Tafenoquine and NPC-1161B require CYP 2D metabolism for anti-malarial activity: implications for the 8-aminoquinoline class of anti-malarial compounds.

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Title: Tafenoquine and NPC-1161B require CYP 2D metabolism for anti-malarial activity: implications for the 8-aminoquinoline class of anti-malarial compounds.
Authors: Marcsisin SR; Division of Experimental Therapeutics, Military Malaria Research Program, Walter Reed Army Institute of Research, 503 Robert Grant Ave, Silver Spring, MD 20910, USA. sean.r.marcsisin.mil@mail.mil., Sousa JC, Reichard GA, Caridha D, Zeng Q, Roncal N, McNulty R, Careagabarja J, Sciotti RJ, Bennett JW, Zottig VE, Deye G, Li Q, Read L, Hickman M, Dhammika Nanayakkara NP, Walker LA, Smith B, Melendez V, Pybus BS
Source: Malaria journal [Malar J] 2014 Jan 03; Vol. 13, pp. 2. Date of Electronic Publication: 2014 Jan 03.
Publication Type: Journal Article
Journal Info: Publisher: BioMed Central Country of Publication: England NLM ID: 101139802 Publication Model: Electronic Cited Medium: Internet ISSN: 1475-2875 (Electronic) Linking ISSN: 14752875 NLM ISO Abbreviation: Malar J Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: Tafenoquine and NPC-1161B require CYP 2D metabolism for anti-malarial activity: implications for the 8-aminoquinoline class of anti-malarial compounds.
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  Data: <searchLink fieldCode="AU" term="%22Marcsisin+SR%22">Marcsisin SR</searchLink>; Division of Experimental Therapeutics, Military Malaria Research Program, Walter Reed Army Institute of Research, 503 Robert Grant Ave, Silver Spring, MD 20910, USA. sean.r.marcsisin.mil@mail.mil.<br /><searchLink fieldCode="AU" term="%22Sousa+JC%22">Sousa JC</searchLink><br /><searchLink fieldCode="AU" term="%22Reichard+GA%22">Reichard GA</searchLink><br /><searchLink fieldCode="AU" term="%22Caridha+D%22">Caridha D</searchLink><br /><searchLink fieldCode="AU" term="%22Zeng+Q%22">Zeng Q</searchLink><br /><searchLink fieldCode="AU" term="%22Roncal+N%22">Roncal N</searchLink><br /><searchLink fieldCode="AU" term="%22McNulty+R%22">McNulty R</searchLink><br /><searchLink fieldCode="AU" term="%22Careagabarja+J%22">Careagabarja J</searchLink><br /><searchLink fieldCode="AU" term="%22Sciotti+RJ%22">Sciotti RJ</searchLink><br /><searchLink fieldCode="AU" term="%22Bennett+JW%22">Bennett JW</searchLink><br /><searchLink fieldCode="AU" term="%22Zottig+VE%22">Zottig VE</searchLink><br /><searchLink fieldCode="AU" term="%22Deye+G%22">Deye G</searchLink><br /><searchLink fieldCode="AU" term="%22Li+Q%22">Li Q</searchLink><br /><searchLink fieldCode="AU" term="%22Read+L%22">Read L</searchLink><br /><searchLink fieldCode="AU" term="%22Hickman+M%22">Hickman M</searchLink><br /><searchLink fieldCode="AU" term="%22Dhammika+Nanayakkara+NP%22">Dhammika Nanayakkara NP</searchLink><br /><searchLink fieldCode="AU" term="%22Walker+LA%22">Walker LA</searchLink><br /><searchLink fieldCode="AU" term="%22Smith+B%22">Smith B</searchLink><br /><searchLink fieldCode="AU" term="%22Melendez+V%22">Melendez V</searchLink><br /><searchLink fieldCode="AU" term="%22Pybus+BS%22">Pybus BS</searchLink>
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  Data: <searchLink fieldCode="JN" term="%22101139802%22">Malaria journal</searchLink> [Malar J] 2014 Jan 03; Vol. 13, pp. 2. <i>Date of Electronic Publication: </i>2014 Jan 03.
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22BioMed+Central%22">BioMed Central </searchLink><i>Country of Publication: </i>England <i>NLM ID: </i>101139802 <i>Publication Model: </i>Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1475-2875 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2214752875%22">14752875 </searchLink><i>NLM ISO Abbreviation: </i>Malar J <i>Subsets: </i>MEDLINE
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