Discovery of pyrazolo[1,5-a]pyrimidine-based Pim inhibitors: a template-based approach.

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Title: Discovery of pyrazolo[1,5-a]pyrimidine-based Pim inhibitors: a template-based approach.
Authors: Dwyer MP; Department of Chemical Research, Merck Research Laboratories, 2015 Galloping Hill Road, Kenilworth, NJ 07033, United States. Electronic address: michael.dwyer@merck.com., Keertikar K, Paruch K, Alvarez C, Labroli M, Poker C, Fischmann TO, Mayer-Ezell R, Bond R, Wang Y, Azevedo R, Guzi TJ
Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2013 Nov 15; Vol. 23 (22), pp. 6178-82. Date of Electronic Publication: 2013 Sep 07.
Publication Type: Journal Article
Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: Discovery of pyrazolo[1,5-a]pyrimidine-based Pim inhibitors: a template-based approach.
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  Data: <searchLink fieldCode="AU" term="%22Dwyer+MP%22">Dwyer MP</searchLink>; Department of Chemical Research, Merck Research Laboratories, 2015 Galloping Hill Road, Kenilworth, NJ 07033, United States. Electronic address: michael.dwyer@merck.com.<br /><searchLink fieldCode="AU" term="%22Keertikar+K%22">Keertikar K</searchLink><br /><searchLink fieldCode="AU" term="%22Paruch+K%22">Paruch K</searchLink><br /><searchLink fieldCode="AU" term="%22Alvarez+C%22">Alvarez C</searchLink><br /><searchLink fieldCode="AU" term="%22Labroli+M%22">Labroli M</searchLink><br /><searchLink fieldCode="AU" term="%22Poker+C%22">Poker C</searchLink><br /><searchLink fieldCode="AU" term="%22Fischmann+TO%22">Fischmann TO</searchLink><br /><searchLink fieldCode="AU" term="%22Mayer-Ezell+R%22">Mayer-Ezell R</searchLink><br /><searchLink fieldCode="AU" term="%22Bond+R%22">Bond R</searchLink><br /><searchLink fieldCode="AU" term="%22Wang+Y%22">Wang Y</searchLink><br /><searchLink fieldCode="AU" term="%22Azevedo+R%22">Azevedo R</searchLink><br /><searchLink fieldCode="AU" term="%22Guzi+TJ%22">Guzi TJ</searchLink>
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  Data: <searchLink fieldCode="JN" term="%229107377%22">Bioorganic & medicinal chemistry letters</searchLink> [Bioorg Med Chem Lett] 2013 Nov 15; Vol. 23 (22), pp. 6178-82. <i>Date of Electronic Publication: </i>2013 Sep 07.
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