /><searchLink fieldCode="AU" term="%22Goldberg+SD%22">Goldberg SD</searchLink><br /><searchLink fieldCode="AU" term="%22Hack+MD%22">Hack MD</searchLink><br /><searchLink fieldCode="AU" term="%22Bounds+AD%22">Bounds AD</searchLink><br /><searchLink fieldCode="AU" term="%22Yang+Y%22">Yang Y</searchLink><br /><searchLink fieldCode="AU" term="%22Wagaman+PC%22">Wagaman PC</searchLink><br /><searchLink fieldCode="AU" term="%22Phuong+VK%22">Phuong VK</searchLink><br /><searchLink fieldCode="AU" term="%22Ameriks+AP%22">Ameriks AP</searchLink><br /><searchLink fieldCode="AU" term="%22Barrett+TD%22">Barrett TD</searchLink><br /><searchLink fieldCode="AU" term="%22Kanelakis+KC%22">Kanelakis KC</searchLink><br /><searchLink fieldCode="AU" term="%22Chuang+JC%22">Chuang JC</searchLink><br /><searchLink fieldCode="AU" term="%22Shankley+NP%22">Shankley NP</searchLink><br /><searchLink fieldCode="AU" term="%22Rabinowitz+MH%22">Rabinowitz MH</searchLink>
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  Data: <searchLink fieldCode="JN" term="%229107377%22">Bioorganic & medicinal chemistry letters</searchLink> [Bioorg Med Chem Lett] 2009 Dec 01; Vol. 19 (23), pp. 6548-51. <i>Date of Electronic Publication: </i>2009 Oct 13.
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Elsevier+Science+Ltd%22">Elsevier Science Ltd </searchLink><i>Country of Publication: </i>England <i>NLM ID: </i>9107377 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1464-3405 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%220960894X%22">0960894X </searchLink><i>NLM ISO Abbreviation: </i>Bioorg Med Chem Lett <i>Subsets: </i>MEDLINE
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        Value: 10.1016/j.bmcl.2009.10.033
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              Text: 2009 Dec 01
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