4-Bicyclic heteroaryl-piperidine derivatives as potent, orally bioavailable Stearoyl-CoA desaturase-1 (SCD1) inhibitors. Part 1: urea-based analogs.

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Title: 4-Bicyclic heteroaryl-piperidine derivatives as potent, orally bioavailable Stearoyl-CoA desaturase-1 (SCD1) inhibitors. Part 1: urea-based analogs.
Authors: Yang SM; Cardiovascular and Metabolism Research, Janssen Research and Development, LLC, Welsh & McKean Roads, Spring House, PA 19477, USA. Electronic address: shyhyang99@yahoo.com., Tang Y, Zhang R, Lu H, Kuo GH, Gaul MD, Li Y, Ho G, Conway JG, Liang Y, Lenhard JM, Demarest KT, Murray WV
Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2013 Dec 15; Vol. 23 (24), pp. 6773-6. Date of Electronic Publication: 2013 Oct 09.
Publication Type: Journal Article
Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: 4-Bicyclic heteroaryl-piperidine derivatives as potent, orally bioavailable Stearoyl-CoA desaturase-1 (SCD1) inhibitors. Part 1: urea-based analogs.
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  Data: <searchLink fieldCode="AU" term="%22Yang+SM%22">Yang SM</searchLink>; Cardiovascular and Metabolism Research, Janssen Research and Development, LLC, Welsh & McKean Roads, Spring House, PA 19477, USA. Electronic address: shyhyang99@yahoo.com.<br /><searchLink fieldCode="AU" term="%22Tang+Y%22">Tang Y</searchLink><br /><searchLink fieldCode="AU" term="%22Zhang+R%22">Zhang R</searchLink><br /><searchLink fieldCode="AU" term="%22Lu+H%22">Lu H</searchLink><br /><searchLink fieldCode="AU" term="%22Kuo+GH%22">Kuo GH</searchLink><br /><searchLink fieldCode="AU" term="%22Gaul+MD%22">Gaul MD</searchLink><br /><searchLink fieldCode="AU" term="%22Li+Y%22">Li Y</searchLink><br /><searchLink fieldCode="AU" term="%22Ho+G%22">Ho G</searchLink><br /><searchLink fieldCode="AU" term="%22Conway+JG%22">Conway JG</searchLink><br /><searchLink fieldCode="AU" term="%22Liang+Y%22">Liang Y</searchLink><br /><searchLink fieldCode="AU" term="%22Lenhard+JM%22">Lenhard JM</searchLink><br /><searchLink fieldCode="AU" term="%22Demarest+KT%22">Demarest KT</searchLink><br /><searchLink fieldCode="AU" term="%22Murray+WV%22">Murray WV</searchLink>
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  Data: <searchLink fieldCode="JN" term="%229107377%22">Bioorganic & medicinal chemistry letters</searchLink> [Bioorg Med Chem Lett] 2013 Dec 15; Vol. 23 (24), pp. 6773-6. <i>Date of Electronic Publication: </i>2013 Oct 09.
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              Text: 2013 Dec 15
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