Discovery of pyrazolo[1,5-a]pyrimidine-based CHK1 inhibitors: a template-based approach--part 2.
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| Title: | Discovery of pyrazolo[1,5-a]pyrimidine-based CHK1 inhibitors: a template-based approach--part 2. |
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| Authors: | Labroli M; Merck Research Laboratories, 2015 Galloping Hill Road, Kenilworth, NJ 07033, United States. marc.labroli@merck.com, Paruch K, Dwyer MP, Alvarez C, Keertikar K, Poker C, Rossman R, Duca JS, Fischmann TO, Madison V, Parry D, Davis N, Seghezzi W, Wiswell D, Guzi TJ |
| Source: | Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2011 Jan 01; Vol. 21 (1), pp. 471-4. Date of Electronic Publication: 2010 Oct 28. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 21094607 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Discovery of pyrazolo[1,5-a]pyrimidine-based CHK1 inhibitors: a template-based approach--part 2. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Labroli+M%22">Labroli M</searchLink>; Merck Research Laboratories, 2015 Galloping Hill Road, Kenilworth, NJ 07033, United States. marc.labroli@merck.com<br /><searchLink fieldCode="AU" term="%22Paruch+K%22">Paruch K</searchLink><br /><searchLink fieldCode="AU" term="%22Dwyer+MP%22">Dwyer MP</searchLink><br /><searchLink fieldCode="AU" term="%22Alvarez+C%22">Alvarez C</searchLink><br /><searchLink fieldCode="AU" term="%22Keertikar+K%22">Keertikar K</searchLink><br /><searchLink fieldCode="AU" term="%22Poker+C%22">Poker C</searchLink><br /><searchLink fieldCode="AU" term="%22Rossman+R%22">Rossman R</searchLink><br /><searchLink fieldCode="AU" term="%22Duca+JS%22">Duca JS</searchLink><br /><searchLink fieldCode="AU" term="%22Fischmann+TO%22">Fischmann TO</searchLink><br /><searchLink fieldCode="AU" term="%22Madison+V%22">Madison V</searchLink><br /><searchLink fieldCode="AU" term="%22Parry+D%22">Parry D</searchLink><br /><searchLink fieldCode="AU" term="%22Davis+N%22">Davis N</searchLink><br /><searchLink fieldCode="AU" term="%22Seghezzi+W%22">Seghezzi W</searchLink><br /><searchLink fieldCode="AU" term="%22Wiswell+D%22">Wiswell D</searchLink><br /><searchLink fieldCode="AU" term="%22Guzi+TJ%22">Guzi TJ</searchLink> – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%229107377%22">Bioorganic & medicinal chemistry letters</searchLink> [Bioorg Med Chem Lett] 2011 Jan 01; Vol. 21 (1), pp. 471-4. <i>Date of Electronic Publication: </i>2010 Oct 28. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Elsevier+Science+Ltd%22">Elsevier Science Ltd </searchLink><i>Country of Publication: </i>England <i>NLM ID: </i>9107377 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1464-3405 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%220960894X%22">0960894X </searchLink><i>NLM ISO Abbreviation: </i>Bioorg Med Chem Lett <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=21094607 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1016/j.bmcl.2010.10.114 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 471 Titles: – TitleFull: Discovery of pyrazolo[1,5-a]pyrimidine-based CHK1 inhibitors: a template-based approach--part 2. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Labroli M – PersonEntity: Name: NameFull: Paruch K – PersonEntity: Name: NameFull: Dwyer MP – PersonEntity: Name: NameFull: Alvarez C – PersonEntity: Name: NameFull: Keertikar K – PersonEntity: Name: NameFull: Poker C – PersonEntity: Name: NameFull: Rossman R – PersonEntity: Name: NameFull: Duca JS – PersonEntity: Name: NameFull: Fischmann TO – PersonEntity: Name: NameFull: Madison V – PersonEntity: Name: NameFull: Parry D – PersonEntity: Name: NameFull: Davis N – PersonEntity: Name: NameFull: Seghezzi W – PersonEntity: Name: NameFull: Wiswell D – PersonEntity: Name: NameFull: Guzi TJ IsPartOfRelationships: – BibEntity: Dates: – D: 01 M: 01 Text: 2011 Jan 01 Type: published Y: 2011 Identifiers: – Type: issn-electronic Value: 1464-3405 Numbering: – Type: volume Value: 21 – Type: issue Value: 1 Titles: – TitleFull: Bioorganic & medicinal chemistry letters Type: main |
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