Fragment-based lead discovery: screening and optimizing fragments for thermolysin inhibition.

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Title: Fragment-based lead discovery: screening and optimizing fragments for thermolysin inhibition.
Authors: Englert L; Philipps-Universität Marburg, Institut für Pharmazeutische Chemie, Marbacher Weg 6, 35032 Marburg, Germany., Silber K, Steuber H, Brass S, Over B, Gerber HD, Heine A, Diederich WE, Klebe G
Source: ChemMedChem [ChemMedChem] 2010 Jun 07; Vol. 5 (6), pp. 930-40.
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
Journal Info: Publisher: Wiley-VCH Country of Publication: Germany NLM ID: 101259013 Publication Model: Print Cited Medium: Internet ISSN: 1860-7187 (Electronic) Linking ISSN: 18607179 NLM ISO Abbreviation: ChemMedChem Subsets: MEDLINE
Database: MEDLINE Ultimate
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DbLabel: MEDLINE Ultimate
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AccessLevel: 2
PubType: Academic Journal
PubTypeId: academicJournal
PreciseRelevancyScore: 0
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  Data: Fragment-based lead discovery: screening and optimizing fragments for thermolysin inhibition.
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  Data: <searchLink fieldCode="AU" term="%22Englert+L%22">Englert L</searchLink>; Philipps-Universität Marburg, Institut für Pharmazeutische Chemie, Marbacher Weg 6, 35032 Marburg, Germany.<br /><searchLink fieldCode="AU" term="%22Silber+K%22">Silber K</searchLink><br /><searchLink fieldCode="AU" term="%22Steuber+H%22">Steuber H</searchLink><br /><searchLink fieldCode="AU" term="%22Brass+S%22">Brass S</searchLink><br /><searchLink fieldCode="AU" term="%22Over+B%22">Over B</searchLink><br /><searchLink fieldCode="AU" term="%22Gerber+HD%22">Gerber HD</searchLink><br /><searchLink fieldCode="AU" term="%22Heine+A%22">Heine A</searchLink><br /><searchLink fieldCode="AU" term="%22Diederich+WE%22">Diederich WE</searchLink><br /><searchLink fieldCode="AU" term="%22Klebe+G%22">Klebe G</searchLink>
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  Data: <searchLink fieldCode="JN" term="%22101259013%22">ChemMedChem</searchLink> [ChemMedChem] 2010 Jun 07; Vol. 5 (6), pp. 930-40.
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  Data: Journal Article; Research Support, Non-U.S. Gov't
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Wiley-VCH%22">Wiley-VCH </searchLink><i>Country of Publication: </i>Germany <i>NLM ID: </i>101259013 <i>Publication Model: </i>Print <i>Cited Medium: </i>Internet <i>ISSN: </i>1860-7187 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2218607179%22">18607179 </searchLink><i>NLM ISO Abbreviation: </i>ChemMedChem <i>Subsets: </i>MEDLINE
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        Value: 10.1002/cmdc.201000084
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      – Code: eng
        Text: English
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        StartPage: 930
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      – TitleFull: Fragment-based lead discovery: screening and optimizing fragments for thermolysin inhibition.
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            NameFull: Englert L
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            NameFull: Silber K
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            NameFull: Steuber H
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            NameFull: Brass S
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            – D: 07
              M: 06
              Text: 2010 Jun 07
              Type: published
              Y: 2010
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              Value: 1860-7187
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              Value: 5
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              Value: 6
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