Discovery of pyrazolo[1,5-a]pyrimidine-based Pim inhibitors: a template-based approach.
Saved in:
| Title: | Discovery of pyrazolo[1,5-a]pyrimidine-based Pim inhibitors: a template-based approach. |
|---|---|
| Authors: | Dwyer MP; Department of Chemical Research, Merck Research Laboratories, 2015 Galloping Hill Road, Kenilworth, NJ 07033, United States. Electronic address: michael.dwyer@merck.com., Keertikar K, Paruch K, Alvarez C, Labroli M, Poker C, Fischmann TO, Mayer-Ezell R, Bond R, Wang Y, Azevedo R, Guzi TJ |
| Source: | Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2013 Nov 15; Vol. 23 (22), pp. 6178-82. Date of Electronic Publication: 2013 Sep 07. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
|---|---|
| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 24091081 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
| IllustrationInfo | |
| Items | – Name: Title Label: Title Group: Ti Data: Discovery of pyrazolo[1,5-a]pyrimidine-based Pim inhibitors: a template-based approach. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Dwyer+MP%22">Dwyer MP</searchLink>; Department of Chemical Research, Merck Research Laboratories, 2015 Galloping Hill Road, Kenilworth, NJ 07033, United States. Electronic address: michael.dwyer@merck.com.<br /><searchLink fieldCode="AU" term="%22Keertikar+K%22">Keertikar K</searchLink><br /><searchLink fieldCode="AU" term="%22Paruch+K%22">Paruch K</searchLink><br /><searchLink fieldCode="AU" term="%22Alvarez+C%22">Alvarez C</searchLink><br /><searchLink fieldCode="AU" term="%22Labroli+M%22">Labroli M</searchLink><br /><searchLink fieldCode="AU" term="%22Poker+C%22">Poker C</searchLink><br /><searchLink fieldCode="AU" term="%22Fischmann+TO%22">Fischmann TO</searchLink><br /><searchLink fieldCode="AU" term="%22Mayer-Ezell+R%22">Mayer-Ezell R</searchLink><br /><searchLink fieldCode="AU" term="%22Bond+R%22">Bond R</searchLink><br /><searchLink fieldCode="AU" term="%22Wang+Y%22">Wang Y</searchLink><br /><searchLink fieldCode="AU" term="%22Azevedo+R%22">Azevedo R</searchLink><br /><searchLink fieldCode="AU" term="%22Guzi+TJ%22">Guzi TJ</searchLink> – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%229107377%22">Bioorganic & medicinal chemistry letters</searchLink> [Bioorg Med Chem Lett] 2013 Nov 15; Vol. 23 (22), pp. 6178-82. <i>Date of Electronic Publication: </i>2013 Sep 07. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Elsevier+Science+Ltd%22">Elsevier Science Ltd </searchLink><i>Country of Publication: </i>England <i>NLM ID: </i>9107377 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1464-3405 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%220960894X%22">0960894X </searchLink><i>NLM ISO Abbreviation: </i>Bioorg Med Chem Lett <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=24091081 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1016/j.bmcl.2013.08.110 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 6178 Titles: – TitleFull: Discovery of pyrazolo[1,5-a]pyrimidine-based Pim inhibitors: a template-based approach. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Dwyer MP – PersonEntity: Name: NameFull: Keertikar K – PersonEntity: Name: NameFull: Paruch K – PersonEntity: Name: NameFull: Alvarez C – PersonEntity: Name: NameFull: Labroli M – PersonEntity: Name: NameFull: Poker C – PersonEntity: Name: NameFull: Fischmann TO – PersonEntity: Name: NameFull: Mayer-Ezell R – PersonEntity: Name: NameFull: Bond R – PersonEntity: Name: NameFull: Wang Y – PersonEntity: Name: NameFull: Azevedo R – PersonEntity: Name: NameFull: Guzi TJ IsPartOfRelationships: – BibEntity: Dates: – D: 15 M: 11 Text: 2013 Nov 15 Type: published Y: 2013 Identifiers: – Type: issn-electronic Value: 1464-3405 Numbering: – Type: volume Value: 23 – Type: issue Value: 22 Titles: – TitleFull: Bioorganic & medicinal chemistry letters Type: main |
| ResultId | 1 |